Zobrazeno 1 - 10
of 29
pro vyhledávání: '"Diseroad, Benjamin A."'
Autor:
Price, Louise S., McMahon, Jennifer A., Lingireddy, Sreenivas R., Lau, Suk-Fai, Diseroad, Benjamin A., Price, Sarah L., Reutzel-Edens, Susan M.
Publikováno v:
In Journal of Molecular Structure 25 December 2014 1078:26-42
Autor:
Robert F. Bruns, Qi Chen, Paloma Vidal, John Mehnert Schaus, Charles R. Yang, Stephen N. Mitchell, Steven Marc Massey, Nuria Diaz, Xushan Wang, David Andrew Coates, Rebecca A. Wright, Beverly A. Heinz, Kevin Matthew Gardinier, Greg Stephenson, James P. Beck, Rajni M. Bhardwaj, Julie F. Falcone, Bruce A. Dressman, Deanna L Maren, Anette M. Johansson, David Michael Remick, Jeff W. Cramer, Cohen Michael Philip, Brian Morgan Watson, Jeffery Richardson, Kjell Svensson, Xin Zhou, Erik James Hembre, Serge Louis Boulet, Reinhard Matthew Robert, Daniel S. Richards, Junliang Hao, David M. Bender, Guy Carter, Christopher David Beadle, Brian G. Getman, Wolfangel Craig Daniel, Diseroad Benjamin Alan, Jason K. Myers, Joseph H. Krushinski, David Edward Tupper
Publikováno v:
Journal of Medicinal Chemistry. 62:8711-8732
Clinical development of catechol-based orthosteric agonists of the dopamine D1 receptor has thus far been unsuccessful due to multiple challenges. To address these issues, we identified LY3154207 (...
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::5a353395d3c6f7ca6dfa78c95a347dd4
https://doi.org/10.1021/acs.jmedchem.9b01234
https://doi.org/10.1021/acs.jmedchem.9b01234
Autor:
Baertschi, Steven W., Brunner, Heiko, Bunnell, Charles A., Cooke, Gary G., Diseroad, Benjamin, Dorman, Douglas E., Jansen, Patrick J. *, Kemp, Craig A.J., Maple, Steven R., McCune, Karen A., Speakman, Jeffrey L.
Publikováno v:
In Journal of Pharmaceutical Sciences February 2008 97(2):883-892
Autor:
Frances Lu, Bryan G. Johnson, Daniel Ursu, Joan H. Carter, Lisa M. Broad, Kofi Adragni, Shane Atwell, Jing Wang, David K. Clawson, Beverly A. Heinz, Steven P. Swanson, James A. Monn, Qi Chen, Helene E. Sanger, David B. Shaw, Steven Marc Massey, Xushan Wang, Marijane Russell, Steven S. Henry, Junliang Hao, Rajni M. Bhardwaj, Diseroad Benjamin Alan, David L. McKinzie, Brian G. Getman, John T. Catlow
Publikováno v:
Journal of Medicinal Chemistry. 61:2303-2328
Multiple therapeutic opportunities have been suggested for compounds capable of selective activation of metabotropic glutamate 3 (mGlu3) receptors, but small molecule tools are lacking. As part of our ongoing efforts to identify potent, selective, an
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::34fd3a986aac486e41e6ea738f1a4465
https://doi.org/10.1021/acs.jmedchem.7b01481
https://doi.org/10.1021/acs.jmedchem.7b01481
Akademický článek
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Autor:
Steven D. Kahl, Kelly L. Wilbur, Warshawsky Alan M, Jayana Pankaj Lineswala, Siddaramaiah Cr, Pranab Maiti, Sweetana Stephanie Ann, Diseroad Benjamin Alan, Lisa A. Adams, Yanyun Chen, Richard W. Zink, Anne Reifel Miller, Grace L. Neathery, Anjana Patel Lewis, Over Cabrera, Alison N. Campbell, Guemalli R. Cardona, Nathan Yumibe, Keyue Chen, Keith A. Otto, Cecilia Bouaichi, Xiaosu Ma, Chafiq Hamdouchi, Amy C. DeBaillie, Chahrzad Montrose-Rafizadeh
Publikováno v:
Journal of medicinal chemistry. 61(3)
As a part of our program to identify potent GPR40 agonists capable of being dosed orally once daily in humans, we incorporated fused heterocycles into our recently disclosed spiropiperidine and tetrahydroquinoline acid derivatives 1, 2, and 3 with th
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ba33126a14f55ea8f6b1d4d12011e1a1
https://pubmed.ncbi.nlm.nih.gov/29236497
https://pubmed.ncbi.nlm.nih.gov/29236497
Autor:
Sreenivas R. Lingireddy, Suk-Fai Lau, Diseroad Benjamin Alan, Sarah L. Price, Jennifer A. McMahon, Louise S. Price, Susan M. Reutzel-Edens
Publikováno v:
Journal of Molecular Structure. 1078:26-42
Almost twenty years after the crystal polymorphism of tazofelone was first studied at Lilly, the compound was revisited by calculating the crystal energy landscape and complementing the calculations with experimental work for calibration purposes. Th
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4e5219090b381e82e64746cfddb522fb
https://doi.org/10.1016/j.molstruc.2014.01.014
https://doi.org/10.1016/j.molstruc.2014.01.014
Akademický článek
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Akademický článek
Tento výsledek nelze pro nepřihlášené uživatele zobrazit.
K zobrazení výsledku je třeba se přihlásit.
K zobrazení výsledku je třeba se přihlásit.
Autor:
Diseroad Benjamin Alan, Raj Suryanarayanan, Gregory A. Stephenson, Naveen K. Thakral, Aktham Aburub, Timothy Andrew Woods, Jeffrey A. Peterson, Robert J. Behme
Publikováno v:
Molecular pharmaceutics. 13(12)
Disproportionation propensity of salts (HCl, HBr, heminapadisylate) and adipic acid cocrystal of corticotropin releasing hormone receptor-1 antagonist was studied using model free kinetics. Using thermogravimetic weight loss profile or heat flow curv
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f4aef677085b85cb39b5161e8cabdf33
https://pubmed.ncbi.nlm.nih.gov/27766882
https://pubmed.ncbi.nlm.nih.gov/27766882