Zobrazeno 1 - 8
of 8
pro vyhledávání: '"Dieter Seidelmann"'
Autor:
Martin Krüger, Martin Haberey, Andreas Huth, Josef Brüggen, Jürgen Mestan, Guido Bold, Gerhard Siemeister, Jeanette Marjorie Wood, Paul W. Manley, Dieter Seidelmann, Eckhard Ottow, Karl-Heinz Thierauch, Andreas Menrad, Thomas F. Meyer, Christian Schnell, Pascal Furet
Publikováno v:
Journal of medicinal chemistry. 45(26)
Two readily synthesized anthranilamide, VEGF receptor tyrosine kinase inhibitors have been prepared and evaluated as angiogenesis inhibitors. 2-[(4-Pyridyl)methyl]amino-N-[3-(trifluoromethyl)phenyl]benzamide (5) and N-3-isoquinolinyl-2-[(4-pyridinylm
Autor:
Volker Bähr, Wolfgang Oelkers, S. Diederich, Patrick Burkhardt, C Bumke-Vogt, Ekkehard Eigendorff, Dieter Seidelmann, Peter Esperling, Marina Rochel, Marcus Quinkler
Publikováno v:
The Journal of clinical endocrinology and metabolism. 87(12)
The 11β-hydroxysteroid dehydrogenase (11β-HSD) system plays a pivotal role in glucocorticoid (GC) and mineralocorticoid (MC) action. Although 11β-HSD activities are important determinants for the efficacy of synthetic MCs and GCs, corresponding ph
Autor:
Branislava Mitrovic, Herbert Schneider, Helmut Wachtel, Eckhard Ottow, Daryl Faulds, H. Daniel Perez, Dieter Seidelmann, Jenny Tse, Meredith Halks-Miller, David Asarnow, Harald Dinter, Henry Laurent, Vincent K. Tuohy, Peter Esperling, Gerald Kirsch, James Onuffer
Publikováno v:
Journal of neuroimmunology. 108(1-2)
Experimental autoimmune encephalomyelitis (EAE) is an autoimmune disease with pathological features reminiscent of those seen in multiple sclerosis and thus serves as an animal model for this disease. Inhibition of type IV phosphodiesterase (PDE IV)
Publikováno v:
Psychopharmacology. 121(1)
The present series of experiments examined the effects of five benzodiazepine receptor (BZR) partial inverse agonists on the behaviour of rats on an elevated plus maze. The drugs were tested in a standard plus maze with 3-cm walls added to the open a
Publikováno v:
HETEROCYCLES. 48:31
Publikováno v:
Justus Liebigs Annalen der Chemie. 714:43-56
Zum Aufbau der tetrasubstituierten Athane 5–9 wird von den bekannten Hexan-Derivaten 10 und 11 sowie vom Butan-Derivat 12 ausgegangen. Die Funfring-Verbindungen 5–7 konnen – nach Erzeugung unterschiedlicher Sauerstoff-Funktionen – durch oxyda
Autor:
Wolfgang Kehr, Claus Braestrup, Dieter Seidelmann, Ralph Schmiechen, Herbert Schneider, Leif Helth Jensen, Erling N. Petersen, Tage Honore, David N. Stephens
Publikováno v:
Psychopharmacology. 83(3)
We describe here biochemical and pharmacological effects of the β-carboline ZK 93426, a new and potent benzodiazepine (BZ) receptor antagonist. ZK 93426 was compared with Ro 15-1788 and CGS 8216, two compounds previously described as BZ receptor ant
Autor:
Elke Schoffers, Dieter Seidelmann, Ulrich Eder, Dieter Rahtz, Andreas Huth, Ralph Schmischen, G殤ter Neef
Publikováno v:
HETEROCYCLES. 20:1295