Zobrazeno 1 - 10
of 183
pro vyhledávání: '"Frans, Compernolle"'
Publikováno v:
ARKIVOC, Vol 2003, Iss 4, Pp 3-21 (2002)
Externí odkaz:
https://doaj.org/article/00161562a20a4669a455da1aee2511fa
Publikováno v:
Acta Crystallographica Section E, Vol 64, Iss 1, Pp m93-m93 (2008)
The title compound, [Pd(C12H10ClN2O2)Cl(C18H15P)2], is the intermediate of the reduction of a 3,5-dichloropyrazinone [Loosen, Tutonda, Khorasani, Compernolle & Hoornaert (1991). Tetrahedron, 47, 9259–9268]. This species is formed by oxidative addit
Externí odkaz:
https://doaj.org/article/26d2b9cab16b497aaf974636f26d0b6a
Autor:
Frans Compernolle, Wim Dehaen
Publikováno v:
ARKIVOC, Vol 2003, Iss 4, Pp 1-2 (2003)
Externí odkaz:
https://doaj.org/article/03919fa74e4b419a9a66f3077d6ab653
Autor:
Margriet Ovaere, Frans Compernolle, Jo Nelissen, Wim M. De Borggraeve, An Van den Bogaert, Luc Van Meervelt
Publikováno v:
European Journal of Organic Chemistry. 2010:5397-5401
Benzodiazepines show a broad spectrum of biological activities. In an ongoing effort to extend molecular diversity in this type of systems, we developed a strategy for synthesizing 3,4-dihydro-1H-pyrido[2,3-e][1,4]diazepine-2,5-dione compounds starti
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::09095092d06696ae9427d05977e1a36f
https://doi.org/10.1002/ejoc.201000549
https://doi.org/10.1002/ejoc.201000549
Publikováno v:
European Journal of Organic Chemistry. 2009:643-654
Derivatives of 6,8-bridged 5,6,7,8-tetrahydro-1,6-naphthyridines, designed as analogues of huperzine A, were synthesised and evaluated as inhibitors of acetylcholinesterase. In a first approach, C3-bridged naphthyridines were constructed by internal
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::e8a367fc68124a6dff17f51efd00b33e
https://doi.org/10.1002/ejoc.200800972
https://doi.org/10.1002/ejoc.200800972
Autor:
Amuri Kilonda, Wim Dehaen, Frans Compernolle, Suzanne Toppet, Luc Pieters, Isabelle E.J.A. François, Dulce María González Mosquera, Bruno P. A. Cammue, Sandra Apers, Armando Cuellar Cuellar
Publikováno v:
Planta medica: natural products and medicinal plant research
Phytochemical analysis of the leaves of BOLDOA PURPURASCENS Cav. led to isolation of four flavone glycosides, three of which are new compounds. Their structures have been determined by mass spectrometry and by 1 D and 2 D NMR analysis, i. e., 4',5-di
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9860822838f60996978643eab4a01afd
https://doi.org/10.1055/s-2008-1081332
https://doi.org/10.1055/s-2008-1081332
Publikováno v:
Tetrahedron. 64:8128-8133
A convenient synthesis of substituted pyrazino[1,2-a]benzimidazol-1(2H)ones starting from 3,5-dichloropyrazinones has been accomplished. Various 3-anilino-pyrazinones were easily converted to the desired tricyclic structures by applying a microwave a
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::a55169f9cea9c10c63b9bc5e698e0248
https://doi.org/10.1016/j.tet.2008.06.056
https://doi.org/10.1016/j.tet.2008.06.056
Autor:
Frans Compernolle, Arnout Voet, Sofie Vanlaer, Marc De Maeyer, Wim M. De Borggraeve, Constant Gielens
Publikováno v:
European Journal of Organic Chemistry. 2008:2571-2581
Spirocyclic pyridoazepines, designed as simplified analogues of the alkaloid galanthamine, were synthesised and evaluated as inhibitors of acetylcholinesterase. The key cyclisation step involved internal displacement of 2-chloro or 2-iodopyridine by
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::72db98fb0603db3f492ecd5e45e019ae
https://doi.org/10.1002/ejoc.200800062
https://doi.org/10.1002/ejoc.200800062
Publikováno v:
European Journal of Organic Chemistry. 2007:4995-4998
In this report we describe the synthesis of spirocyclic pyridoazepines starting from easily available precursors. The key step of our synthesis is an intramolecular nucleophilic aromatic substitution of the appropriate 3-substituted 2-chloropyridines
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::d4fc22c6404145db2137ed4f8e3def92
https://doi.org/10.1002/ejoc.200700614
https://doi.org/10.1002/ejoc.200700614
Autor:
Laila Kamoune, Arnout Voet, Frans Compernolle, Marc De Maeyer, Koen Robeyns, Wim M. De Borggraeve, Constant Gielens, Georges J. Hoornaert, Luc Van Meervelt
Publikováno v:
European Journal of Organic Chemistry. 2007:2977-2986
Recent efforts in the field of thrombin inhibitor research have focused on the identification of pyrazinone-containing compounds. In this manuscript we describe the synthesis of the new pyrazinones 12-36. All the targets were fully characterised and
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::5aa98989172a6f8594b629e5d88f2335
https://doi.org/10.1002/ejoc.200700180
https://doi.org/10.1002/ejoc.200700180