Zobrazeno 1 - 3
of 3
pro vyhledávání: '"Elie Amine Tabet"'
Autor:
Matthew Jude Sharp, Will L. Canoy, Kae M. Bullock, Eric Eugene Boros, Xiao-ming M. Zhou, Richard T. Matsuoka, Greg A. Erickson, Vassil I. Elitzin, Mark B. Mitchell, Matthew C. Salmon, David H. Igo, Nicole M. Deschamps, Daniel W. Reynolds, Andrew D. Brown, Gregory E. Peckham, Istvan Kaldor, Jennifer F. Toczko, Shannon Condon, Carpenter Andrew J, Elie Amine Tabet, Jing M. Fang, Biren K. Joshi, Lianming Michael Wu, Jeremy D. Cobb
Publikováno v:
Organic Process Research & Development. 20:1469-1475
Practical and scalable syntheses were developed that were used to prepare multikilogram batches of GSK1292263A (1) and GSK2041706A (15), two potent G protein-coupled receptor 119 (GPR119) agonists. Both syntheses employed relatively cheap and readily
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::82876eef78eb10aca7f33fb50ec6c1c0
https://doi.org/10.1021/acs.oprd.6b00157
https://doi.org/10.1021/acs.oprd.6b00157
Autor:
B. Liu, Vassil I. Elitzin, J. Powers, Daniel E. Patterson, Roman Davis, Elie Amine Tabet, Chong Pek Yoke, Matthew Salmons, M. Toczko, Mark A. Hatcher, Kae M. Bullock, M. Jackson
Publikováno v:
Topics in Catalysis. 55:446-452
Transition metal catalysis by Cu (CF3Cu), Ir (C–H activation), and Ru (ring-closing metathesis) were applied to prepare a complicated tetra substituted pyrazolopyridine drug candidate at GlaxoSmithKline. CuI/FSO2CF2CO2Me was utilized to install a C
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::86a49cac259c11c359deec285714ae7c
https://doi.org/10.1007/s11244-012-9809-z
https://doi.org/10.1007/s11244-012-9809-z
Autor:
Chong Pek Yoke, Mark A. Hatcher, Elie Amine Tabet, Vassil I. Elitzin, Roman Davis, Matthew Salmons, Bing Liu
Publikováno v:
Tetrahedron Letters. 53:6786-6788
Two syntheses of 7-trifluoromethylpyrazolo[1,5-a]pyridine dicarboxylate have been described. Approach A utilizes a nucleophilic addition of a trifluoromethyl group to N-p-toluenesulfonyliminopyridinium ylide followed by aromatization and subsequent c
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::0697a2a19b36a73e186f07ec52c5d866
https://doi.org/10.1016/j.tetlet.2012.09.136
https://doi.org/10.1016/j.tetlet.2012.09.136