Zobrazeno 1 - 10
of 10
pro vyhledávání: '"Ezhaya Antoine"'
Autor:
Ezhaya Antoine, Giovanbattista Schiavi, Angelo Sagrada, E. Bellora, Arturo Donetti, Henri Doods, Enzo Cereda
Publikováno v:
European Journal of Medicinal Chemistry. 29:411-421
A series of new 3-tropanol and 3-quinuclidinol esters of phenyl-substituted pyrrolidin-, piperidin- and azepin-2-oxocarboxylic acid were synthesized and tested for antimuscarinic activity. The compounds showed a preferential in vitro activity at M1 a
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::ba8113c1be1f84a9b725dcb07b6815c8
https://doi.org/10.1016/0223-5234(94)90068-x
https://doi.org/10.1016/0223-5234(94)90068-x
Publikováno v:
Tetrahedron Letters. 42:4951-4953
[3+2] Cycloaddition of alkynes to resin bound nitrile oxides gives after cleavage of 3,4,5 trisubstituted isoxazoles in acceptable yields and fair to good purity, depending on the alkyne substituents. The reaction has been automated on the ACT 496 sy
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::927678efc08830cb92fa4adfbd255f37
https://doi.org/10.1016/s0040-4039(01)00904-2
https://doi.org/10.1016/s0040-4039(01)00904-2
Autor:
Giovanbattista Schiavi, Arturo Donetti, Enzo Cereda, Angelo Sagrada, Henri Doods, Ezhaya Antoine, E. Bellora
Publikováno v:
ChemInform. 25
A series of new 3-tropanol and 3-quinuclidinol esters of phenyl-substituted pyrrolidin-, piperidin- and azepin-2-oxocarboxylic acid were synthesized and tested for antimuscarinic activity. The compounds showed a preferential in vitro activity at M1 a
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::5a2be8a256c68892b43d695a3c71e8d7
https://doi.org/10.1002/chin.199445228
https://doi.org/10.1002/chin.199445228
Autor:
E. Bellora, Enrica Dubini, Arturo Donetti, Ezhaya Antoine, Giovanni Battista Schiavi, Alessandro Brambilla, Rosella Micheletti, Antonio Schiavone, Enzo Cereda, Myrna Gil Quintero
Publikováno v:
Journal of Medicinal Chemistry. 33:2108-2113
Amidines (guanidine, formamidine, and acetamidine) were introduced as substitutes for the cationic heads present in atropine, scopolamine, and corresponding quaternary derivatives. Amidine systems are intermediate in structure between tertiary amines
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::78599fea63e587980a1f4a446489f6c5
https://doi.org/10.1021/jm00170a010
https://doi.org/10.1021/jm00170a010
Publikováno v:
In Tetrahedron Letters 23 July 2001 42(30):4951-4953
Autor:
E. Bellora, Ferdinando Pagani, Alessandro Brambilla, Arturo Donetti, Marco Turconi, Enzo Cereda, Ezhaya Antoine
Publikováno v:
European Journal of Medicinal Chemistry. 22:527-537
A series of substituted sulfinyl benzimidazoles were prepared and tested for gastric anti-secretory activity. Following initial screening, two compounds were tested for anti-ulcer activity. The new compounds showed pharmacological properties differen
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::e32fd807dff7faf4f85be53f030d6d37
https://doi.org/10.1016/0223-5234(87)90293-5
https://doi.org/10.1016/0223-5234(87)90293-5
Publikováno v:
Journal of medicinal chemistry. 32(5)
Three N-fluoroethyl-substituted (imidazolylphenyl)formamidine derivatives, namely, 2-fluoroethyl (3b), 2,2-difluoroethyl (3c), and 2,2,2-trifluoroethyl (3d), were prepared to test the effect of fluorine substitution on basicity and, then, on H2-antag
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::aa7f88d359fe4841ba5053c95eda7b4f
https://pubmed.ncbi.nlm.nih.gov/2565401
https://pubmed.ncbi.nlm.nih.gov/2565401
Publikováno v:
Chemischer Informationsdienst. 11
Some new N-substituted 6,7-benzomorphans were prepared and tested for analgetic activity. The compounds (I) and (II), which proved the most active in a preliminary screening, were submitted to a more detailed investigation, and their ED50 was determi
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::72efdeda9bcdd34669b63323c074bdca
https://doi.org/10.1002/chin.198041228
https://doi.org/10.1002/chin.198041228
Publikováno v:
Synthesis; January 1980, Vol. 1980 Issue: 12 p1009-1011, 3p
Autor:
Cereda, Enzo, Turconi, Marco, Ezhaya, Antoine, Bellora, Elio, Brambilla, Alessandro, Pagani, Ferdinando, Donetti, Arturo
Publikováno v:
In European Journal of Medicinal Chemistry 1987 22(6):527-537