Zobrazeno 1 - 4
of 4
pro vyhledávání: '"Enrica Granci"'
Autor:
Laurie J. Gordon, Anna-Maria Capelli, Laura Zonzini, Manuela Borriello, Romano Di-Fabio, Enrica Granci, Massimo Gianotti, Roberto Arban, Simone Spada, Barbara Bertani, Stefania Faedo, Valeria Zucchelli, Alessandra Pasquarello, Angela Worby, Steven Mark Bromidge
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 20:7092-7096
5-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]ethyl}-2(1H)-quinolinones and 3,4-dihydro-2(1H)-quinolinones have been identified with different combinations of 5-HT(1) autoreceptor antagonist and hSerT potencies and excellent rat PK profiles. The avai
Autor:
Ilaria Sartori, Laura Zonzini, Laurie J. Gordon, Angela Worby, Stefano Fontana, Manuela Borriello, Silvia Bison, Jeannette M. Watson, Steven Mark Bromidge, Giovanna Dal Forno, Colin Philip Leslie, Alessandra Pasquarello, Anna Sava, Luca G. Moccia, Barbara Bertani, Roberto Arban, Daniele Donati, Enrica Granci, Valeria Zucchelli, Paolo Cavanni, Massimo Gianotti, Romano Di-Fabio
Publikováno v:
Journal of Medicinal Chemistry. 53:5827-5843
Bioisoteric replacement of the metabolically labile N-methyl amide group of a series of benzoxazinones with small heterocyclic rings has led to novel series of fused tricyclic benzoxazines which are potent 5-HT1A/B/D receptor antagonists with and wit
Autor:
Alessia Vesentini, Luigi Piero Stasi, Barbara Bertani, Matthew Hill, Jeannette M. Watson, Steven Mark Bromidge, Enrica Granci, Laura Zonzini, Valeria Zucchelli, Howard Robert Marshall, Stefania Faedo, Giancarlo Merlo, Laurie J. Gordon, Manuela Borriello
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 18:5653-5656
Investigation of a series 6-[2-(4-aryl-1-piperazinyl)ethyl]-2H-1,4-benzoxazin-3(4H)-ones has led to the discovery of potent 5-HT(1A/1B/1D) receptor antagonists with and without additional SerT affinity. Modulation of the different target activities g
Autor:
Steven M, Bromidge, Roberto, Arban, Barbara, Bertani, Silvia, Bison, Manuela, Borriello, Paolo, Cavanni, Giovanna, Dal Forno, Romano, Di-Fabio, Daniele, Donati, Stefano, Fontana, Massimo, Gianotti, Laurie J, Gordon, Enrica, Granci, Colin P, Leslie, Luca, Moccia, Alessandra, Pasquarello, Ilaria, Sartori, Anna, Sava, Jeannette M, Watson, Angela, Worby, Laura, Zonzini, Valeria, Zucchelli
Publikováno v:
Journal of medicinal chemistry. 53(15)
Bioisoteric replacement of the metabolically labile N-methyl amide group of a series of benzoxazinones with small heterocyclic rings has led to novel series of fused tricyclic benzoxazines which are potent 5-HT(1A/B/D) receptor antagonists with and w