Zobrazeno 1 - 8
of 8
pro vyhledávání: '"Fodil Bouazza"'
Autor:
Emeline Appert, Agnès Martin‐Mingot, Omar Karam, Fabien Zunino, Bastien Michelet, Fodil Bouazza, Sébastien Thibaudeau
Publikováno v:
Chemistry (Weinheim an der Bergstrasse, Germany). 28(49)
The field of medicinal chemistry is currently witnessing a deuterium rush owing to the remarkable properties of this element as bioisoster of hydrogen atom. Aromatic hydrogen isotope exchange (HIE) is one of the most studied strategies nowadays as it
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::272a4f6b955a9aa6c56bef85e8eca3d6
https://pubmed.ncbi.nlm.nih.gov/35689822
https://pubmed.ncbi.nlm.nih.gov/35689822
Autor:
Omar Karam, Fabien Zunino, Agnès Martin-Mingot, Sébastien Thibaudeau, Alexander Mamontov, Benoît Métayer, Fodil Bouazza
Publikováno v:
Chemistry – A European Journal. 26:10411-10416
Site-selective functionalization of arenes that is complementary to classical aromatic substitution reactions remains a long-standing quest in organic synthesis. Exploiting the generation of halenium ion through oxidative process and the protonation
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::720171dd4ef57fac7c746ef21eb22f92
https://doi.org/10.1002/chem.202000902
https://doi.org/10.1002/chem.202000902
Autor:
Sébastien Alazet, Célestine Nkounkou Loumpangou, Thierry Billard, Hélène Carreyre, Jean-Maurille Ouamba, Sébastien Thibaudeau, Agnès Martin-Mingot, Gino Greco, Longin Justin Clair Bonazaba Milandou, Fodil Bouazza
Publikováno v:
Angewandte Chemie International Edition. 56:169-172
Upon activation under superacid conditions, functionalized tailor-made N-SCF3 sulfenamides served as reagents for the trifluoromethylthiolation of aromatic amines. This method has a broad substrate scope and can be used for the late-stage functionali
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::512dbc45e7cf7aad6bdbeaa73b43e3e6
https://doi.org/10.1002/anie.201609574
https://doi.org/10.1002/anie.201609574
Autor:
Ugo Castelli, Sébastien Thibaudeau, Alexandre Le Darz, Jérôme Marrot, Naima Mokhtari, Omar Karam, Fodil Bouazza, Agnès Martin-Mingot
Publikováno v:
Tetrahedron
Tetrahedron, Elsevier, 2016, 72, pp.674-689 ⟨10.1016/j.tet.2015.12.013⟩
Tetrahedron, Elsevier, 2016, 72, pp.674-689 ⟨10.1016/j.tet.2015.12.013⟩
An efficient and straightforward regio-controlled route to β-fluoro-γ-chlorinated amines was developed via an ammonium–chloronium superelectrophilic activation in superacid HF/SbF5. Through halogen directing effect the method was extended to a va
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7a7d192ac4488b7363fed9f84e0f3e61
https://doi.org/10.1016/j.tet.2015.12.013
https://doi.org/10.1016/j.tet.2015.12.013
Autor:
Hélène Carreyre, Longin Justin Clair Bonazaba Milandou, Sébastien Alazet, Fodil Bouazza, Célestine Nkounkou Loumpangou, Jean-Maurille Ouamba, Gino Greco, Thierry Billard, Agnès Martin-Mingot, Sébastien Thibaudeau
Publikováno v:
Angewandte Chemie International Edition
Angewandte Chemie International Edition, Wiley-VCH Verlag, 2017, 56 (1), pp.417-417. ⟨10.1002/anie.201611312⟩
Angewandte Chemie International Edition, Wiley-VCH Verlag, 2017, 56 (1), pp.417-417. ⟨10.1002/anie.201611312⟩
International audience
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::dc578e4f7d3be3236b4fb23657af4f7b
https://hal.archives-ouvertes.fr/hal-01610196
https://hal.archives-ouvertes.fr/hal-01610196
Autor:
Ugo Castelli, Jérôme Marrot, Sébastien Thibaudeau, Omar Karam, Fodil Bouazza, Alexandre Le Darz, Agnès Martin-Mingot, Naima Mokhtari
Publikováno v:
ChemInform. 47
An efficient and straightforward regio-controlled route to β-fluoro-γ-chlorinated amines was developed via an ammonium–chloronium superelectrophilic activation in superacid HF/SbF5. Through halogen directing effect the method was extended to a va
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::8e5aa43f69ce68a8027052528f17d008
https://doi.org/10.1002/chin.201622042
https://doi.org/10.1002/chin.201622042
Publikováno v:
Organic Letters. 5:4049-4052
[reaction: see text]. (-)-PF1163B, a new macrocyclic antifungal antibiotic isolated from Streptomyces sp., has been prepared in eight steps from (S)-citronellene. The key step is a ring-closing metathesis reaction of an ester and amide derivative obt
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e39fd43972dddfcf4cbc9be1a0d756c9
https://doi.org/10.1021/ol035309c
https://doi.org/10.1021/ol035309c
Autor:
Claudiu T. Supuran, Sébastien Thibaudeau, Ugo Castelli, Omar Karam, Muhammet Tanc, Agnès Mingot, Fodil Bouazza, Alexandre Le Darz
Publikováno v:
Journal of enzyme inhibition and medicinal chemistry. 30(5)
A series of substituted pyrrolidines and piperidines were synthesized using superacid HF/SbF5 chemistry. Investigated as inhibitors of several human carbonic anhydrase (hCA, EC 4.2.1.1) isoforms, i.e. the cytosolic hCA I and II as well as the tumor-a
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5cc89aec7ff1fa88c28bd2601c8778e5
https://pubmed.ncbi.nlm.nih.gov/25431145
https://pubmed.ncbi.nlm.nih.gov/25431145