Design, synthesis and mechanistic study of N-4-Piperazinyl Butyryl Thiazolidinedione derivatives of ciprofloxacin with Anticancer Activity via Topoisomerase I/II inhibition.

Autor: Aziz HA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, New Valley University, New Valley, 72511, Egypt.; Department of Medicinal Chemistry, Minia University, Minia, 61519, Egypt., El-Saghier AM; Department of Chemistry, Faculty of Science, Sohag University, Sohag, 82524, Egypt., Badr M; Department of Biochemistry, Faculty of Pharmacy, Menoufia University, Menoufia, Egypt., Elsadek BEM; Department of Biochemistry and Molecular Biology, Faculty of pharmacy, Assiut Branch, Al-Azhar University, Assiut, 71524, Egypt., Abuo-Rahma GEA; Department of Medicinal Chemistry, Minia University, Minia, 61519, Egypt. gamal.aborahma@mu.edu.eg.; Department of Pharmaceutical Chemistry, Deraya University, New Minya, 61768, Minia, Egypt. gamal.aborahma@mu.edu.eg.; Department of pharmaceutical chemistry, Deraya University, New Minia, 61768, Egypt. gamal.aborahma@mu.edu.eg., Shoman ME; Department of Medicinal Chemistry, Minia University, Minia, 61519, Egypt. mai_shoman@mu.edu.eg.

Publikováno v: Scientific reports [Sci Rep] 2024 Oct 15; Vol. 14 (1), pp. 24101. Date of Electronic Publication: 2024 Oct 15.

Correction: Synthesis, docking and biological evaluation of purine-5- N -isosteres as anti-inflammatory agents.

Autor: El-Saghier AM; Chemistry Department, Faculty of Science, Sohag University Sohag 282524 Egypt el.saghier@science.sohag.edu.eg., Enaili SS; Chemistry Department, Faculty of Science, Sohag University Sohag 282524 Egypt el.saghier@science.sohag.edu.eg.; Chemistry Department, Faculty of Science, Al Zawiya University Al Zawiya Libya., Abdou A; Chemistry Department, Faculty of Science, Sohag University Sohag 282524 Egypt el.saghier@science.sohag.edu.eg., Hamed AM; Chemistry Department, Faculty of Science, Sohag University Sohag 282524 Egypt el.saghier@science.sohag.edu.eg., Kadry AM; Chemistry Department, Faculty of Science, Sohag University Sohag 282524 Egypt el.saghier@science.sohag.edu.eg.

Publikováno v: RSC advances [RSC Adv] 2024 Jul 12; Vol. 14 (31), pp. 22091. Date of Electronic Publication: 2024 Jul 12 (Print Publication: 2024).

Thiadiazole/Thiadiazine Derivatives as Insecticidal Agent: Design, Synthesis, and Biological Assessment of 1,3,4-(Thiadiazine/Thiadiazole)-Benzenesulfonamide Derivatives as IGRs Analogues against Spodoptera littoralis .

Autor: El-Saghier AM; Chemistry Department, Faculty of Science, Sohag University, 82524 Sohag, Egypt., Enaili SS; Chemistry Department, Faculty of Science, Sohag University, 82524 Sohag, Egypt.; Chemistry Department, Faculty of Science, Al Zawia University, 16418 Al Zawia, Libya., Abdou A; Chemistry Department, Faculty of Science, Sohag University, 82524 Sohag, Egypt., Alzahrani AYA; Chemistry Department, Faculty of Science and Arts, King Khalid University, Mohail, 61421 Assir, Saudi Arabia., Ben Moussa S; Chemistry Department, Faculty of Science and Arts, King Khalid University, Mohail, 61421 Assir, Saudi Arabia., Gad MA; Research Institute of Plant Protection, Agricultural Research Center, 12619 Giza, Egypt., Kadry AM; Chemistry Department, Faculty of Science, Sohag University, 82524 Sohag, Egypt.

Publikováno v: Journal of agricultural and food chemistry [J Agric Food Chem] 2024 May 22; Vol. 72 (20), pp. 11369-11380. Date of Electronic Publication: 2024 May 10.

Green synthesis, biological and molecular docking of some novel sulfonamide thiadiazole derivatives as potential insecticidal against Spodoptera littoralis.

Autor: El-Saghier AM; Chemistry Department, Faculty of Science, Sohag University, Sohag, 282524, Egypt. el.saghier@science.sohag.edu.eg., Enaili SS; Chemistry Department, Faculty of Science, Sohag University, Sohag, 282524, Egypt.; Chemistry Department, Faculty of Science, Al Zawiya University, Al Zawiya, Libya., Kadry AM; Chemistry Department, Faculty of Science, Sohag University, Sohag, 282524, Egypt., Abdou A; Chemistry Department, Faculty of Science, Sohag University, Sohag, 282524, Egypt., Gad MA; Research Institute of Plant Protection, Agricultural Research Center, Giza, 12619, Egypt.

Publikováno v: Scientific reports [Sci Rep] 2023 Nov 06; Vol. 13 (1), pp. 19142. Date of Electronic Publication: 2023 Nov 06.

Novel 2-Acetamido-2-ylidene-4-imidazole Derivatives (El-Saghier Reaction): Green Synthesis, Biological Assessment, and Molecular Docking.

Autor: El-Saghier AM; Chemistry Department, Faculty of Science, Sohag University, Sohag 82524, Egypt., Abdou A; Chemistry Department, Faculty of Science, Sohag University, Sohag 82524, Egypt., Mohamed MAA; Chemistry Department, Faculty of Science, Sohag University, Sohag 82524, Egypt., Abd El-Lateef HM; Chemistry Department, Faculty of Science, Sohag University, Sohag 82524, Egypt.; Department of Chemistry, College of Science, King Faisal University, Al-Ahsa 31982, Saudi Arabia., Kadry AM; Chemistry Department, Faculty of Science, Sohag University, Sohag 82524, Egypt.

Publikováno v: ACS omega [ACS Omega] 2023 Aug 09; Vol. 8 (33), pp. 30519-30531. Date of Electronic Publication: 2023 Aug 09 (Print Publication: 2023).