Zobrazeno 1 - 10
of 84
pro vyhledávání: '"Donald T. Ward"'
Publikováno v:
Frontiers in Physiology, Vol 14 (2023)
As both a sensor of extracellular calcium (Ca2+o) concentration and a key controller of Ca2+o homeostasis, one of the most interesting properties of the calcium-sensing receptor (CaR) is its sensitivity to, and modulation by, ions and small ligands o
Externí odkaz:
https://doaj.org/article/0eaee1cbbf1b4c45bdc45d9c8ad21c45
Autor:
Patricia P. Centeno, Amanda Herberger, Hee-Chang Mun, Chialing Tu, Edward F. Nemeth, Wenhan Chang, Arthur D. Conigrave, Donald T. Ward
Publikováno v:
Nature Communications, Vol 10, Iss 1, Pp 1-12 (2019)
Elevated inorganic phosphate levels promote excessive parathyroid hormone secretion, which contributes to the aetiology of secondary hyperparathyroidism. Here, the authors show that phosphate directly inhibits the calcium-sensing receptor, the main r
Externí odkaz:
https://doaj.org/article/c08a3a761322408bb35d7a424c6b5065
Autor:
Cecilia Romagnoli, Preeti Sharma, Roberto Zonefrati, Gaia Palmini, Elena Lucattelli, Donald T. Ward, Isabella Ellinger, Marco Innocenti, Maria Luisa Brandi
Publikováno v:
International Journal of Molecular Sciences, Vol 22, Iss 14, p 7282 (2021)
Skeletal muscle has an outstanding capacity for regeneration in response to injuries, but there are disorders in which this process is seriously impaired, such as sarcopenia. Pharmacological treatments to restore muscle trophism are not available, th
Externí odkaz:
https://doaj.org/article/65cc040601504a59a2b349e600f02fff
Autor:
Polina Yarova, Donald T. Ward, Dolores Shoback, Daniela Riccardi, Katie Leach, Fadil Hannan, Arthur Conigrave, Wenhan Chang, Edward M. Brown, Hans Bräuner-Osborne, Daniel Bikle
Publikováno v:
IUPHAR/BPS Guide to Pharmacology CITE. 2023
The calcium-sensing receptor (CaS, provisional nomenclature as recommended by NC-IUPHAR [47] and subsequently updated [77]) responds to multiple endogenous ligands, including extracellular calcium and other divalent/trivalent cations, polyamines and
Autor:
Martin Schepelmann, Marianna Ranieri, Irene Lopez-Fernandez, Thomas S. Webberley, Sarah C. Brennan, Polina L. Yarova, Joao Graca, Umar-Khetaab Hanif, Christian Müller, Teresa Manhardt, Martina Salzmann, Helen Quasnichka, Sally A. Price, Donald T. Ward, Thierry Gilbert, Vladimir V. Matchkov, Robert A. Fenton, Amanda Herberger, Jenna Hwong, Christian Santa Maria, Chia-Ling Tu, Enikö Kallay, Giovanna Valenti, Wenhan Chang, Daniela Riccardi
Publikováno v:
J Am Soc Nephrol
Schepelmann, M, Ranieri, M, Lopez-Fernandez, I, Webberley, T S, Brennan, S C, Yarova, P L, Graca, J, Hanif, U-K, Müller, C, Manhardt, T, Salzmann, M, Quasnichka, H, Price, S A, Ward, D T, Gilbert, T, Matchkov, V V, Fenton, R A, Herberger, A, Hwong, J, Santa Maria, C, Tu, C-L, Kallay, E, Valenti, G, Chang, W & Riccardi, D 2022, ' Impaired Mineral Ion Metabolism in a Mouse Model of Targeted Calcium-Sensing Receptor (CaSR) Deletion from Vascular Smooth Muscle Cells ', Journal of the American Society of Nephrology : JASN, vol. 33, no. 7, pp. 1323-1340 . https://doi.org/10.1681/ASN.2021040585
