Zobrazeno 1 - 10
of 93
pro vyhledávání: '"Florent Perret"'
Autor:
Boglárka Papp, Marc Le Borgne, Florent Perret, Christelle Marminon, Liza Józsa, Ágota Pető, Dóra Kósa, Lajos Nagy, Sándor Kéki, Zoltán Ujhelyi, Ádám Pallér, István Budai, Ildikó Bácskay, Pálma Fehér
Publikováno v:
Pharmaceutics, Vol 15, Iss 12, p 2701 (2023)
The aim of this study was to formulate and characterize CK2 inhibitor-loaded alginate microbeads via the polymerization method. Different excipients were used in the formulation to improve the penetration of an active agent and to stabilize our prepa
Externí odkaz:
https://doaj.org/article/e21b1301af1e4f0b92f5cff9c9f4e2cb
Autor:
Anthony Prandina, Lars Herfindal, Sylvie Radix, Pål Rongved, Stein O. Døskeland, Marc Le Borgne, Florent Perret
Publikováno v:
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 33, Iss 1, Pp 370-375 (2018)
Phenazine is known to regroup planar nitrogen-containing heterocyclic compounds. It was used here to enhance the bioavailability of the biologically important compound iodinin, which is near insoluble in aqueous solutions. Its water solubility has le
Externí odkaz:
https://doaj.org/article/f8efd2d694984d28a404868dc1bc4ce7
Autor:
Eszter Róka, Zoltán Ujhelyi, Mária Deli, Alexandra Bocsik, Éva Fenyvesi, Lajos Szente, Ferenc Fenyvesi, Miklós Vecsernyés, Judit Váradi, Pálma Fehér, Rudolf Gesztelyi, Caroline Félix, Florent Perret, Ildikó Katalin Bácskay
Publikováno v:
Molecules, Vol 20, Iss 11, Pp 20269-20285 (2015)
Cyclodextrins, even the 6-membered α-cyclodextrin, are approved in the various pharmacopoeias as pharmaceutical excipients for solubilizing and stabilizing drugs as well as for controlling drug release. Recently α-cyclodextrin has also been markete
Externí odkaz:
https://doaj.org/article/6f3edd0d79334feaa6d1a9ea9e7aa483
Autor:
Yannick Tauran, José Pedro Cerón-Carrasco, Moez Rhimi, Florent Perret, Beomjoon Kim, Dominique Collard, Anthony W. Coleman, Horacio Pérez-Sánchez
Publikováno v:
Antibiotics, Vol 8, Iss 2, p 73 (2019)
Inhibition of H3N2 influenza PA endonuclease activity by a panel of anionic calix[n]arenes and β-cyclodextrin sulfate has been studied. The joint experimental and theoretical results reveal that the larger, more flexible and highly water-soluble sul
Externí odkaz:
https://doaj.org/article/fe405d54e471465fac252a06a4717ea7
Autor:
Petra Arany, Eszter Róka, Laurent Mollet, Anthony W. Coleman, Florent Perret, Beomjoon Kim, Renátó Kovács, Adrienn Kazsoki, Romána Zelkó, Rudolf Gesztelyi, Zoltán Ujhelyi, Pálma Fehér, Judit Váradi, Ferenc Fenyvesi, Miklós Vecsernyés, Ildikó Bácskay
Publikováno v:
Pharmaceutics, Vol 11, Iss 6, p 277 (2019)
3D printing is attracting considerable interest for its capacity to produce prototypes and small production runs rapidly. Fused deposit modeling (FDM) was used to produce polyvalent test plates for investigation of the physical, chemical, and in-vitr
Externí odkaz:
https://doaj.org/article/93e40dde11d948069d2a5e52c7088486
Publikováno v:
Molecules, Vol 18, Iss 5, Pp 5993-6007 (2013)
The anionic calixarenes para-sulphonatocalix[4]arene and 1,3-di-Ophosphonatocalix[ 4]arene, have been used to cap silver nanoparticles. The binding of these functional particles with regard to various serum albumins (bovine serum albumin, human serum
Externí odkaz:
https://doaj.org/article/cce52d8aceff42d4989e05878c6ef791
Autor:
Abdelhamid Nacereddine, Andre Bollacke, Eszter Róka, Christelle Marminon, Zouhair Bouaziz, Ferenc Fenyvesi, Ildikó Katalin Bácskay, Joachim Jose, Florent Perret, Marc Le Borgne
Publikováno v:
Pharmaceuticals, Vol 11, Iss 1, p 10 (2018)
Since the approval of imatinib in 2001, kinase inhibitors have revolutionized cancer therapies. Inside this family of phosphotransferases, casein kinase 2 (CK2) is of great interest and numerous scaffolds have been investigated to design CK2 inhibito
Externí odkaz:
https://doaj.org/article/6a035e87689e4152973bb3407ecd5675
Autor:
Oleksandr Shkurenko, Kinga Suwinska, Florent Perret, Katia Sigaud, Antoine Leydier, Said Jebors, Anthony W. Coleman
Publikováno v:
Chemistry Journal of Moldova: General, Industrial and Ecological Chemistry, Vol 4, Iss 2, Pp 86-93 (2009)
Diamino-bicycloundecane mono-deprotonates H-calix[4]arene and the solid-structure of the resulting salt has been determined by X-ray crystallography. Two different complexes are present in the structure with the Diamino-bicycloundecane cation held in
Externí odkaz:
https://doaj.org/article/ece91d2a9bea41ac8d23644e6d0b07b0
Autor:
Florent Perret, Yannick Tauran, Kinga Suwinska, Beomjoon Kim, Cyrielle Chassain-Nely, Maxime Boulet, Anthony W. Coleman
Publikováno v:
Journal of Chemistry, Vol 2013 (2013)
A series of six anionic calix[4]arenes, having sulphonate, carboxylate, or phosphonate functions at either the para-aromatic position or the phenolic face were used to cap silver nanoparticles. Their molecular recognition properties were studied with
Externí odkaz:
https://doaj.org/article/edb732bcbe53419baa54b5c86c681786
Autor:
Laurent Vial, Julien Leclaire, Florent PERRET, Ivan Huc, Pradeep Kumar Mandal, Elise Dumont, Olivier Cala, Nicolas Vanthuyne, Ana M Belenguer, Christian Duchamp, Titouan Chetot, Emeric Jeamet, Pierre-Thomas Skowron, Benjamin Ourri, Yuan Zhang
The diastereoselective assembly of achiral constituents through a single spontaneous process into complex covalent architectures bearing multiple stereogenic elements still remains a challenge for synthetic chemists. Here, we show that such an extrem
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::31dbcca0ffb242a8718930216d72822c
https://www.repository.cam.ac.uk/handle/1810/350710
https://www.repository.cam.ac.uk/handle/1810/350710
