Zobrazeno 1 - 7
of 7
pro vyhledávání: '"Erica Gazzillo"'
Autor:
Ester Colarusso, Erica Gazzillo, Eleonora Boccia, Stefania Terracciano, Ines Bruno, Giuseppe Bifulco, Maria Giovanna Chini, Gianluigi Lauro
Publikováno v:
Molecules, Vol 29, Iss 17, p 4025 (2024)
A 3D structure-based pharmacophore model built for bromodomain-containing protein 4 (BRD4) is reported here, specifically developed for investigating and identifying the key structural features of the (+)-JQ1 known inhibitor within the BRD4 binding s
Externí odkaz:
https://doaj.org/article/4c4d5af09cf840049e468ff4e7d95879
Autor:
Valentina Parisi, Giuliana Donadio, Maria Laura Bellone, Soumia Belaabed, Ammar Bader, Angela Bisio, Valeria Iobbi, Erica Gazzillo, Maria Giovanna Chini, Giuseppe Bifulco, Immacolata Faraone, Antonio Vassallo
Publikováno v:
Plants, Vol 12, Iss 13, p 2421 (2023)
Premna, a genus consisting of approximately 200 species, predominantly thrives in tropical and subtropical areas. Many of these species have been utilized in ethnopharmacology for diverse medicinal applications. In Saudi Arabia, Premna resinosa (Hoch
Externí odkaz:
https://doaj.org/article/9ccbc0c663a04effa485b601e93ed751
Autor:
Erica Gazzillo, Stefania Terracciano, Dafne Ruggiero, Marianna Potenza, Maria Giovanna Chini, Gianluigi Lauro, Katrin Fischer, Robert Klaus Hofstetter, Assunta Giordano, Oliver Werz, Ines Bruno, Giuseppe Bifulco
Publikováno v:
Molecules, Vol 27, Iss 12, p 3866 (2022)
The development of new bioactive compounds represents one of the main purposes of the drug discovery process. Various tools can be employed to identify new drug candidates against pharmacologically relevant biological targets, and the search for new
Externí odkaz:
https://doaj.org/article/968f9ee74c334cf49eabf861eeb7485d
Autor:
Vassallo, Valentina Parisi, Giuliana Donadio, Maria Laura Bellone, Soumia Belaabed, Ammar Bader, Angela Bisio, Valeria Iobbi, Erica Gazzillo, Maria Giovanna Chini, Giuseppe Bifulco, Immacolata Faraone, Antonio
Publikováno v:
Plants; Volume 12; Issue 13; Pages: 2421
Premna, a genus consisting of approximately 200 species, predominantly thrives in tropical and subtropical areas. Many of these species have been utilized in ethnopharmacology for diverse medicinal applications. In Saudi Arabia, Premna resinosa (Hoch
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=multidiscipl::1659f35374e98c887816beaafb10c2b8
Autor:
Ester Colarusso, Sara Ceccacci, Maria Chiara Monti, Erica Gazzillo, Assunta Giordano, Maria Giovanna Chini, Maria Grazia Ferraro, Marialuisa Piccolo, Dafne Ruggiero, Carlo Irace, Stefania Terracciano, Ines Bruno, Giuseppe Bifulco, Gianluigi Lauro
Targeting bromodomain-containing protein 9 (BRD9) represents a promising strategy for the development of new agents endowed with anticancer properties. With this aim, a set of 2,4,5-trisubstituted-2,4-dihydro-3H-1,2,4-triazol-3-one-based compounds wa
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b262d7a006b1739ffe998ec105fe5174
https://hdl.handle.net/11386/4826617
https://hdl.handle.net/11386/4826617
Autor:
Maria Grazia Ferraro, Stefania Terracciano, Giuseppe Bifulco, Gianluigi Lauro, Erica Gazzillo, Francesco Maione, Marialuisa Piccolo, Ines Bruno, Maria Giovanna Chini, Martina Pierri, Carlo Irace
Publikováno v:
Bioorganic chemistry. 118
A well-structured in silico workflow is here reported for disclosing structure-based pharmacophore models against bromodomain-containing protein 9 (BRD9), accelerating virtual screening campaigns and facilitating the identification of novel binders.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::27aa6efe33248726f54eb7d99ad900e1
https://pubmed.ncbi.nlm.nih.gov/34823196
https://pubmed.ncbi.nlm.nih.gov/34823196