Schepelmann, M, Ranieri, M, Lopez-Fernandez, I, Webberley, T S, Brennan, S C, Yarova, P L, Graca, J, Hanif, U-K, Müller, C, Manhardt, T, Salzmann, M, Quasnichka, H, Price, S A, Ward, D T, Gilbert, T, Matchkov, V V, Fenton, R A, Herberger, A, Hwong, J, Santa Maria, C, Tu, C-L, Kallay, E, Valenti, G, Chang, W & Riccardi, D 2022, ' Impaired Mineral Ion Metabolism in a Mouse Model of Targeted Calcium-Sensing Receptor (CaSR) Deletion from Vascular Smooth Muscle Cells ', Journal of the American Society of Nephrology : JASN . https://doi.org/10.1681/ASN.2021040585
Schepelmann, M, Ranieri, M, Lopez-Fernandez, I, Webberley, T S, Brennan, S C, Yarova, P L, Graca, J, Hanif, U-K, Müller, C, Manhardt, T, Salzmann, M, Quasnichka, H, Price, S A, Ward, D T, Gilbert, T, Matchkov, V V, Fenton, R A, Herberger, A, Hwong, J, Santa Maria, C, Tu, C-L, Kallay, E, Valenti, G, Chang, W & Riccardi, D 2022, ' Impaired Mineral Ion Metabolism in a Mouse Model of Targeted Calcium-Sensing Receptor (CaSR) Deletion from Vascular Smooth Muscle Cells ', Journal of the American Society of Nephrology : JASN, vol. 33, no. 7, pp. 1323-1340 . https://doi.org/10.1681/ASN.2021040585
Schepelmann, M, Ranieri, M, Lopez-Fernandez, I, Webberley, T S, Brennan, S C, Yarova, P L, Graca, J, Hanif, U-K, Müller, C, Manhardt, T, Salzmann, M, Quasnichka, H, Price, S A, Ward, D T, Gilbert, T, Matchkov, V V, Fenton, R A, Herberger, A, Hwong, J, Santa Maria, C, Tu, C-L, Kallay, E, Valenti, G, Chang, W & Riccardi, D 2022, ' Impaired Mineral Ion Metabolism in a Mouse Model of Targeted Calcium-Sensing Receptor (CaSR) Deletion from Vascular Smooth Muscle Cells ', Journal of the American Society of Nephrology : JASN . https://doi.org/10.1681/ASN.2021040585
BACKGROUND: Impaired mineral ion metabolism is a hallmark of CKD-metabolic bone disorder. It can lead to pathologic vascular calcification and is associated with an increased risk of cardiovascular mortality. Loss of calcium-sensing receptor (CaSR) e
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7a80a8762e559e8d9063bbc47564db68
https://europepmc.org/articles/PMC9257819/
https://europepmc.org/articles/PMC9257819/
Autor:
James Lai, Edward F. Nemeth, Kevin J. Martin, Jiahong Xu, Debra Drayer, Donald T. Ward, Carol Moore, William G. Goodman, Yun Chon
Publikováno v:
J Am Soc Nephrol
Goodman, W G, Ward, D T, Martin, K J, Drayer, D, Moore, C, Xu, J, Lai, J, Chon, Y & Nemeth, E F 2022, ' Activation of the Calcium Receptor by Calcimimetic Agents Is Preserved Despite Modest Attenuating Effects of Hyperphosphatemia ', Journal of the American Society of Nephrology : JASN, vol. 33, no. 1, pp. 201-212 . https://doi.org/10.1681/ASN.2021060825
Goodman, W G, Ward, D T, Martin, K J, Drayer, D, Moore, C, Xu, J, Lai, J, Chon, Y & Nemeth, E F 2022, ' Activation of the Calcium Receptor by Calcimimetic Agents Is Preserved Despite Modest Attenuating Effects of Hyperphosphatemia ', Journal of the American Society of Nephrology : JASN, vol. 33, no. 1, pp. 201-212 . https://doi.org/10.1681/ASN.2021060825
