Zobrazeno 1 - 10
of 42
pro vyhledávání: '"Dinesh Chimmanamada"'
Autor:
Weiwen Ying, Dinesh Chimmanamada, Richard C. Bates, Sami Osman, Noriaki Tatsuta, Takayo Inoue, Igor Astsaturov, Vladimir Khazak, Chaohua Zhang, Suqin He, Jaime Acquaviva, Manuel Sequeira, Luisa Shin Ogawa, Jim Sang, John-Paul Jimenez, Junyi Zhang, Donald L. Smith, David A. Proia
Plasma stability assay
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::16576181af7e8366e9045c5c59596d21
https://doi.org/10.1158/1535-7163.22506805.v1
https://doi.org/10.1158/1535-7163.22506805.v1
Autor:
Weiwen Ying, Dinesh Chimmanamada, Richard C. Bates, Sami Osman, Noriaki Tatsuta, Takayo Inoue, Igor Astsaturov, Vladimir Khazak, Chaohua Zhang, Suqin He, Jaime Acquaviva, Manuel Sequeira, Luisa Shin Ogawa, Jim Sang, John-Paul Jimenez, Junyi Zhang, Donald L. Smith, David A. Proia
The clinical benefits of chemotherapy are commonly offset by insufficient drug exposures, narrow safety margins, and/or systemic toxicities. Over recent decades, a number of conjugate-based targeting approaches designed to overcome these limitations
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::96f9bc9986cb6f4f2bd1cefcc5ef01b1
https://doi.org/10.1158/1535-7163.c.6538495.v1
https://doi.org/10.1158/1535-7163.c.6538495.v1
Autor:
Weiwen Ying, Dinesh Chimmanamada, Richard C. Bates, Sami Osman, Noriaki Tatsuta, Takayo Inoue, Igor Astsaturov, Vladimir Khazak, Chaohua Zhang, Suqin He, Jaime Acquaviva, Manuel Sequeira, Luisa Shin Ogawa, Jim Sang, John-Paul Jimenez, Junyi Zhang, Donald L. Smith, David A. Proia
HSP90 binding promotes the intracellular retention of HSP90 inhibitor-BODIPY probes in tumor cell lines.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::014519ba899563e4f1919adfd2ea71c7
https://doi.org/10.1158/1535-7163.22506823.v1
https://doi.org/10.1158/1535-7163.22506823.v1
Autor:
Weiwen Ying, Dinesh Chimmanamada, Richard C. Bates, Sami Osman, Noriaki Tatsuta, Takayo Inoue, Igor Astsaturov, Vladimir Khazak, Chaohua Zhang, Suqin He, Jaime Acquaviva, Manuel Sequeira, Luisa Shin Ogawa, Jim Sang, John-Paul Jimenez, Junyi Zhang, Donald L. Smith, David A. Proia
Cross-species plasma stability of STA-12-8666 as a function of time
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b22d113ac9042df40dbd281707cfed92
https://doi.org/10.1158/1535-7163.22506802.v1
https://doi.org/10.1158/1535-7163.22506802.v1
Autor:
Weiwen Ying, Dinesh Chimmanamada, Richard C. Bates, Sami Osman, Noriaki Tatsuta, Takayo Inoue, Igor Astsaturov, Vladimir Khazak, Chaohua Zhang, Suqin He, Jaime Acquaviva, Manuel Sequeira, Luisa Shin Ogawa, Jim Sang, John-Paul Jimenez, Junyi Zhang, Donald L. Smith, David A. Proia
Supplementary Figure Legends
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::56261c0c5a501d4768495f05342f25f7
https://doi.org/10.1158/1535-7163.22506808.v1
https://doi.org/10.1158/1535-7163.22506808.v1
Publikováno v:
In Tetrahedron 16 June 2000 56(25):4267-4277
Autor:
Masazumi Nagai, Mitsunori Ono, Shoujun Chen, Minghu Song, Teresa Przewloka, Jun Jiang, David James, Lijun Sun, Dinesh Chimmanamada, Zhi-Qiang Xia, Keizo Koya, Shijie Zhang, Rongzhen Lu, Elena Kostik
Publikováno v:
Med. Chem. Commun.. 2:176-180
A series of novel indolizine 2-oxoacetamides were designed and synthesized as PDE4 inhibitors. Preliminary SAR of this new class of compounds revealed key structural features required for high potency. Compounds 1ab and 2a are among the most potent i
Autor:
Teresa Przewloka, David James, Shijie Zhang, Shoujun Chen, Hao Li, Elena Kostik, Lijun Sun, Keizo Koya, Dinesh Chimmanamada, Zhi-Qiang Xia
Publikováno v:
Tetrahedron Letters. 48:5739-5742
A number of 3-acylated indolizines were synthesized in good to excellent yields by a newly established reaction between picolinium salts and the methylsulfate salt of A (R = Me), the adduct formed from DMF–Me2SO4 as the key reagent. The low cost, s
Autor:
John-Paul Jimenez, Vladimir Khazak, Chaohua Zhang, Luisa Shin Ogawa, Suqin He, Igor Astsaturov, Dinesh Chimmanamada, Donald L. Smith, Noriaki Tatsuta, Jaime Acquaviva, Weiwen Ying, Manuel Sequeira, Sami Osman, Junyi Zhang, Takayo Inoue, David A. Proia, Jim Sang, Richard C. Bates
Publikováno v:
Molecular cancer therapeutics. 14(11)
The clinical benefits of chemotherapy are commonly offset by insufficient drug exposures, narrow safety margins, and/or systemic toxicities. Over recent decades, a number of conjugate-based targeting approaches designed to overcome these limitations
Autor:
Weiwen Ying, Dinesh Chimmanamada, Anna S. Nikonova, David A. Proia, Brian L. Egleston, Ilya G. Serebriiskii, Harvey Hensley, Tatiana Kent, Kathy Q. Cai, Tamina Seeger-Nukpezah, Erica A. Golemis
Publikováno v:
Proceedings of the National Academy of Sciences of the United States of America. 110(31)
Autosomal dominant polycystic kidney disease (ADPKD) is a progressive genetic syndrome with an incidence of 1:500 in the population, arising from inherited mutations in the genes for polycystic kidney disease 1 ( PKD1 ) or polycystic kidney disease 2