Zobrazeno 1 - 10
of 18
pro vyhledávání: '"E. Bourgier"'
Autor:
Andreas Marzinzik, Silvio Ofner, Jean-Michel Rondeau, Wolfgang Jahnke, Chrystelle Henry, S. Lehmann, E. Bourgier, Xavier Pelle, Jonathan Green, J. Constanze D. Hartwieg, Rene Hemmig, Simona Cotesta, Guido Bold, Frédéric Stauffer
Publikováno v:
Angewandte Chemie. 127:14783-14787
Die Wirksamkeit und Vertraglichkeit eines Medikaments kann verbessert werden, indem dieses gezielt an den gewunschten Wirkungsort gebracht wird. Bisphosphonate sind Prototypen derartiger Medikamente; allerdings ist ihre Affinitat zum Knochen eher zu
Autor:
Jean-Michel Rondeau, E. Bourgier, Marjo Götte, Johann Zimmermann, Armin Widmer, Steven J. Stout, Andreas Marzinzik, René Amstutz, Wolfgang Jahnke, S. Lehmann, Xavier Pelle, Christelle Henry, Frédéric Stauffer, Silvio Ofner, Simona Cotesta, Guido Bold, Thomas Zoller, J. Fraser Glickman, Thomas P. Roddy, J. Constanze D. Hartwieg
Publikováno v:
ChemMedChem. 10(11)
Farnesyl pyrophosphate synthase (FPPS) is an established target for the treatment of bone diseases, but also shows promise as an anticancer and anti-infective drug target. Currently available anti-FPPS drugs are active-site-directed bisphosphonate in
Autor:
Frédéric Stauffer, Jean-Michel Rondeau, Simona Cotesta, Jonathan Green, Rene Hemmig, J. Constanze D. Hartwieg, Guido Bold, Andreas Marzinzik, Xavier Pelle, Silvio Ofner, E. Bourgier, Chrystelle Henry, Wolfgang Jahnke, S. Lehmann
Publikováno v:
Angewandte Chemie (International ed. in English). 54(48)
Targeting drugs to their desired site of action can increase their safety and efficacy. Bisphosphonates are prototypical examples of drugs targeted to bone. However, bisphosphonate bone affinity is often considered too strong and cannot be significan
Autor:
Wolfgang Jahnke, Antonin V. Tutter, Qin Hao, Andras J. Bauer, Gregory A. Michaud, John A. Tallarico, Jean-Michel Rondeau, Michael Salcius, E. Bourgier, Jacob Raphael, Shu Li
Publikováno v:
Journal of biomolecular screening. 19(6)
Bioactive small molecules are an invaluable source of therapeutics and chemical probes for exploring biological pathways. Yet, significant hurdles in drug discovery often come from lacking a comprehensive view of the target(s) for both early tool mol
Publikováno v:
Bone. 38:60-61
Autor:
Francis Bitsch, M. Kroemer, Rene Hemmig, E. Bourgier, J.-M. Rondeau, Wolfgang Jahnke, S. Lehmann, Martin Geiser, André Strauss, S. Rieffel, J.R. Green, Paul Ramage
Publikováno v:
Acta Crystallographica Section A Foundations of Crystallography. 63:s119-s119
Autor:
Paul Ramage, André Strauss, M. Kroemer, Francis Bitsch, E. Bourgier, S. Rieffel, J.R. Green, J.-M. Rondeau, Martin Geiser, Wolfgang Jahnke, S. Lehmann, Rene Hemmig
Publikováno v:
Bone. 38:61
Autor:
Francis Bitsch, Martin Geiser, André Strauss, Rene Hemmig, J.-M. Rondeau, Wolfgang Jahnke, S. Lehmann, M. Kroemer, Paul Ramage, E. Bourgier, S. Rieffel, J.R. Green
Publikováno v:
Bone. 38:61
Publikováno v:
Bone. 38:44
Autor:
Paul Ramage, Martin Geiser, M. Kroemer, Jean-Michel Rondeau, S. Rieffel, André Strauss, Wolfgang Jahnke, S. Lehmann, E. Bourgier, Rene Hemmig, Jonathan Green, Francis Bitsch
Publikováno v:
ChemMedChem. 1:165-165