Zobrazeno 1 - 7
of 7
pro vyhledávání: '"Evelyne Cerede"'
Publikováno v:
Il Farmaco. 59:981-986
The study of the relative binding affinity (RBA) to the human alpha and beta estrogen receptors (ERs) of various 7-hydroxycoumarins substituted at 4- and 3,4- positions is weak and lacks in selectivity for both ERalpha and ERbeta. The 4-(4-hydroxyphe
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5f3259d98cfa6b521e601731dcfa9524
https://doi.org/10.1016/j.farmac.2004.08.004
https://doi.org/10.1016/j.farmac.2004.08.004
Autor:
F. Nique, Evelyne Cerede, Francoise Bouchoux, G. Teutsch, Daniel Philibert, D. Gofflo, G. Lemoine
Publikováno v:
Annals of the New York Academy of Sciences. 761:5-28
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::87b6c809c13b31d1735a06b4bc93512b
https://doi.org/10.1111/j.1749-6632.1995.tb31365.x
https://doi.org/10.1111/j.1749-6632.1995.tb31365.x
Autor:
D. Gofflo, Evelyne Cerede, T. Battmann, G. Teutsch, Martine Gaillard-Kelly, A. Bonfils, Daniel Philibert, Francoise Bouchoux, Francois Goubet
Publikováno v:
The Journal of Steroid Biochemistry and Molecular Biology. 48:111-119
New N-substituted arylthiohydantoin antiandrogens were synthesized. These compounds presented exceptionally high relative binding affinities (RBAs) for the rat androgen receptor (AR): up to 3 times that of testosterone (T) and 100 times the RBAs of n
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2b010fd3f3b732626498cf6d6f8415a3
https://doi.org/10.1016/0960-0760(94)90257-7
https://doi.org/10.1016/0960-0760(94)90257-7
Publikováno v:
Steroids. 59:22-26
The synthesis of RU 45196, an 11β-substituted 19-norsteroid of the estra-4,9-diene series, incorporating the nitrobenzoxadiazole (NBD) fluorophore, is reported. The highly fluorescent target compound displayed remarkable affinity for both the proges
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b20e1dcdb4a0cb63f58b78ebee816d19
https://doi.org/10.1016/0039-128x(94)90040-x
https://doi.org/10.1016/0039-128x(94)90040-x
Publikováno v:
ChemInform. 36
The study of the relative binding affinity (RBA) to the human α and β estrogen receptors (ERs) of various 7-hydroxycoumarins substituted at 4- and 3,4- positions is weak and lacks in selectivity for both ERα and ERβ. The 4-(4-hydroxyphenyl)-7-hyd
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::dc109a0f54580f7e4437590b03469675
https://doi.org/10.1002/chin.200516124
https://doi.org/10.1002/chin.200516124
Synthesis and Relative Binding Affinity to Human Steroid Receptors of Substituted 3-Aryloxycoumarins
Autor:
Serge Kirkiacharian, Francoise Bouchoux, Francois Terrier, Evelyne Cerede, Michele Resche‐Rigon, Robert Bakhchinian
Publikováno v:
ChemInform. 35
The synthesis of a set of substituted 3-aryloxycoumarins was performed. The study of the relations between their structure and their relative binding affinity to human androgen, progesterone, α and β estrogen receptors was achieved.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8f5c43faaa678432fee166743cc8758c
https://doi.org/10.1002/chin.200409113
https://doi.org/10.1002/chin.200409113
Autor:
G. Teutsch, Francoise Bouchoux, Martine Gaillard-Kelly, Francois Goubet, Daniel Philibert, C. Branche, Evelyne Cerede, T. Battmann
Publikováno v:
The Journal of steroid biochemistry and molecular biology. 64(1-2)
The pharmacological profile of RU 58642, a new non-steroidal antiandrogen was investigated both in vitro and in vivo. In vitro, the compound displays a strong and specific affinity for androgen receptor. In vivo, its antiandrogenic activity was evalu
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::723916b80a51217c6b671092d6e11182
https://pubmed.ncbi.nlm.nih.gov/9569015
https://pubmed.ncbi.nlm.nih.gov/9569015