Zobrazeno 1 - 5
of 5
pro vyhledávání: '"Emma R. Shore"'
Autor:
Paul M. O’Neill, Richard K. Amewu, Susan A. Charman, Sunil Sabbani, Nina F. Gnädig, Judith Straimer, David A. Fidock, Emma R. Shore, Natalie L. Roberts, Michael H.-L. Wong, W. David Hong, Chandrakala Pidathala, Chris Riley, Ben Murphy, Ghaith Aljayyoussi, Francisco Javier Gamo, Laura Sanz, Janneth Rodrigues, Carolina Gonzalez Cortes, Esperanza Herreros, Iñigo Angulo-Barturén, María Belén Jiménez-Díaz, Santiago Ferrer Bazaga, María Santos Martínez-Martínez, Brice Campo, Raman Sharma, Eileen Ryan, David M. Shackleford, Simon Campbell, Dennis A. Smith, Grennady Wirjanata, Rintis Noviyanti, Ric N. Price, Jutta Marfurt, Michael J. Palmer, Ian M. Copple, Amy E. Mercer, Andrea Ruecker, Michael J. Delves, Robert E. Sinden, Peter Siegl, Jill Davies, Rosemary Rochford, Clemens H. M. Kocken, Anne-Marie Zeeman, Gemma L. Nixon, Giancarlo A. Biagini, Stephen A. Ward
Publikováno v:
Nature Communications, Vol 8, Iss 1, Pp 1-10 (2017)
Artemisinin-resistantPlasmodium is an increasing problem. Here, using a medicinal chemistry programme, the authors identify a tetraoxane-based drug candidate that shows no cross-resistance with an artemisinin-resistant strain (PfK13-C580Y) and is eff
Externí odkaz:
https://doaj.org/article/d0b09995908d4fd1a466aa398f702f2f
Autor:
Sunil Sabbani, Jill Davies, Paul McGillan, Paul O´Neill, Ben Murphy, Richard Amewu, Matthew J. Schnaderbeck, Christopher Riley, Gemma L. Nixon, Emma R. Shore, Stephen A. Ward, Natalie L. Roberts
Publikováno v:
TETRAHEDRON
An efficient route to the synthesis of potent antimalarial aryloxy 1,2,4,5-tetraoxanes is described that permits parallel synthesis for Structure–Activity Relationship (SAR) investigations. Brief details of the in vitro and in vivo antimalarial eva
Autor:
Diane Latawiec, Sravan R. Pandalaneni, Li Wen, N.M. Kershaw, Emma R. Shore, Neil G. Berry, David N. Criddle, Muhammad A. Javed, Robert Sutton, Paul M. O'Neill, Muhammad Awais, Robert R. Gibson, Lu-Yun Lian
Publikováno v:
Journal of Medicinal Chemistry. 59:2596-2611
Opening of the mitochondrial permeability transition pore (MPTP) causes mitochondrial dysfunction and necrosis in acute pancreatitis (AP), a condition without specific drug treatment. Cyclophilin D (CypD) is a mitochondrial matrix peptidyl-prolyl iso
Autor:
Afthab Hussain, Amy E. Chadwick, Paul M. O'Neill, Maria Lurdes Santos Cristiano, Neil G. Berry, Richard Cosstick, James W. Firman, Lília I. L. Cabral, Cerys Bateman, Sunil Sabbani, Louise La Pensee, Nuna Araújo, Raman Sharma, Omar Janneh, Yi Hang Wu, Adelina Gavrila, Inder Bhamra, Emma R. Shore, Paul A. Stocks, Stephen A. Ward
Publikováno v:
Repositório Científico de Acesso Aberto de Portugal
Repositório Científico de Acesso Aberto de Portugal (RCAAP)
instacron:RCAAP
Repositório Científico de Acesso Aberto de Portugal (RCAAP)
instacron:RCAAP
Artemisinin-based combination therapies (ACTs) are currently the recommended treatment for uncomplicated and severe cases of malaria.[1] Additionally, artemisinins, as well as a number of other sesquiterpene lactones (SLs), are currently in phase I
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1d86c0624586a16d1eedea7c67f116d3
https://hdl.handle.net/10400.1/4230
https://hdl.handle.net/10400.1/4230
Autor:
Cerys Bateman, Paul M. O'Neill, Richard Cosstick, Sunil Sabbani, Louise La Pensee, Omar Janneh, Afthab Hussain, Raman Sharma, Yi Hang Wu, James W. Firman, Nuna Araújo, Inder Bhamra, Stephen A. Ward, Paul A. Stocks, Lília I. L. Cabral, Maria Lurdes Santos Cristiano, Neil G. Berry, Amy E. Chadwick, Adelina Gavrila, Emma R. Shore
Publikováno v:
ChemMedChem. 8:674-674