BACKGROUND: Phosphorus levels in the range seen clinically among patients undergoing dialysis have been reported to attenuate calcium receptor activation and modify parathyroid hormone (PTH) release from isolated parathyroid glands in vitro. Some cli
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b4159c89124255059d327b10b8253af7
https://europepmc.org/articles/PMC8763177/
https://europepmc.org/articles/PMC8763177/
Autor:
Nigel J. M. Birdsall, Stephen J Lolait, Hans-Jürgen Wester, Paul L. Chazot, Sadashiva S. Karnik, Simon D. Harding, Celine Valant, Stephen P.H. Alexander, Olivier Civelli, Zsolt Csaba, Mastgugu Horiuchi, Khuraijam Dhanachandra Singh, Theodore L. Goodfriend, Morley D. Hollenberg, Duuamene Nyimanu, Shlomo Melmed, G. Enrico Rovati, Xavier Norel, Leigh A. Stoddart, Klemens Kaupmann, Robyn Macrae, Nicholas D. Holliday, Deborah L. Segaloff, Justo P. Castaño, Tony Ngo, Gordon Dent, Jean-Martin Beaulieu, Thomas L Williams, Antonia Cianciulli, Paweł Kozielewicz, Xaria X. Li, Jyrki P. Kukkonen, Craig A. McArdle, John D. Lee, Philippe Rondard, Steven D. Douglas, Hubert Vaudry, Khaled A. Al-Hosaini, Nan Chiang, Bernhard Bettler, Giovanni Tulipano, Corinne Bousquet, Karen J. Gregory, Craig Gerard, Robert T. Jensen, Stefan Schulz, Rithwik Ramachandran, Ross A. D. Bathgate, Deepa Jonnalagadda, David M. Thal, Takio Kitazawa, Manisha Ray, Bice Chini, Thomas Unger, Marta Fumagalli, Jean-Pierre Vilardaga, Donald T. Ward, Roger G. Pertwee, Stefan Offermanns, Marvin C. Gershengorn, Marc Parmentier, Pieter Timmermans, Eamonn Kelly, Yukihiko Sugimoto, Hamiyet Unal, Vincenzo Mitolo, Alistair Mathie, Emma L. Veale, Andrew L. Gundlach, Anthony P. Davenport, Mark T. Quinn, Jérôme Leprince, Christa E. Müller, Geoffrey Burnstock, Akos Heinemann, Jacqueline R. Kemp, Richard D. Ye, Bernard Mouillac, Roger J. Summers, Raul R. Gainetdinov, Girolamo Calò, Philip N. Murphy, Amelie Lupp, Kalyan C. Tirupula, Walter G. Thomas, Julien Hanson, Ahsan Husain, Katie Leach, Lucie H. Clapp, Hans Bräuner-Osborne, Gunnar Schulte, Kenneth E. Bernstein, Jean Mazella, Torsten Schöneberg, Satoru Eguchi, Martin C. Michel, Maria Antonietta Panaro, Kevin J. Catt, Rainer K. Reinscheid, Hans-Jürgen Kreienkamp, Wayne R. Alexander, Emanuel Escher, Anne Marie O'Carroll, Magnus Bäck, Laurence J. Miller, Jane F. Armstrong, Chiara Ruzza, Trent M. Woodruff, Daniel Hoyer, Chengcan Yao, Maria P. Abbracchio, John A. Peters, Gary B. Willars, Jean-Philippe Pin, David Vaudry, Debbie L. Hay, François Boulay, Davide Lecca, Eric R. Prossnitz, Arthur Christopoulos, Victoria A. Blaho, Yasuyuki Kihara, Charles Kennedy, Christopher Southan, László Hunyady, Pascal Dournaud, Fernand Gobeil, Cyril Goudet, Charles N. Serhan, Claes Dahlgren, Jörg Hamann, Tobias Langenhan, Ralf Jockers, Nicholas M. Barnes, Jean-Louis Nahon, Richard L. Hauger, Adam J. Pawson, Gareth J. Sanger, Tung Fong, Susan E. Leeman, Elena Faccenda, Edward J. Filardo, Valerie P. Tan, Marc de Gasparo, Ji Ming Wang, Jamie A. Davies, Jerold Chun, Stefania Ceruti, Tadashi Inagami, Réjean Couture, Kenneth A. Jacobson, Patrick Vanderheyden, Adriaan P. IJzerman, Janet J. Maguire, Christopher S. Walker
