Zobrazeno 1 - 10
of 15
pro vyhledávání: '"Ferenc Andrasi"'
Publikováno v:
Brain Research Bulletin. 66:43-49
Cerebroprotection after administration of glutamate receptor antagonists has been well documented. The present study is intended to determine whether the non-competitive alpha-amino-3-hydroxy-methyl-4-isoxazolyl-propionic acid (AMPA) receptor antagon
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 10:899-902
Some 5-methyl analogues (14a-e) of the non-competitive AMPA antagonists 3-acylated 1-(4-aminophenyl)-4-methyl-7,8-methylenedioxy-4,5-dihydro-3H-2,3-benzodi azepines (2,3) have been synthesized. Generally they show diminished or low biological activit
Autor:
Peter Botka, Jeno Korosi, Pal Berzsenyi, István Tarnawa, Ferenc Andrasi, István Ling, Tamas Hamori
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 3:99-104
A series of N-substituted 1-(4'-aminophenyl)-4-methyl-3,4-dihydro-7,8-methylene-dioxy5H-2,3-benzodiazepines, structural analogues of the selective non-NMDA antagonist GYKI 52466, has been synthesized and tested for biological activity, in vivo and in
Publikováno v:
ChemInform. 31
Some 5-methyl analogues (14a-e) of the non-competitive AMPA antagonists 3-acylated 1-(4-aminophenyl)-4-methyl-7,8-methylenedioxy-4,5-dihydro-3H-2,3-benzodi azepines (2,3) have been synthesized. Generally they show diminished or low biological activit
Autor:
Ferenc Andrasi
Publikováno v:
ChemInform. 32
The development of therapeutic agents against peptic ulcer at the Institute for Drug Research at Budapest is reviewed. Among others, the genesis of the omeprazole molecule is described.
Publikováno v:
Brain research bulletin. 68(4)
The neuroprotective effect of talampanel, a negative allosteric modulator of alpha-amino-3-hydroxy-methyl-4-isoxazolyl-propionic acid (AMPA) receptors has been described previously. However, in these studies the histological changes and not the funct
Autor:
Gizella Ábrahám, István Tarnawa, Laszlo Gabor Harsing, Miklós Patthy, István Ling, Ferenc Andrasi, Tamas Hamori, K.M. Horvath, Pal Berzsenyi, Sandor Solyom, Istvan Kiraly, Istvan Pallagi, Gabor Kapus, Gyula Horváth, Emese Csuzdi
Publikováno v:
Bioorganicmedicinal chemistry. 8(8)
New halogen atom substituted 2,3-benzodiazepine derivatives condensed with an azole ring on the seven membered part of the ring system of type 3 and 4 as well as 5 and 6 were synthesized. It was found that chloro-, dichloro- and bromo-substitutions i
Autor:
J. Lango, E. K. Bozo, Ferenc Andrasi, T. Somorai, J. Janaky, Géza Szilágyi, Jozsef Reiter, G. Nagy
Publikováno v:
ChemInform. 21
Publikováno v:
European Journal of Pharmacology. 183:295-296
Publikováno v:
European Journal of Pharmacology. 183:1416-1417