Synthesis of new C-6 alkyliden penicillin derivatives as β-lactamase inhibitors

Autor: Di Giacomo, B ^*, Tarzia, G, Bedini, A, Gatti, G, Bartoccini, F, Balsamini, C, Tontini, A, Baffone, W, Di Modugno, E, Felici, A

Publikováno v: In Il Farmaco 2002 57(4):273-283

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Reassessing the melatonin pharmacophore--enantiomeric resolution, pharmacological activity, structure analysis, and molecular modeling of a constrained chiral melatonin analogue

Autor: Rivara S., Diamantini G., Di Giacomo B., Lamba D., Gatti G., Lucini V., Pannacci M., Mor M., Spadoni G., Tarzia G.

Publikováno v: Bioorganic & medicinal chemistry
14 (2006): 3383–3391.
info:cnr-pdr/source/autori:Rivara S., Diamantini G., Di Giacomo B., Lamba D., Gatti G., Lucini V., Pannacci M., Mor M., Spadoni G., Tarzia G./titolo:Reassessing the melatonin pharmacophore--enantiomeric resolution, pharmacological activity, structure analysis, and molecular modeling of a constrained chiral melatonin analogue/doi:/rivista:Bioorganic & medicinal chemistry (Print)/anno:2006/pagina_da:3383/pagina_a:3391/intervallo_pagine:3383–3391/volume:14

3-(Acetylaminomethyl)-2-(ethoxycarbonyl)-6-methoxy-1,3,4,5-tetrahydrobenzo[cd]indole (2) is a rigid melatonin analogue that as a racemate displays about the same affinity and intrinsic activity of melatonin (1) in in vitro experiments. We report here

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=cnr_________::27f298ea7715d20482eb7bbf4d9d7365
http://www.cnr.it/prodotto/i/19618

1-(2-Alkanamidoethyl)-6-methoxyindole derivatives: a new class of potent indole melatonin analogues

Autor: D. Esposti, Bojidar Stankov, Gilberto Spadoni, Marilou Pannacci, Lucini, Franco Fraschini, Romolo Nonno, G. Tarzia, Giuseppe Diamantini, Di Giacomo B

Publikováno v: Journal of medicinal chemistry. 40(13)

A new series of indole melatonin analogues, bearing the amido ethyl side chain attached at the N-1 position of the indole nucleus, were synthesized and tested for their affinity for the melatonin receptor isolated from quail optic tecta in a series o

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7e08ce4f39c60e475f7e4a51750832b4
https://pubmed.ncbi.nlm.nih.gov/9207941

Robot-based dedicated measuring system with data redundancy for profile inspection.

Autor: Di Giacomo, B., Tsunaki, R.H., Paziani, F.T.

Publikováno v: 2005 IEEE/RSJ International Conference on Intelligent Robots & Systems; 2005, p1392-1395, 4p