Publikováno v:
British Journal of Pharmacology, 178, S27-S156. Wiley
Alexander, S P, Christopoulos, A, Davenport, A P, Kelly, E, Mathie, A, Peters, J A, Veale, E L, Armstrong, J F, Faccenda, E, Harding, S D, Pawson, A J, Southan, C, Davies, J A, Abbracchio, M P, Alexander, W, Al-Hosaini, K, Bäck, M, Barnes, N M, Bathgate, R, Beaulieu, J-M, Bernstein, K E, Bettler, B, Birdsall, N J M, Blaho, V, Boulay, F, Bousquet, C, Bräuner-Osborne, H, Burnstock, G, Caló, G, Castaño, J P, Catt, K J, Ceruti, S, Chazot, P, Chiang, N, Chini, B, Chun, J, Cianciulli, A, Civelli, O, Clapp, L H, Couture, R, Csaba, Z, Dahlgren, C, Dent, G, Singh, K D, Douglas, S D, Dournaud, P, Eguchi, S, Escher, E, Filardo, E J, Fong, T, Fumagalli, M, Gainetdinov, R R, Gasparo, M D, Gerard, C, Gershengorn, M, Gobeil, F, Goodfriend, T L, Goudet, C, Gregory, K J, Gundlach, A L, Hamann, J, Hanson, J, Hauger, R L, Hay, D L, Heinemann, A, Hollenberg, M D, Holliday, N D, Horiuchi, M, Hoyer, D, Hunyady, L, Husain, A, IJzerman, A P, Inagami, T, Jacobson, K A, Jensen, R T, Jockers, R, Jonnalagadda, D, Karnik, S, Kaupmann, K, Kemp, J, Kennedy, C, Kihara, Y, Kitazawa, T, Kozielewicz, P, Kreienkamp, H-J, Kukkonen, J P, Langenhan, T, Leach, K, Lecca, D, Lee, J D, Leeman, S E, Leprince, J, Li, X X, Williams, T L, Lolait, S J, Lupp, A, Macrae, R, Maguire, J, Mazella, J, McArdle, C A, Melmed, S, Michel, M C, Miller, L J, Mitolo, V, Mouillac, B, Müller, C E, Murphy, P, Nahon, J-L, Ngo, T, Norel, X, Nyimanu, D, O'Carroll, A-M, Offermanns, S, Panaro, M A, Parmentier, M, Pertwee, R G, Pin, J-P, Prossnitz, E R, Quinn, M, Ramachandran, R, Ray, M, Reinscheid, R K, Rondard, P, Rovati, G E, Ruzza, C, Sanger, G J, Schöneberg, T, Schulte, G, Schulz, S, Segaloff, D L, Serhan, C N, Stoddart, L A, Sugimoto, Y, Summers, R, Tan, V P, Thal, D, Thomas, W W, Timmermans, P B M W M, Tirupula, K, Tulipano, G, Unal, H, Unger, T, Valant, C, Vanderheyden, P, Vaudry, D, Vaudry, H, Vilardaga, J-P, Walker, C S, Wang, J M, Ward, D T, Wester, H-J, Willars, G B, Woodruff, T M, Yao, C & Ye, R D 2021, ' THE CONCISE GUIDE TO PHARMACOLOGY 2021/22 : G protein-coupled receptors ', British Journal of Pharmacology, vol. 178 Suppl 1, no. S1, pp. S27-S156 . https://doi.org/10.1111/bph.15538
British journal of pharmacology, 178(S1), S27-S156. Wiley-Blackwell
