Zobrazeno 1 - 10
of 785
pro vyhledávání: '"Eticlopride"'
Akademický článek
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Publikováno v:
Chinese Journal of Physiology, Vol 64, Iss 1, Pp 1-15 (2021)
Dopamine (DA) is important for the performance of operant behavior as revealed by psychopharmacological studies that manipulate the activity of DA subtype receptors. However, the effects of SKF83959, an atypical DA D1 receptor agonist, on operant beh
Externí odkaz:
https://doaj.org/article/ff039b669ad648fa88189c179753d95b
Akademický článek
Tento výsledek nelze pro nepřihlášené uživatele zobrazit.
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Autor:
Alessandro Bonifazi, Comfort A. Boateng, Francisco O. Battiti, Amy Hauck Newman, Jianjing Cao, Saiprasad Ravi, Kuo Hao Lee, Anver Basha Shaik, Lei Shi, Rezvan Chitsazi, Li Chen
Publikováno v:
Journal of Medicinal Chemistry. 64:15313-15333
The crystal structure of the dopamine D3 receptor (D3R) in complex with eticlopride inspired the design of bitopic ligands that explored (1) N-alkylation of the eticlopride's pyrrolidine ring, (2) shifting of the position of the pyrrolidine nitrogen,
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::03167bb15eeae9f2fd9ae627de73ecf4
https://doi.org/10.1021/acs.jmedchem.1c01353
https://doi.org/10.1021/acs.jmedchem.1c01353
Akademický článek
Tento výsledek nelze pro nepřihlášené uživatele zobrazit.
K zobrazení výsledku je třeba se přihlásit.
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Autor:
Eunju Shin, Carlo Lisci, Elisabetta Tronci, Camino Fidalgo, Roberto Stancampiano, Anders Björklund, Manolo Carta
Publikováno v:
Neurobiology of Disease, Vol 62, Iss , Pp 233-240 (2014)
Graft-induced dyskinesia (GID) is a serious complication induced by dopamine (DA) cell transplantation in parkinsonian patients. We have recently shown that DA D2 receptor blockade produces striking blockade of dyskinesia induced by amphetamine in gr
Externí odkaz:
https://doaj.org/article/ccbe828bd39b41b18b422cb486e391bc
Publikováno v:
ACS Omega, Vol 6, Iss 23, Pp 14748-14764 (2021)
ACS Omega
ACS Omega
We have performed theoretical calculations with 70 drugs that have been considered in 231 clinical trials as possible candidates to repurpose drugs for schizophrenia based on their interactions with the dopaminergic system. A hypothesis of shared pha
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::101dac0ecb93b92cf7e9181c41a21018
https://doi.org/10.1021/acsomega.0c05984
https://doi.org/10.1021/acsomega.0c05984
Autor:
Luiz F. Ferrari, Norman E. Taylor, Michael Zickella, Charles Rey, Anna Ramirez, Jacqueline Zickella, JunZhu Pei
Publikováno v:
Neuroscience
Dopamine neurons in the periaqueductal gray (PAG)/dorsal raphe are key modulators of antinociception with known supraspinal targets. However, no study has directly tested whether these neurons contribute to descending pain inhibition. We hypothesized
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::57702e9f25ce835102238b7ff7307249
https://doi.org/10.1016/j.neuroscience.2021.03.035
https://doi.org/10.1016/j.neuroscience.2021.03.035
Publikováno v:
Alcohol. 91:61-73
The rising popularity of alcohol mixed with energy drinks (AmEDs) has become a significant public health concern, with AmED users reporting higher levels of alcohol intake than non-AmED users. One mechanism proposed to explain this heightened level o
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::27af7db12f75e3bb32e0e9fbc9ca2d6c
https://doi.org/10.1016/j.alcohol.2020.12.004
https://doi.org/10.1016/j.alcohol.2020.12.004
Autor:
Bingwu Huang, Binbin Wu, Jiangfan Chen, Zhanglei Dong, Han Lin, Chenchen Jiang, Qingquan Lian
Publikováno v:
Neurochemical Research
Propofol has shown strong addictive properties in rats and humans. Adenosine A2A receptors (A2AR) in the nucleus accumbens (NAc) modulate dopamine signal and addictive behaviors such as cocaine- and amphetamine-induced self-administration. However, w
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::63c4c2f1d58cc4a9f9fc99b7e54d34cc
https://doi.org/10.1007/s11064-021-03238-9
https://doi.org/10.1007/s11064-021-03238-9