Zobrazeno 1 - 10
of 14
pro vyhledávání: '"Enrico, Rango"'
Autor:
Enrico Rango, Salvatore Di Maria, Claudio Zamperini, Federica Poggialini, Emmanuele Crespan, Cecilia Perini, Samantha Sabetta, Simona Saponara, Fabio Fusi, Giovanni Maga, Adriano Angelucci, Eugenio Gaudio, Francesco Berton, Silvia Schenone, Lorenzo Botta, Elena Dreassi, Maurizio Botta
Publikováno v:
Pharmaceutical Chemistry Journal. 56:1616-1626
Autor:
Enrico Rango, Fabio Pastorino, Chiara Brignole, Arianna Mancini, Federica Poggialini, Salvatore Di Maria, Claudio Zamperini, Giulia Iovenitti, Anna Lucia Fallacara, Samantha Sabetta, Letizia Clementi, Massimo Valoti, Silvia Schenone, Adriano Angelucci, Mirco Ponzoni, Elena Dreassi, Maurizio Botta
Publikováno v:
Biomedicines, Vol 10, Iss 3, p 659 (2022)
Si306, a pyrazolo[3,4-d]pyrimidine derivative recently identified as promising anticancer agent, has shown favorable in vitro and in vivo activity profile against neuroblastoma (NB) models by acting as a competitive inhibitor of c-Src tyrosine kinase
Externí odkaz:
https://doaj.org/article/76fcd042be33447e9734d22a84d6e765
Autor:
Lorenzo J. I. Balestri, Ilaria D’Agostino, Enrico Rango, Chiara Vagaggini, Rosalba Marchitiello, Melinda Mariotti, Alexandru Casian, Davide Deodato, Giuseppina I. Truglio, Francesco Orofino, Maurizio Sanguinetti, Francesca Bugli, Lorenzo Botta, Elena Dreassi
Publikováno v:
Molecular Diversity. 26:3399-3409
The rise of antimicrobial-resistant phenotypes and the spread of the global pandemic of COVID-19 are worsening the outcomes of hospitalized patients for invasive fungal infections. Among them, candidiases are seriously worrying, especially since the
Autor:
Francesca Migliorini, Elena Cini, Elena Dreassi, Federica Finetti, Giovanni Ievoli, Giulia Macrì, Elena Petricci, Enrico Rango, Lorenza Trabalzini, Maurizio Taddei
Publikováno v:
Chemical communications (Cambridge, England). 58(75)
We report a new 1-6 self-immolative, traceless crosslinker derived from the natural product gallic acid. The linker acts through a pH-dependent mechanism for drug release. This 5-(hydroxymethyl)pyrogallol orthoester derivative (HMPO) was stable for 2
Autor:
Anna Lucia Fallacara, Claudio Zamperini, Ana Podolski-Renić, Jelena Dinić, Tijana Stanković, Marija Stepanović, Arianna Mancini, Enrico Rango, Giulia Iovenitti, Alessio Molinari, Francesca Bugli, Maurizio Sanguinetti, Riccardo Torelli, Maurizio Martini, Laura Maccari, Massimo Valoti, Elena Dreassi, Maurizio Botta, Milica Pešić, Silvia Schenone
Publikováno v:
Cancers, Vol 11, Iss 6, p 848 (2019)
Overexpression of P-glycoprotein (P-gp) and other ATP-binding cassette (ABC) transporters in multidrug resistant (MDR) cancer cells is responsible for the reduction of intracellular drug accumulation, thus decreasing the efficacy of chemotherapeutics
Externí odkaz:
https://doaj.org/article/9caea2c9a38346f69aba9354c133ee07
Autor:
Enrico, Rango, Fabio, Pastorino, Chiara, Brignole, Arianna, Mancini, Federica, Poggialini, Salvatore, Di Maria, Claudio, Zamperini, Giulia, Iovenitti, Anna Lucia, Fallacara, Samantha, Sabetta, Letizia, Clementi, Massimo, Valoti, Silvia, Schenone, Adriano, Angelucci, Mirco, Ponzoni, Elena, Dreassi, Maurizio, Botta
Publikováno v:
Biomedicines. 10(3)
Si306, a pyrazolo[3,4
Autor:
Ilaria D'Agostino, Claudia Ardino, Giulio Poli, Filomena Sannio, Massimiliano Lucidi, Federica Poggialini, Daniela Visaggio, Enrico Rango, Silvia Filippi, Elena Petricci, Paolo Visca, Lorenzo Botta, Jean-Denis Docquier, Elena Dreassi
The ever-faster rise of antimicrobial resistance (AMR) represents a major global Public Health challenge. New chemical entities with innovative Modes of Action (MoAs) are thus desirable. We recently reported the development of a novel class of broad-
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::69e3288bdfd5d4a35b97fe92a18a8663
https://hdl.handle.net/11590/399659
https://hdl.handle.net/11590/399659
Autor:
Elena Dreassi, Ilaria Vicenti, Frank J. M. van Kuppeveld, Matteo Incerti, Marco Radi, Simona Bertoni, Lisa Bauer, Emmanuele Crespan, Adele Boccuto, Maurizio Zazzi, Noemi Olivieri, Marleen Zwaagstra, Marika Allodi, Giovanni Maga, Enrico Rango, Maria Grazia Martina
Publikováno v:
ChemMedChem, 16(23), 3548. John Wiley and Sons Ltd
Chemmedchem
Chemmedchem
Over half a century since the description of the first antiviral drug, “old” re‐emerging viruses and “new” emerging viruses still represent a serious threat to global health. Their high mutation rate and rapid selection of resistance toward
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5b2b2d5dd1fc50f7a61c2488ee2fca91
https://dspace.library.uu.nl/handle/1874/417563
https://dspace.library.uu.nl/handle/1874/417563
Autor:
Nicola Perrotti, Silvia Schenone, Stefano Marianelli, Annarita Cianciusi, Claudia Immacolata Trivisani, Arianna Mancini, Lucia D'Antona, Annalaura Brai, Alessio Molinari, Elena Dreassi, Claudio Zamperini, Enrico Rango, Anna Lucia Fallacara, Maurizio Botta, Giulia Iovenitti
Publikováno v:
European journal of medicinal chemistry. 223
Si113, a pyrazolo[3,4-d]pyrimidine derivative, gained more attention as an anticancer agent due to its potent anticancer activity on both in vitro and in vivo hepatocellular carcinomas (HCC) and ovarian carcinoma models. But the drawback is the low w
Autor:
Giulia Vignaroli, Giulia Iovenitti, Arianna Mancini, Elena Dreassi, Adriano Angelucci, Maurizio Botta, Monia Chebbi, Silvia Schenone, Alessio Molinari, Francesco Orofino, Maura Caruana, Enrico Rango, Giovanni Luca Gravina
Publikováno v:
ACS Med Chem Lett
[Image: see text] Gold-nanoparticle (AuNP)-conjugated drugs represent a promising and innovative antitumor therapeutic approach. In our study, we describe the design, the synthesis, the preparation, and the characterization of AuNPs conjugated with t
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f25cc5fb81adfcd90acb6d0841042ce0
http://hdl.handle.net/11365/1105986
http://hdl.handle.net/11365/1105986