Zobrazeno 1 - 10
of 10
pro vyhledávání: '"Eugene D. Thorsett"'
Autor:
Brent Blackburn, Lawrence R. McGee, Eugene D. Thorsett, Mcdowell Robert S, Thomas R. Gadek, Thomas E. Rawson, Kirk Robarge, Todd C. Somers, Mark Reynolds
Publikováno v:
Journal of the American Chemical Society. 116:5077-5083
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::8a3e8bf91f52222a8ef22c977b44ce3b
https://doi.org/10.1021/ja00091a008
https://doi.org/10.1021/ja00091a008
Autor:
Peter L. Barker, Eugene D. Thorsett, Nicholas J. Skelton, Martin E. Struble, Mcdowell Robert S, Kathyrn S. Chan, Clifford Quan, Daniel J. Burdick, Thomas R. Gadek
Publikováno v:
Journal of the American Chemical Society. 116:5069-5076
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::9e1e3b22c14048ca239617de3a81001f
https://doi.org/10.1021/ja00091a007
https://doi.org/10.1021/ja00091a007
Autor:
Thomas R. Gadek, Rob Webb, Mark Reynolds, Todd C. Somers, Thomas E. Rawson, Robert S. McDowell, Maureen H. Tischler, Eugene D. Thorsett, Lawrence Mcgee, Michael C. Venuti, Kirk Robarge, Brent Blackburn
Publikováno v:
ChemInform. 25
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::964bdbc9d9745e58a64143fa2eee280f
https://doi.org/10.1002/chin.199447184
https://doi.org/10.1002/chin.199447184
Autor:
Michel C. Maillard, Roy K. Hom, Timothy E. Benson, Joseph B. Moon, Shumeye Mamo, Michael Bienkowski, Alfredo G. Tomasselli, Danielle D. Woods, D. Bryan Prince, Donna J. Paddock, Thomas L. Emmons, John A. Tucker, Michael S. Dappen, Louis Brogley, Eugene D. Thorsett, Nancy Jewett, Sukanto Sinha, Varghese John
Publikováno v:
Journal of Medicinal Chemistry; Feb2007, Vol. 50 Issue 4, p776-781, 6p
Autor:
Edgar H. Ulm, Theodore C. Vassil, Eugene D. Thorsett, William J. Greenlee, Arthur A. Patchett, Elbert E. Harris, E. R. Peterson
Publikováno v:
Proceedings of the National Academy of Sciences. 79:2176-2180
Several phosphonamides, phosphoramides, and phosphates having the general structure R-Y-P(O)(OH)-X-CH(CH3)-CO-Pro have been synthesized and tested for inhibition of angiotensin-converting enzyme (dipeptidyl carboxypeptidase; peptidyl-dipeptide hydrol
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::943b5066530d7aa2ef5915b5532866df
https://doi.org/10.1073/pnas.79.7.2176
https://doi.org/10.1073/pnas.79.7.2176
Publikováno v:
Chemischer Informationsdienst. 10
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::b4cecc48c5b97b39c3b265cc96b19394
https://doi.org/10.1002/chin.197918237
https://doi.org/10.1002/chin.197918237
Autor:
Aster Sd, T. C. Vassil, Elbert E. Harris, Arthur A. Patchett, E. R. Peterson, David Taub, E. H. Ulm, Eugene D. Thorsett
Publikováno v:
Biochemical and biophysical research communications. 111(1)
A series of potent inhibitors of angiotensin-converting enzyme (dipeptidyl carboxy-peptidase, E.C. 3.4.15.1) is described which addresses conformational aspects of the enzyme-inhibitor interaction. Conformational probes were derived from simple lacta
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::70eea43927e5865f0a2a60e4cafba168
https://pubmed.ncbi.nlm.nih.gov/6299286
https://pubmed.ncbi.nlm.nih.gov/6299286
Autor:
B.I. Lamont, J. L. Davidson, David Taub, Eugene D. Thorsett, William H. Parsons, Aster Sd, Arthur A. Patchett, E. H. Ulm
Publikováno v:
Biochemical and biophysical research communications. 117(1)
A series of potent inhibitors of angiotensin-converting enzyme (dipeptidyl carboxy-peptidase, E.C. 3.4.15.1) derived from benzofused 1-carboxyalkyl-3-(1-carboxy-3-phenylpropylamino) lactams ( III ) is described. In the most effective inhibitors (I50
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::aa81478caf4a6103042edecc91444c40
https://pubmed.ncbi.nlm.nih.gov/6318742
https://pubmed.ncbi.nlm.nih.gov/6318742
Autor:
William J. Greenlee, T. C. Vassil, Eugene D. Thorsett, James P. Springer, Arthur A. Patchett, E. H. Ulm
Publikováno v:
Biochemical and biophysical research communications. 122(2)
A class of potent inhibitors of angiotensin-converting enzyme (dipeptidyl carboxypeptidase, E.C. 3.4.15.1) is reported, in which an alpha-aza substitution into the substituted N-carboxymethyl dipeptide structure of enalapril is made. The inhibitors 2
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8d7a58e9d39e146a5452414859ab53c8
https://pubmed.ncbi.nlm.nih.gov/6087816
https://pubmed.ncbi.nlm.nih.gov/6087816
Autor:
Matthew J. Wyvratt, C. S. Sweet, E. R. Peterson, D. L. Ondeyka, ten Broeke J, Robinson Fm, Aster Sd, T. C. Vassil, T.J. Ikeler, Hirschmann Ralph F, Henry Joshua, William J. Greenlee, Tristram Edward W, Dennis M. Gross, Nancy S. Lohr, John W. Rothrock, Elbert E. Harris, Hoffsommer Rd, Arthur A. Patchett, E. H. Ulm, Alan L. Maycock, Stone Ca, David Taub, William V Ruyle, Eugene D. Thorsett, Mu Tsu Wu, L.G. Payne
Publikováno v:
Nature. 288(5788)
Much current attention focuses on the renin-angiotensin system in relation to mechanisms controlling blood pressure and renal function. Recent demonstrations (ref. 1, ref. 2 and refs therein) that angiotensin-converting enzyme inhibitors show promisi
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e321c67a3452bf870a3b1074f49f3f2d
https://pubmed.ncbi.nlm.nih.gov/6253826
https://pubmed.ncbi.nlm.nih.gov/6253826