Alexander, S P, Christopoulos, A, Davenport, A P, Kelly, E, Mathie, A, Peters, J A, Veale, E L, Armstrong, J F, Faccenda, E, Harding, S D, Pawson, A J, Southan, C, Davies, J A, Abbracchio, M P, Alexander, W, Al-Hosaini, K, Bäck, M, Barnes, N M, Bathgate, R, Beaulieu, J-M, Bernstein, K E, Bettler, B, Birdsall, N J M, Blaho, V, Boulay, F, Bousquet, C, Bräuner-Osborne, H, Burnstock, G, Caló, G, Castaño, J P, Catt, K J, Ceruti, S, Chazot, P, Chiang, N, Chini, B, Chun, J, Cianciulli, A, Civelli, O, Clapp, L H, Couture, R, Csaba, Z, Dahlgren, C, Dent, G, Singh, K D, Douglas, S D, Dournaud, P, Eguchi, S, Escher, E, Filardo, E J, Fong, T, Fumagalli, M, Gainetdinov, R R, Gasparo, M D, Gerard, C, Gershengorn, M, Gobeil, F, Goodfriend, T L, Goudet, C, Gregory, K J, Gundlach, A L, Hamann, J, Hanson, J, Hauger, R L, Hay, D L, Heinemann, A, Hollenberg, M D, Holliday, N D, Horiuchi, M, Hoyer, D, Hunyady, L, Husain, A, IJzerman, A P, Inagami, T, Jacobson, K A, Jensen, R T, Jockers, R, Jonnalagadda, D, Karnik, S, Kaupmann, K, Kemp, J, Kennedy, C, Kihara, Y, Kitazawa, T, Kozielewicz, P, Kreienkamp, H-J, Kukkonen, J P, Langenhan, T, Leach, K, Lecca, D, Lee, J D, Leeman, S E, Leprince, J, Li, X X, Williams, T L, Lolait, S J, Lupp, A, Macrae, R, Maguire, J, Mazella, J, McArdle, C A, Melmed, S, Michel, M C, Miller, L J, Mitolo, V, Mouillac, B, Müller, C E, Murphy, P, Nahon, J-L, Ngo, T, Norel, X, Nyimanu, D, O'Carroll, A-M, Offermanns, S, Panaro, M A, Parmentier, M, Pertwee, R G, Pin, J-P, Prossnitz, E R, Quinn, M, Ramachandran, R, Ray, M, Reinscheid, R K, Rondard, P, Rovati, G E, Ruzza, C, Sanger, G J, Schöneberg, T, Schulte, G, Schulz, S, Segaloff, D L, Serhan, C N, Stoddart, L A, Sugimoto, Y, Summers, R, Tan, V P, Thal, D, Thomas, W W, Timmermans, P B M W M, Tirupula, K, Tulipano, G, Unal, H, Unger, T, Valant, C, Vanderheyden, P, Vaudry, D, Vaudry, H, Vilardaga, J-P, Walker, C S, Wang, J M, Ward, D T, Wester, H-J, Willars, G B, Woodruff, T M, Yao, C & Ye, R D 2021, ' THE CONCISE GUIDE TO PHARMACOLOGY 2021/22 : G protein-coupled receptors ', British Journal of Pharmacology, vol. 178, no. S1, pp. S27-S156 . https://doi.org/10.1111/bph.15538
Alexander, S P, Christopoulos, A, Davenport, A P, Kelly, E, Mathie, A, Peters, J A, Veale, E L, Armstrong, J F, Faccenda, E, Harding, S D, Pawson, A J, Southan, C, Davies, J A, Abbracchio, M P, Alexander, W, Al-Hosaini, K, Bäck, M, Barnes, N M, Bathgate, R, Beaulieu, J-M, Bernstein, K E, Bettler, B, Birdsall, N J M, Blaho, V, Boulay, F, Bousquet, C, Bräuner-Osborne, H, Burnstock, G, Caló, G, Castaño, J P, Catt, K J, Ceruti, S, Chazot, P, Chiang, N, Chini, B, Chun, J, Cianciulli, A, Civelli, O, Clapp, L H, Couture, R, Csaba, Z, Dahlgren, C, Dent, G, Singh, K D, Douglas, S D, Dournaud, P, Eguchi, S, Escher, E, Filardo, E J, Fong, T, Fumagalli, M, Gainetdinov, R R, Gasparo, M D, Gerard, C, Gershengorn, M, Gobeil, F, Goodfriend, T L, Goudet, C, Gregory, K J, Gundlach, A L, Hamann, J, Hanson, J, Hauger, R L, Hay, D L, Heinemann, A, Hollenberg, M D, Holliday, N D, Horiuchi, M, Hoyer, D, Hunyady, L, Husain, A, IJzerman, A P, Inagami, T, Jacobson, K A, Jensen, R T, Jockers, R, Jonnalagadda, D, Karnik, S, Kaupmann, K, Kemp, J, Kennedy, C, Kihara, Y, Kitazawa, T, Kozielewicz, P, Kreienkamp, H-J, Kukkonen, J P, Langenhan, T, Leach, K, Lecca, D, Lee, J D, Leeman, S E, Leprince, J, Li, X X, Williams, T L, Lolait, S