Výsledky vyhledávání - "Dmitry G. Tentler"

5-Chloro-2-thiophenyl-1,2,3-triazolylmethyldihydroquinolines as dual inhibitors of Mycobacterium tuberculosis and influenza virus: Synthesis and evaluation

Autor: Vagolu Siva Krishna, Alexandrina S. Volobueva, Dharmarajan Sriram, Sandeep Kumar Marvadi, Vladimir V. Zarubaev, Ekaterina O. Sinegubova, Dmitry G. Tentler, Yana L Esaulkova, Srinivas Kantevari, Anna A. Muryleva

Publikováno v: Bioorganic & Medicinal Chemistry Letters. 29:2664-2669

This study describes synthesis and evaluation of novel 5-Chloro-2-thiophenyl-1,2,3-triazolylmethyldihydroquinolines 7a-o as dual inhibitors of Mycobacterium tuberculosis and influenza virus. Huisgen’s [3+2] dipolar cycloaddition of 6-(azidomethyl)-

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::00be46294ecdfeb39d5b61aa7861a2f9
https://doi.org/10.1016/j.bmcl.2019.07.040

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Synthesis of novel derivatives of 7,8-dihydro-6H-imidazo[2,1-b][1,3]benzothiazol-5-one and their virus-inhibiting activity against influenza A virus

Autor: Dmitry G. Tentler, Irina N. Lavrenteva, Nagaraju Chirra, Srinivas Kantevari, Anastasia V. Galochkina, Rakesh K Bollikanda, Vladimir V. Zarubaev, Alexander V. Slita

Publikováno v: Archiv der Pharmazie. 352(2)

Influenza remains a highly pathogenic and hardly controlled human infection. The ability of selecting drug-resistant variants necessitates the search and development of novel anti-influenza drugs. Herein, we describe the synthesis and evaluation of a

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::606f4a32d0c0131af237fa2c0362ee27
https://pubmed.ncbi.nlm.nih.gov/30520524

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