Zobrazeno 1 - 10
of 10
pro vyhledávání: '"Eric Carnazzi"'
Autor:
Sonia Cantel, Philippe Marin, Jean-Louis Banères, Gilbert Bergé, Karine Puget, Jean Martinez, Charlène Valmalle, Gilles Subra, Anne-Claire Coyne, Céline M'Kadmi, Jérémie Neasta, Jean-Claude Galleyrand, Valérie Daugé, Nicole Bernad, Jacky Marie, Didier Gagne, Eric Carnazzi, Marie-Lou Kemel
Publikováno v:
British Journal of Pharmacology. 173:1314-1328
Background and PurposeUsing an in-house bioinformatics programme, we identified and synthesized a novel nonapeptide, H-Pro-Pro-Thr-Thr-Thr-Lys-Phe-Ala-Ala-OH. Here, we have studied its biological activity, in vitro and in vivo, and have identified it
Autor:
Chantal Escrieut, Philippe Crespy, Eric Carnazzi, Daniel Fourmy, Jean Martinez, Catherine Oiry, Jean Claude Galleyrand, Géraldine Ibarz, Didier Gagne
Publikováno v:
British Journal of Pharmacology. 147:951-958
In cells overexpressing active MEKK1 to enhance c-Jun trans-activation, expression of rat cholecystokinin 1 receptor increased the activity of c-Jun while in the same experimental conditions overexpression of mouse cholecystokinin 1 receptor represse
Publikováno v:
Journal of Medicinal Chemistry. 48:3379-3388
We designed and synthesized new photoactivatable linear vasopressin analogues containing benzophenone photophores. All compounds were monitored and purified using RP-HPLC and characterized by mass spectrometry. Affinity and selectivity were determine
Autor:
Christophe Breton, Eric Carnazzi, Claude Barberis, Laurent Guillou, André Aumelas, René Seyer, Bernard Mouillac
Publikováno v:
Journal of Medicinal Chemistry. 44:3022-3030
Using a segment strategy, we have synthesized four iodinated photoactivatable cyclic peptidic ligands of oxytocin, bearing a beta-mercapto-betabeta-cyclopentamethylene propionic group (Pmp) on their N-terminus. All the syntheses were RP-HPLC monitore
Autor:
Thierry Durroux, Claude Barberis, Hichem Chellil, Majida Kabbaj-Benmansour, Eric Carnazzi, Hans H. Zingg, Christophe Breton, Bernard Mouillac, Denis Morin, René Seyer, Sylvie Phalipou
Publikováno v:
Journal of Biological Chemistry. 276:26931-26941
Understanding of the molecular determinants responsible for antagonist binding to the oxytocin receptor should provide important insights that facilitate rational design of potential therapeutic agents for the treatment of preterm labor. To study lig
Autor:
Nathalie Cotte, Bernard Mouillac, Serge Jard, Sylvie Phalipou, Eric Carnazzi, Claude Barberis, Eve Mahe, René Seyer
Publikováno v:
Journal of Biological Chemistry. 272:26536-26544
The study of antagonist-binding domains of the human V1a vasopressin receptor was performed using a radioiodinated photoreactive peptide antagonist. This ligand displayed a high affinity for the receptor expressed in Chinese hamster ovary cell membra
Publikováno v:
Journal of Medicinal Chemistry. 37:1841-1849
A series of new linear photoactivatable and iodinatable antagonists of the neuropeptidic hormone vasopressin was designed and synthesized by a combination of PyBOP-mediated Boc/solid-phase peptide synthesis and solution synthesis approaches. These we
Autor:
Sylvie Phalipou, André Aumelas, Eric Carnazzi, Gilles Guillon, Bernard Mouillac, René Seyer, Claude Barberis
Publikováno v:
European journal of biochemistry. 247(3)
We have synthesized and fully characterized by fast-atom-bombardment-mass, NMR and ultraviolet spectroscopies the vasopressin antagonist 3-azidophenylpropionyl-D-Tyr(Me)-Phe-Gln-Asn-Arg-Pro-Arg-Tyr(3I )-NH2. Easily radioiodinatable just before use, i
Publikováno v:
International journal of peptide and protein research. 44(4)
The Ser(P)-containing peptide corresponding to phospholamban 11-19, Ac-Ala-Ile-Arg-Are-Ala-Ser(P)-Thr-Ile-Glu-NH2, was prepared by the use of Boc-Ser(PO3Ph2)-OH in Boc/solid-phase peptide synthesis followed by HF cleavage of the peptide from the poly
Publikováno v:
Peptides 1992 ISBN: 9789401046466
Peptides 1992
Peptides 1992
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::4b9156d1c4588c88d4e5b856e5f4b05f
https://doi.org/10.1007/978-94-011-1470-7_289
https://doi.org/10.1007/978-94-011-1470-7_289