J, Lupp, A, Macrae, R, Maguire, J, Mazella, J, McArdle, C A, Melmed, S, Michel, M C, Miller, L J, Mitolo, V, Mouillac, B, Müller, C E, Murphy, P, Nahon, J-L, Ngo, T, Norel, X, Nyimanu, D, O'Carroll, A-M, Offermanns, S, Panaro, M A, Parmentier, M, Pertwee, R G, Pin, J-P, Prossnitz, E R, Quinn, M, Ramachandran, R, Ray, M, Reinscheid, R K, Rondard, P, Rovati, G E, Ruzza, C, Sanger, G J, Schöneberg, T, Schulte, G, Schulz, S, Segaloff, D L, Serhan, C N, Stoddart, L A, Sugimoto, Y, Summers, R, Tan, V P, Thal, D, Thomas, W W, Timmermans, P B M W M, Tirupula, K, Tulipano, G, Unal, H, Unger, T, Valant, C, Vanderheyden, P, Vaudry, D, Vaudry, H, Vilardaga, J-P, Walker, C S, Wang, J M, Ward, D T, Wester, H-J, Willars, G B, Woodruff, T M, Yao, C & Ye, R D 2021, ' THE CONCISE GUIDE TO PHARMACOLOGY 2021/22 : G protein-coupled receptors ', British Journal of Pharmacology, vol. 178 Suppl 1, no. S1, pp. S27-S156 . https://doi.org/10.1111/bph.15538
British journal of pharmacology, 178(S1), S27-S156. Wiley-Blackwell
Alexander, S P, Christopoulos, A, Davenport, A P, Kelly, E, Mathie, A, Peters, J A, Veale, E L, Armstrong, J F, Faccenda, E, Harding, S D, Pawson, A J, Southan, C, Davies, J A, Abbracchio, M P, Alexander, W, Al-Hosaini, K, Bäck, M, Barnes, N M, Bathgate, R, Beaulieu, J-M, Bernstein, K E, Bettler, B, Birdsall, N J M, Blaho, V, Boulay, F, Bousquet, C, Bräuner-Osborne, H, Burnstock, G, Caló, G, Castaño, J P, Catt, K J, Ceruti, S, Chazot, P, Chiang, N, Chini, B, Chun, J, Cianciulli, A, Civelli, O, Clapp, L H, Couture, R, Csaba, Z, Dahlgren, C, Dent, G, Singh, K D, Douglas, S D, Dournaud, P, Eguchi, S, Escher, E, Filardo, E J, Fong, T, Fumagalli, M, Gainetdinov, R R, Gasparo, M D, Gerard, C, Gershengorn, M, Gobeil, F, Goodfriend, T L, Goudet, C, Gregory, K J, Gundlach, A L, Hamann, J, Hanson, J, Hauger, R L, Hay, D L, Heinemann, A, Hollenberg, M D, Holliday, N D, Horiuchi, M, Hoyer, D, Hunyady, L, Husain, A, IJzerman, A P, Inagami, T, Jacobson, K A, Jensen, R T, Jockers, R, Jonnalagadda, D, Karnik, S, Kaupmann, K, Kemp, J, Kennedy, C, Kihara, Y, Kitazawa, T, Kozielewicz, P, Kreienkamp, H-J, Kukkonen, J P, Langenhan, T, Leach, K, Lecca, D, Lee, J D, Leeman, S E, Leprince, J, Li, X X, Williams, T L, Lolait, S J, Lupp, A, Macrae, R, Maguire, J, Mazella, J, McArdle, C A, Melmed, S, Michel, M C, Miller, L J, Mitolo, V, Mouillac, B, Müller, C E, Murphy, P, Nahon, J-L, Ngo, T, Norel, X, Nyimanu, D, O'Carroll, A-M, Offermanns, S, Panaro, M A, Parmentier, M, Pertwee, R G, Pin, J-P, Prossnitz, E R, Quinn, M, Ramachandran, R, Ray, M, Reinscheid, R K, Rondard, P, Rovati, G E, Ruzza, C, Sanger, G J, Schöneberg, T, Schulte, G, Schulz, S, Segaloff, D L, Serhan, C N, Stoddart, L A, Sugimoto, Y, Summers, R, Tan, V P, Thal, D, Thomas, W W, Timmermans, P B M W M, Tirupula, K, Tulipano, G, Unal, H, Unger, T, Valant, C, Vanderheyden, P, Vaudry, D, Vaudry, H, Vilardaga, J-P, Walker, C S, Wang, J M, Ward, D T, Wester, H-J, Willars, G B, Woodruff, T M, Yao, C & Ye, R D 2021, ' THE CONCISE GUIDE TO PHARMACOLOGY 2021/22 : G protein-coupled receptors ', British Journal of Pharmacology, vol. 178, no. S1, pp. S27-S156 . https://doi.org/10.1111/bph.15538
