Zobrazeno 1 - 2
of 2
pro vyhledávání: '"Ellen Schouteden"'
Autor:
Frank Meeussen, Dirk Van den Heuvel, Tom Callewaert, Peter Van der Donck, Erika De Bie, Didier Philippe Robert Schils, Ellen Schouteden, Fred Stappers, Michelle Coppens, Kristof Eersels, Richard van Heck, Geoffrey François Freddy Ghislain Solberghe
Publikováno v:
Organic Process Research & Development. 12:530-536
The aniline derivative 3 is a key building block of rilpivirine (TMC278) 2, a new potent NNRTI compound under clinical evaluation. In this paper we describe the development of a new synthesis of 3 based on a Heck coupling between a halogenated anilin
Autor:
Didier Schils, Fred Stappers, Geoffrey Solberghe, Richard van Heck, Michelle Coppens, Dirk Van den Heuvel, Peter Van der Donck, Tom Callewaert, Frank Meeussen, Erika De Bie, Kristof Eersels, Ellen Schouteden
Publikováno v:
Organic Process Research & Development; Apr2008, Vol. 12 Issue 3, p530-536, 7p