4-Hydroxy-3-nitro-1,4-dihydrotriazolo[5,1- c ][1,2,4]triazines: synthesis, antiviral activity, and electrochemical characteristics.

Autor: Drokin RA; Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 ul. Mira, 620002 Yekaterinburg, Russian Federation., Fesenko EA; Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 ul. Mira, 620002 Yekaterinburg, Russian Federation., Mozharovskaia PN; Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 ul. Mira, 620002 Yekaterinburg, Russian Federation., Medvedeva MV; Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 ul. Mira, 620002 Yekaterinburg, Russian Federation., Svalova TS; Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 ul. Mira, 620002 Yekaterinburg, Russian Federation., Kozitsina AN; Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 ul. Mira, 620002 Yekaterinburg, Russian Federation., Esaulkova YL; St. Petersburg Pasteur Institute, 14 ul. Mira, 197101, St. Petersburg, Russian Federation., Volobueva AS; St. Petersburg Pasteur Institute, 14 ul. Mira, 197101, St. Petersburg, Russian Federation., Zarubaev VV; St. Petersburg Pasteur Institute, 14 ul. Mira, 197101, St. Petersburg, Russian Federation., Rusinov VL; Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 ul. Mira, 620002 Yekaterinburg, Russian Federation.; I. Ya. Postovsky Institute of Organic Synthesis, Ural Branch of Russian Academy of Sciences, 22/20 ul. S. Kovalevskoi, 620108 Yekaterinburg, Russian Federation.

Publikováno v: Russian chemical bulletin = Izvestiia Akademii nauk. Seriia khimicheskaia [Russ Chem Bull] 2022; Vol. 71 (11), pp. 2460-2466. Date of Electronic Publication: 2022 Dec 19.

Synthesis of isomeric 4-( N -methyltetrazolylamino)-2-phenyl-4 H -thiopyrano[2,3- b ]quinoline-3-carbaldehydes and 4-hydroxy-2-phenyl-4 H -thiopyrano[2,3- b ]quinoline-3-carbaldehyde based on tandem thiol-Michael and (aza)-Morita-Baylis-Hillman reactions and an in vitro study of the activity of the obtained compounds against influenza virus.

Autor: Khramchikhin AV; Saint Petersburg State Institute of Technology (Technical University), 26 Moskovsky Ave, Saint Petersburg, 190013 Russia., Skryl'nikova MА; Saint Petersburg State Institute of Technology (Technical University), 26 Moskovsky Ave, Saint Petersburg, 190013 Russia., Pavlyukova YN; Saint Petersburg State Institute of Technology (Technical University), 26 Moskovsky Ave, Saint Petersburg, 190013 Russia., Zarubaev VV; Saint Petersburg Pasteur Research Institute of Epidemiology and Microbiology, 14 Mira St, Saint Petersburg, 197101 Russia., Esaulkova YL; Saint Petersburg Pasteur Research Institute of Epidemiology and Microbiology, 14 Mira St, Saint Petersburg, 197101 Russia., Muryleva AА; Saint Petersburg Pasteur Research Institute of Epidemiology and Microbiology, 14 Mira St, Saint Petersburg, 197101 Russia., Shmanyova NT; Saint Petersburg State Institute of Technology (Technical University), 26 Moskovsky Ave, Saint Petersburg, 190013 Russia., Danagulyan GG; Russian-Armenian University, 123 Hovsep Emin St, 0051 Yerevan, Armenia.; Scientific Technological Center of Organic and Pharmaceutical Chemistry of the National Academy of Sciences of the Republic of Armenia, 26a Azatutyan Ave, 0014 Yerevan, Armenia., Ostrovskii VА; Saint Petersburg State Institute of Technology (Technical University), 26 Moskovsky Ave, Saint Petersburg, 190013 Russia.

Publikováno v: Chemistry of heterocyclic compounds [Chem Heterocycl Compd (N Y)] 2022; Vol. 58 (4-5), pp. 267-270. Date of Electronic Publication: 2022 May 25.

Methods of Synthesis and Antiviral Activity of New 4-Alkyl-3-Nitro-1,4-Dihydroazolo[5,1- c ][1,2,4]Triazin-4-ols.

Autor: Drokin RA; Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St, Yekaterinburg, 620002 Russia., Tiufiakov DV; Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St, Yekaterinburg, 620002 Russia., Voinkov EK; Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St, Yekaterinburg, 620002 Russia., Slepukhin PA; Postovsky Institute of Organic Synthesis, Ural Branch of the Russian Academy of Sciences, 22/20 Sofyi Kovalevskoi St, Yekaterinburg, 620108 Russia., Ulomsky EN; Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St, Yekaterinburg, 620002 Russia.; Postovsky Institute of Organic Synthesis, Ural Branch of the Russian Academy of Sciences, 22/20 Sofyi Kovalevskoi St, Yekaterinburg, 620108 Russia., Esaulkova YL; Saint Petersburg Pasteur Research Institute of Epidemiology and Microbiology, 14 Mira St, Saint Petersburg, 197101 Russia., Volobueva AS; Saint Petersburg Pasteur Research Institute of Epidemiology and Microbiology, 14 Mira St, Saint Petersburg, 197101 Russia., Lantseva KS; Saint Petersburg State University, 7/9 University Embankment, Saint Petersburg, 199034 Russia., Misyurina MA; Saint Petersburg Pasteur Research Institute of Epidemiology and Microbiology, 14 Mira St, Saint Petersburg, 197101 Russia., Zarubaev VV; Saint Petersburg Pasteur Research Institute of Epidemiology and Microbiology, 14 Mira St, Saint Petersburg, 197101 Russia., Rusinov VL; Ural Federal University named after the first President of Russia B. N. Yeltsin, 19 Mira St, Yekaterinburg, 620002 Russia.; Postovsky Institute of Organic Synthesis, Ural Branch of the Russian Academy of Sciences, 22/20 Sofyi Kovalevskoi St, Yekaterinburg, 620108 Russia.

