Zobrazeno 1 - 10 of 20 pro vyhledávání: '"Eiichi Okezaki"'
1
Structure-Activity Relationship (SAR) Studies on Oxazolidinone Antibacterial Agents. 3. Synthesis and Evaluation of 5-Thiocarbamate Oxazolidinones
Autor: Eiichi Okezaki, Ryukou Tokuyama, Nobuhiko Iwasaki, Yoshiei Takahashi, Noriyuki Kado, Masatoshi Tsubouchi, Osamu Nagata, Yayoi Tomita
Publikováno v: Chemical and Pharmaceutical Bulletin. 49:361-367
A series of 5-thiocarbamate oxazolidinones was prepared and tested for in vitro and in vivo antibacterial activities. The results of in vitro antibacterial activity indicated that the 5-thiocarbamate group was a suitable substituent for the activity
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::80b5f5fc60cdf5de0d60850abdc2771f
https://doi.org/10.1248/cpb.49.361
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2
Spontaneous Myeloblastic Leukemia in a Young SD Rat
Autor: Eiichi Okezaki, Takeo Shimo, Yasuji Aoki, Osamu Nagata, Akemi Saito, Junichi Katayama
Publikováno v: Journal of Toxicologic Pathology. 13:123-126
A hematopoietic neoplasm was found in a 14-week-old male Sprague-Dawley (SD) rat. Blood smear examination revealed the existence of numerous blastic cells with large, round or oval nuclei, and scant pale cytoplasm containing no granules. At autopsy,
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::b9df059ea5ce90d93c13892a4cd7a135
https://doi.org/10.1293/tox.13.123
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3
Significance of Intraglomerular Expression of .ALPHA.-Smooth Muscle Actin, Desmin, and PDGF Receptor on Glomerulosclerosis in the Rat Remnant Kidney Model
Autor: Masafumi Ohshita, Takeo Shimo, Junichi Katayama, Eiichi Okezaki, Yasuji Aoki, Osamu Nagata, Akemi Saito
Publikováno v: Journal of Toxicologic Pathology. 11:229-234
To elucidate the possible pathomechanism of glomerulosclerosis by partial nephrectomy, male SD rats received 3/4 nephrectomy and were maintained without further treatment for 8 weeks (3/4 nephrectomized group). Another group received a sham operation
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_________::6eb426ef585d82b5736f59af052b45a9
https://doi.org/10.1293/tox.11.229
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9
In vitro antibacterial activities of new fluoroquinolones against clinical isolates of haemophilus influenzae with ciprofloxacin-resistance-associated alterations in GyrA and ParC
Autor: Eiichi Okezaki, Kazuhiro Tateda, Yoshie Takahashi, Yoshikazu Ishii, Yoshinari Watanabe, Satoshi Yoshizumi
Publikováno v: Chemotherapy. 50(6)
Background: The in vitro antimicrobial activities of new fluoroquinolones were tested against quinolone-resistant Haemophilus influenzae of clinical isolates. Methods: The nucleotide sequences of the gyrA and parC genes from three ciprofloxacin-resis
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::293b71ae768a5be73694868a57f4eb64
https://pubmed.ncbi.nlm.nih.gov/15608441
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10
Structure-activity relationship (SAR) studies on oxazolidinone antibacterial agents. 2. Relationship between lipophilicity and antibacterial activity in 5-thiocarbonyl oxazolidinones
Autor: Toshihiko Yoshida, Yoshiei Takahashi, Osamu Nagata, Nobuhiko Iwasaki, Noriyuki Kado, Yayoi Tomita, Ryukou Tokuyama, Eiichi Okezaki, Masatoshi Tsubouchi
Publikováno v: Chemicalpharmaceutical bulletin. 49(4)
5-Thiourea and 5-dithiocarbamate oxazolidinones were synthesized as a continuation of research on 5-thiocarbonyl oxazolidinone antibacterial agents considering the hydrophobic parameters of the molecule. The structure-activity relationship (SAR) stud
Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::730700ceb02fc471a4c64cd9a060c0fc
https://pubmed.ncbi.nlm.nih.gov/11310657
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