The Concise Guide to PHARMACOLOGY 2021/22 is the fifth in this series of biennial publications. The Concise Guide provides concise overviews, mostly in tabular format, of the key properties of nearly 1900 human drug targets with an emphasis on select
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::eef5f3d1320e3d9fb87604fe0e7987c5
https://cris.maastrichtuniversity.nl/en/publications/e6053af4-7c66-44a3-97bc-f7b87d1745a9
https://cris.maastrichtuniversity.nl/en/publications/e6053af4-7c66-44a3-97bc-f7b87d1745a9
Autor:
Polina Yarova, Daniel D. Bikle, Donald T. Ward, Edward M. Brown, Dolores M. Shoback, Fadil Hannan, Hans Bräuner-Osborne, Daniela Riccardi, Arthur D. Conigrave, Katie Leach, Wenhan Chang
Publikováno v:
IUPHAR/BPS Guide to Pharmacology CITE. 2021
The calcium-sensing receptor (CaS, provisional nomenclature as recommended by NC-IUPHAR [47] and subsequently updated [77]) responds to multiple endogenous ligands, including extracellular calcium and other divalent/trivalent cations, polyamines and
Publikováno v:
Molecular Pharmacology
Ward, D 2019, ' Identification of Serine-875 as an Inhibitory Phosphorylation Site in the Calcium-Sensing Receptor. ', Molecular pharmacology . https://doi.org/10.1124/mol.119.116178
Ward, D 2019, ' Identification of Serine-875 as an Inhibitory Phosphorylation Site in the Calcium-Sensing Receptor. ', Molecular pharmacology . https://doi.org/10.1124/mol.119.116178
The calcium-sensing receptor (CaS) is the principal controller of extracellular calcium (Ca2+o) homeostasis and is inhibited in vitro and in vivo by protein kinase C (PKC)-mediated phosphorylation at CaRT888. However, PKC inhibition enhances signalli
Autor:
Arthur D. Conigrave, Thor C. Møller, Hans Bräuner-Osborne, Andrew N. Keller, Daniela Riccardi, Katie Leach, Donald T. Ward, Enikö Kállay, Fadil M. Hannan, Rebecca S. Mason, Tracy M. Josephs, Rajesh V. Thakker
Publikováno v:
Leach, K, Hannan, F M, Josephs, T M, Keller, A N, Møller, T C, Ward, D T, Kallay, E, Mason, R S, Thakker, R V, Riccardi, D, Conigrave, A D & Bräuner-Osborne, H 2020, ' International Union of Basic and Clinical Pharmacology. CVIII. Calcium-Sensing Receptor Nomenclature, Pharmacology, and Function ', Pharmacological Reviews, vol. 72, no. 3, pp. 558-604 . https://doi.org/10.1124/pr.119.018531
Pharmacological Reviews
Pharmacol Rev
Pharmacological Reviews
Pharmacol Rev
The calcium-sensing receptor (CaSR) is a class C G protein-coupled receptor that responds to multiple endogenous agonists and allosteric modulators, including divalent and trivalent cations, L-amino acids, γ-glutamyl peptides, polyamines, polycation
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::172ef793c4bcbce0c405d4a538a416f0
https://ora.ox.ac.uk/objects/uuid:36ba0adf-bb2b-4474-a8fa-928bf788b385
https://ora.ox.ac.uk/objects/uuid:36ba0adf-bb2b-4474-a8fa-928bf788b385