Zobrazeno 1 - 10
of 15
pro vyhledávání: '"František Zálešák"'
Autor:
Francesco Errani, Annalisa Invernizzi, Marcin Herok, Elena Bochenkova, Fiona Stamm, Ivan Corbeski, Valeria Romanucci, Giovanni Di Fabio, František Zálešák, Amedeo Caflisch
Publikováno v:
JACS Au, Vol 4, Iss 2, Pp 713-729 (2024)
Externí odkaz:
https://doaj.org/article/975b1b3506c844a881e52c14762605d6
Autor:
Yaozong Li, Rajiv Kumar Bedi, Francesco Nai, Valentin von Roten, Aymeric Dolbois, František Zálešák, Raed Nachawati, Danzhi Huang, Amedeo Caflisch
Publikováno v:
European Journal of Medicinal Chemistry Reports, Vol 5, Iss , Pp 100057- (2022)
We report new chemical entities for disrupting the interactions between N6-methyladenosine (m6A) mRNA and its reader YT521-B homology-domain-containing protein 1 (YTHDC1). High-throughput docking was used to screen commercially available databases of
Externí odkaz:
https://doaj.org/article/3173574e74c9400db4818b84271eb889
Publikováno v:
Molecules, Vol 24, Iss 19, p 3558 (2019)
A simple general synthesis of 1-aryl-6-azaisocytosine-5-carbonitriles 4 is described. This method is based on coupling diazonium salts with cyanoacetylcyanamide 2 and then cyclization of the formed 2-arylhydrazono-2-cyanoacetylcyanamides 3. The 6-aza
Externí odkaz:
https://doaj.org/article/c2d1298bb667440aba3e98dc778b17bf
Publikováno v:
ACS Medicinal Chemistry Letters. 13:1500-1509
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::39e14ed3209a4273cfebe9f5a6a0ff21
https://doi.org/10.1021/acsmedchemlett.2c00303
https://doi.org/10.1021/acsmedchemlett.2c00303
Publikováno v:
The Journal of Organic Chemistry. 86:11291-11309
In this paper, we report a unified approach to N-substituted and N,N-disubstituted benzothiazole (BT) sulfonamides. Our approach to BT-sulfonamides starts from simple commercially available building blocks (benzo[d]thiazole-2-thiol and primary and se
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::ec7e0ff8fb57f6f19dc49877f6626993
https://doi.org/10.1021/acs.joc.1c00317
https://doi.org/10.1021/acs.joc.1c00317
Autor:
Ondřej Kováč, David J.-Y.D. Bon, František Zálešák, Lukas Roiser, Lubomír Vojtěch Baar, Mario Waser, Jiri Pospisil
Publikováno v:
The Journal of Organic Chemistry. 85:7192-7206
In this paper, we report the formation of highly electrophilic 1,1-deactivated olefins, their use as novel synthetic building blocks, and their transformation to structurally diverse molecular scaf...
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::39e613deb53ff6f37b68c0e7e879f482
https://doi.org/10.1021/acs.joc.0c00571
https://doi.org/10.1021/acs.joc.0c00571
Autor:
Roman O. Iakovenko, Daniel Chrenko, Jozef Kristek, Eline Desmedt, František Zálešák, Freija De Vleeschouwer, Jiří Pospíšil
Publikováno v:
Organicbiomolecular chemistry. 20(15)
Heteroaryl sulfonamides are important structural motifs in the medicinal and agrochemical industries. However, their synthesis often relies on the use of heteroaryl sulfonyl chlorides, which are unstable and toxic reagents. Herein, we report a protoc
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::eba394d982d7333f6e253882ff37938f
https://pubmed.ncbi.nlm.nih.gov/35343994
https://pubmed.ncbi.nlm.nih.gov/35343994
Publikováno v:
The Journal of organic chemistry. 86(17)
In this paper, we report a unified approach to
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::132837503518d8e26d80314467785368
https://pubmed.ncbi.nlm.nih.gov/34479409
https://pubmed.ncbi.nlm.nih.gov/34479409
Publikováno v:
Monatshefte für Chemie - Chemical Monthly. 149:737-748
A novel approach to the neolignan-core skeletons of boehmenan natural products and to dehydrodiconiferyl alcohol glucosides based on the Fe(III)-promoted oxidative coupling has been achieved. Obtained common intermediates were further selectively mod
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::6467ef4c60d13eace34566e40599f3da
https://doi.org/10.1007/s00706-017-2132-4
https://doi.org/10.1007/s00706-017-2132-4
Publikováno v:
Molecules, Vol 24, Iss 19, p 3558 (2019)
Molecules
Volume 24
Issue 19
Molecules
Volume 24
Issue 19
A simple general synthesis of 1-aryl-6-azaisocytosine-5-carbonitriles 4 is described. This method is based on coupling diazonium salts with cyanoacetylcyanamide 2 and then cyclization of the formed 2-arylhydrazono-2-cyanoacetylcyanamides 3. The 6-aza
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a6a93b8ae783b6e8f503e39eeebe45b7
https://www.mdpi.com/1420-3049/24/19/3558
https://www.mdpi.com/1420-3049/24/19/3558