Zobrazeno 1 - 10
of 19
pro vyhledávání: '"Francesca, Novi"'
Autor:
Millan Mark, Roberto Maggio, Valérie Audinot, Adrian Newman-Tancredi, Jean A. Boutin, Valérie Pasteau, Didier Cussac, Thierry Dubuffet, Francesca Novi, Gilbert Lavielle, Clotilde Mannoury la Cour
Publikováno v:
Journal of Pharmacology and Experimental Therapeutics. 324:587-599
The novel, potential antipsychotic, S33138 (N-[4-[2-[(3aS,9bR)-8-cyano-1,3a,4,9b-tetrahydro[1]benzopyrano[3,4-c]pyrrol-2(3H)-yl)-ethyl]phenylacetamide), displayed approximately 25-fold higher affinity at human (h) dopamine D(3) versus hD(2L) (long is
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::e059054134496c159a41f9e74af6e250
https://doi.org/10.1124/jpet.107.126706
https://doi.org/10.1124/jpet.107.126706
Publikováno v:
FEBS Journal. 272:2939-2946
Although highly controversial just a few years ago, the idea that G-protein-coupled receptors (GPCRs) may undergo homo-oligomerization or hetero-oligomerization has recently gained considerable attention. The recognition that GPCRs may exhibit either
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::411d88fda0892fa0e622b581d3ff296f
https://doi.org/10.1111/j.1742-4658.2005.04729.x
https://doi.org/10.1111/j.1742-4658.2005.04729.x
Publikováno v:
Journal of Neurochemistry. 87:631-641
Recombinant, human dopamine D3 and D2 receptors form functional heterodimers upon co-expression in COS-7 cells. Herein, actions of the antiparkinsonian agents, S32504, ropinirole and pramipexole, at D3/D2L heterodimers were compared to their effects
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::9036df5d36fbb6178a0d92b5d2683562
https://doi.org/10.1046/j.1471-4159.2003.02038.x
https://doi.org/10.1046/j.1471-4159.2003.02038.x
Autor:
Michela Buccioni, Francesca Novi, Roberto Maggio, Alessandro Piergentili, Franco Cantalamessa, Maria Pigini, Cinzia Nasuti, Wilma Quaglia, Piero Angeli, Santi Spampinato, Gabriella Marucci, Mario Giannella, Ahmed R. Qasem
Publikováno v:
Life Sciences. 70:1427-1446
A series of muscarinic agonists, straight chained, branched, cyclic alkyl and aromatic derivatives of the oxime 1 (demox) was designed with the aim of investigating their activity on muscarinic receptor subtypes. Effects on M 1 receptor were assessed
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::1ad87c1259cf821bd1c2e347d40a8bbf
https://doi.org/10.1016/s0024-3205(01)01521-1
https://doi.org/10.1016/s0024-3205(01)01521-1
Autor:
Anna Panighini, Karl-Norbert Klotz, Roberto Maggio, Francesca Novi, Claudia Martini, Simona Daniele, Serena Cuboni, Mario Catena Dell'Osso, Maria Letizia Trincavelli
A2A adenosine receptors are considered an excellent target for drug development in several neurological and psychiatric disorders. It is noteworthy that the responses evoked by A2A adenosine receptors are regulated by D2 dopamine receptor ligands. Th
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::57afe1b3bf3202a07b0be3825011075a
http://hdl.handle.net/11697/12897
http://hdl.handle.net/11697/12897
The effects of aripiprazole, S33592, bifeprunox, N-desmethylclozapine and preclamol acting as partial agonists on recombinant D(2L) and D(3) receptors expressed both separately and concomitantly in COS-7 cells are evaluated here. Aripiprazole, S33592
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0bcd09cd3a1e51703e6bd7160885bd28
http://hdl.handle.net/11568/126400
http://hdl.handle.net/11568/126400
Autor:
Mark J, Millan, Clotilde, Mannoury la Cour, Francesca, Novi, Roberto, Maggio, Valérie, Audinot, Adrian, Newman-Tancredi, Didier, Cussac, Valérie, Pasteau, Jean-A, Boutin, Thierry, Dubuffet, Gilbert, Lavielle
Publikováno v:
The Journal of pharmacology and experimental therapeutics. 324(2)
The novel, potential antipsychotic, S33138 (N-[4-[2-[(3aS,9bR)-8-cyano-1,3a,4,9b-tetrahydro[1]benzopyrano[3,4-c]pyrrol-2(3H)-yl)-ethyl]phenylacetamide), displayed approximately 25-fold higher affinity at human (h) dopamine D(3) versus hD(2L) (long is
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::67f70bd21735391d96e5f37485b8e96f
https://pubmed.ncbi.nlm.nih.gov/18024789
https://pubmed.ncbi.nlm.nih.gov/18024789
Publikováno v:
Journal of neurochemistry. 102(4)
Aripiprazole and the candidate antipsychotics, S33592, bifeprunox, N-desmethylclozapine (NDMC) and preclamol, are partial agonists at D(2) receptors. Herein, we examined their actions at D(2L) and D(3) receptors expressed separately or together in CO
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9472a3a373b17ffd1c7d7418e8454f1c
https://pubmed.ncbi.nlm.nih.gov/17532788
https://pubmed.ncbi.nlm.nih.gov/17532788
Publikováno v:
The FEBS journal. 272(12)
Although highly controversial just a few years ago, the idea that G-protein-coupled receptors (GPCRs) may undergo homo-oligomerization or hetero-oligomerization has recently gained considerable attention. The recognition that GPCRs may exhibit either
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::70ed9790e981a81cc5cc9fb99977be18
https://pubmed.ncbi.nlm.nih.gov/15955054
https://pubmed.ncbi.nlm.nih.gov/15955054
Autor:
Franco Giorgi, Roberto Maggio, Francesca Novi, Giovanni Corsini, Laura Stanasila, Susanna Cotecchia
Publikováno v:
The Journal of biological chemistry. 280(20)
beta-Arrestins regulate the functioning of G protein-coupled receptors in a variety of cellular processes including receptor-mediated endocytosis and activation of signaling molecules such as ERK. A key event in these processes is the G protein-coupl
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ef4c75cdca99125d16d40efc2733aa9b
https://pubmed.ncbi.nlm.nih.gov/15769745
https://pubmed.ncbi.nlm.nih.gov/15769745