Comparative Analysis of Cyclization Techniques in Stapled Peptides: Structural Insights into Protein–Protein Interactions in a SARS-CoV-2 Spike RBD/hACE2 Model System.

Autor: Ferková, Sára¹ (AUTHOR), Froehlich, Ulrike¹ (AUTHOR), Nepveu-Traversy, Marie-Édith¹ (AUTHOR), Murza, Alexandre¹ (AUTHOR), Azad, Taha¹ (AUTHOR), Grandbois, Michel¹ (AUTHOR), Sarret, Philippe¹ (AUTHOR), Lavigne, Pierre¹ (AUTHOR), Boudreault, Pierre-Luc¹ (AUTHOR) pierre-luc.boudreault@usherbrooke.ca

Publikováno v: International Journal of Molecular Sciences. Jan2024, Vol. 25 Issue 1, p166. 22p.

Rational In Silico Design of Selective TMPRSS6 Peptidomimetic Inhibitors via Exploitation of the S2 Subpocket.

Autor: Desgagné, Michael, Désilets, Antoine, Ferková, Sára, Lepage, Matthieu, Perreault, Olivier, Joushomme, Alexandre, Lemieux, Gabriel, Guerrab, Walid, Froehlich, Ulrike, Comeau, Christian, Sarret, Philippe, Leduc, Richard, Boudreault, Pierre-Luc

Publikováno v: Journal of Medicinal Chemistry; 8/8/2024, Vol. 67 Issue 15, p12969-12983, 15p

Comparative Analysis of Cyclization Techniques in Stapled Peptides: Structural Insights into Protein-Protein Interactions in a SARS-CoV-2 Spike RBD/hACE2 Model System.

Autor: Ferková S; Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Institut de Pharmacologie de Sherbrooke, Université de Sherbrooke, 3001 12e Avenue Nord, Sherbrooke, QC J1H 5N4, Canada., Froehlich U; Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Institut de Pharmacologie de Sherbrooke, Université de Sherbrooke, 3001 12e Avenue Nord, Sherbrooke, QC J1H 5N4, Canada., Nepveu-Traversy MÉ; Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Institut de Pharmacologie de Sherbrooke, Université de Sherbrooke, 3001 12e Avenue Nord, Sherbrooke, QC J1H 5N4, Canada., Murza A; Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Institut de Pharmacologie de Sherbrooke, Université de Sherbrooke, 3001 12e Avenue Nord, Sherbrooke, QC J1H 5N4, Canada., Azad T; Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Institut de Pharmacologie de Sherbrooke, Université de Sherbrooke, 3001 12e Avenue Nord, Sherbrooke, QC J1H 5N4, Canada., Grandbois M; Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Institut de Pharmacologie de Sherbrooke, Université de Sherbrooke, 3001 12e Avenue Nord, Sherbrooke, QC J1H 5N4, Canada., Sarret P; Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Institut de Pharmacologie de Sherbrooke, Université de Sherbrooke, 3001 12e Avenue Nord, Sherbrooke, QC J1H 5N4, Canada., Lavigne P; Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Institut de Pharmacologie de Sherbrooke, Université de Sherbrooke, 3001 12e Avenue Nord, Sherbrooke, QC J1H 5N4, Canada., Boudreault PL; Department of Pharmacology and Physiology, Faculty of Medicine and Health Sciences, Institut de Pharmacologie de Sherbrooke, Université de Sherbrooke, 3001 12e Avenue Nord, Sherbrooke, QC J1H 5N4, Canada.

Publikováno v: International journal of molecular sciences [Int J Mol Sci] 2023 Dec 21; Vol. 25 (1). Date of Electronic Publication: 2023 Dec 21.