Zobrazeno 1 - 3
of 3
pro vyhledávání: '"Driss Qasmi"'
Autor:
Michèle Reboud-Ravaux, Nicole Boggetto, Bernard Badet, Loïc René, I. Vergely, Eve de Rosny, Driss Qasmi
Publikováno v:
Bioorganic & Medicinal Chemistry. 5:707-714
A series of novel synthetic peptides containing an N-terminal glyoxylyl function (CHOCO-) have been tested as inhibitors of HIV-1 protease. The N-glyoxylyl peptide CHOCO-Pro-Ile-Val-NH2, which fulfills the specificity requirements of the MA/CA protea
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f77da63a890ac6e7ec34280cf49e25d7
https://doi.org/10.1016/s0968-0896(97)00016-3
https://doi.org/10.1016/s0968-0896(97)00016-3
Autor:
Michel Vilkas, Driss Qasmi
Publikováno v:
Synthetic Communications. 20:2769-2773
A method of preparation of the title compound 1a avoiding the use of gaseous chlorine is described. Tetramethylthiuram disulfide 4 is oxidized with sulfuryl chloride to dime thyl thiocarbamoyl chloride 5, which is converted to 1a by means of phosphor
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::12d2656f406dcbd01265cea7afed11a7
https://doi.org/10.1080/00397919008051488
https://doi.org/10.1080/00397919008051488
Publikováno v:
Tetrahedron Letters. 35:4343-4344
Activated esters of glyoxylic acid di-isopropylthioacetal were prepared by conventional procedures and used in the Solid Phase Peptide Synthesis of N-glyoxylyl-peptides (CHOCO-Peptides).
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::aa40b2efe06012ac43e86977bc7d2b6d
https://doi.org/10.1016/s0040-4039(00)73349-1
https://doi.org/10.1016/s0040-4039(00)73349-1