Publikováno v: Chemistry of heterocyclic compounds [Chem Heterocycl Compd (N Y)] 2021; Vol. 57 (4), pp. 473-478. Date of Electronic Publication: 2021 May 12.

7-Imidazolyl-substituted 4'-methoxy and 3',4'-dimethoxy-containing polyfluoroflavones as promising antiviral agents.

Autor: Shcherbakov KV; Postovsky Institute of Organic Synthesis UD RAS, 22 Kovalevskoy str., Yekaterinburg, 620137, Russian Federation., Artemyeva MA; Postovsky Institute of Organic Synthesis UD RAS, 22 Kovalevskoy str., Yekaterinburg, 620137, Russian Federation., Burgart YV; Postovsky Institute of Organic Synthesis UD RAS, 22 Kovalevskoy str., Yekaterinburg, 620137, Russian Federation., Saloutin VI; Postovsky Institute of Organic Synthesis UD RAS, 22 Kovalevskoy str., Yekaterinburg, 620137, Russian Federation., Volobueva AS; Institut Pasteur in Saint-Petersburg for Research in Epidemiology and Microbiology of Federal Service for Surveillance on Consumer Rights Protection and Human Wellbeing, 14 Mira str., Saint-Petersburg, 197101, Russian Federation., Misiurina MA; Institut Pasteur in Saint-Petersburg for Research in Epidemiology and Microbiology of Federal Service for Surveillance on Consumer Rights Protection and Human Wellbeing, 14 Mira str., Saint-Petersburg, 197101, Russian Federation., Esaulkova YL; Institut Pasteur in Saint-Petersburg for Research in Epidemiology and Microbiology of Federal Service for Surveillance on Consumer Rights Protection and Human Wellbeing, 14 Mira str., Saint-Petersburg, 197101, Russian Federation., Sinegubova EO; Institut Pasteur in Saint-Petersburg for Research in Epidemiology and Microbiology of Federal Service for Surveillance on Consumer Rights Protection and Human Wellbeing, 14 Mira str., Saint-Petersburg, 197101, Russian Federation., Zarubaev VV; Institut Pasteur in Saint-Petersburg for Research in Epidemiology and Microbiology of Federal Service for Surveillance on Consumer Rights Protection and Human Wellbeing, 14 Mira str., Saint-Petersburg, 197101, Russian Federation.

Publikováno v: Journal of fluorine chemistry [J Fluor Chem] 2020 Dec; Vol. 240, pp. 109657. Date of Electronic Publication: 2020 Oct 10.

5-Chloro-2-thiophenyl-1,2,3-triazolylmethyldihydroquinolines as dual inhibitors of Mycobacterium tuberculosis and influenza virus: Synthesis and evaluation.

Autor: Marvadi SK; Fluro and Agrochemicals Division (Organic Chemistry Division-II), CSIR-Indian Institute of Chemical Technology, Hyderabad 500007, Telangana, India., Krishna VS; Medicinal Chemistry and Antimycobacterial Research Laboratory, Pharmacy Group, Birla Institute of Technology and Science-Pilani, Hyderabad Campus, Jawahar Nagar, Hyderabad 500078, Telangana, India., Sinegubova EO; Pasteur Institute of Epidemiology and Microbiology, 14 Mira Str., 197101 St. Petersburg, Russian Federation., Volobueva AS; Pasteur Institute of Epidemiology and Microbiology, 14 Mira Str., 197101 St. Petersburg, Russian Federation., Esaulkova YL; Pasteur Institute of Epidemiology and Microbiology, 14 Mira Str., 197101 St. Petersburg, Russian Federation., Muryleva AA; Pasteur Institute of Epidemiology and Microbiology, 14 Mira Str., 197101 St. Petersburg, Russian Federation., Tentler DG; Institute of Cytology, Russian Academy of Sciences, 4, Tikhorezky Av., 194064, Russian Federation., Sriram D; Medicinal Chemistry and Antimycobacterial Research Laboratory, Pharmacy Group, Birla Institute of Technology and Science-Pilani, Hyderabad Campus, Jawahar Nagar, Hyderabad 500078, Telangana, India., Zarubaev VV; Pasteur Institute of Epidemiology and Microbiology, 14 Mira Str., 197101 St. Petersburg, Russian Federation., Kantevari S; Fluro and Agrochemicals Division (Organic Chemistry Division-II), CSIR-Indian Institute of Chemical Technology, Hyderabad 500007, Telangana, India; Academy of Scientific and Innovative Research, CSIR-Indian Institute of Chemical Technology, Hyderabad 500 007, Telangana, India. Electronic address: ksrinivas@iict.res.in.

Publikováno v: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2019 Sep 15; Vol. 29 (18), pp. 2664-2669. Date of Electronic Publication: 2019 Jul 24.