Zobrazeno 1 - 10
of 41
pro vyhledávání: '"Derek J. Cash"'
Autor:
Tamás Blandl, Edit Simon-Trompler, Julianna Kardos, Ilona Kovács, Miklós Simonyi, Gábor Dörnyei, Csaba Szántay, Nguyen D Luyen, Gábor Blaskó, Derek J. Cash
Publikováno v:
European Journal of Pharmacology. 337:83-86
Enantiomers of norbicuculline, (+)[1S,9R] and (-)[1R,9S]erythro-1-[1'-(4',5'-methylenedioxyphthalidyl)]-6,7-meth ylenedioxy-1,2,3,4-tetrahydroisoquinoline and of the N-methyl derivatives {(+)[1S,9R] and (-)[1R,9S]bicuculline} were found to inhibit th
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::59ee5508bf69d656e3a160f72ad7d2fd
https://doi.org/10.1016/s0014-2999(97)01267-3
https://doi.org/10.1016/s0014-2999(97)01267-3
Autor:
Eszter Gács-Baitz, Gábor Blaskó, Miklós Simonyi, Tamás Blandl, Derek J. Cash, József Kardos, Cs. Szantay, N. D. Luyen, Gábor Dörnyei
Publikováno v:
European Journal of Medicinal Chemistry. 31:761-765
Summary Synthesis of erythro -(±)-[1 SR ,9 RS ]-norbicuculline and threo -(±)-[1 SR ,9 SR ]-noradlumidine from piperonal was performed using Bischler-Napieralski cyclization as a key step. Resolution gave rise to (+)-[1 S ,9 R ]-norbicuculline ([1
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ddb21b78b6d121611a67096d63ea45fe
https://doi.org/10.1016/0223-5234(96)83969-9
https://doi.org/10.1016/0223-5234(96)83969-9
Autor:
Derek J. Cash, Peter Serfozo
Publikováno v:
European Journal of Biochemistry. 228:498-505
l-Glutamate-mediated transmembrane influx of 22Na+ into a native membrane vesicle preparation from rat hippocampus was resolved into components due to glutamate receptor and Na+-glutamate symport, by kinetic analysis and pharmacological specificity.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2b3612a41f993ee24020332ad3b21516
https://doi.org/10.1111/j.1432-1033.1995.0498n.x
https://doi.org/10.1111/j.1432-1033.1995.0498n.x
Autor:
Cs. Szantay, G. Blasko, Miklós Simonyi, Derek J. Cash, Tamás Blandl, Gabor Doernyei, N. D. Luyen, József Kardos, Eszter Gács-Baitz
Publikováno v:
ChemInform. 28
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::6615dd98d43b206d439f2fe7bf02cfe7
https://doi.org/10.1002/chin.199708211
https://doi.org/10.1002/chin.199708211
Autor:
Peter Serfozo, Derek J. Cash
Publikováno v:
FEBS Letters. 310:55-59
Chlordiazepoxide (CDPX) enhanced the rate of chloride exchange mediated by the major GABAA receptor found on sealed native membrane vesicles from rat cerebral cortex. The initial rate constant for chloride exchange for this receptor, (JA), a measure
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::da13453cecf2f9347057e3a575fa9410
https://doi.org/10.1016/0014-5793(92)81145-c
https://doi.org/10.1016/0014-5793(92)81145-c
Publikováno v:
The Journal of Membrane Biology. 145
We used the short-lived radionuclide, ^(82)Br^− to follow γ-aminobutyrate (GABA) receptor-mediated halide exchange into membrane vesicles from rat cerebral cortex in millisecond and second time regions using quench-flow technique. The radioisotope
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::acb32c04e46ac06e5675f3944e5cad4d
https://doi.org/10.1007/bf00232717
https://doi.org/10.1007/bf00232717
Modulation of GABA flux across rat brain membranes resolved by a rapid quenched incubation technique
Publikováno v:
Neuroscience letters. 182(1)
The progress and inhibition of [3H]GABA influx in native plasma membrane vesicles from the rat cerebral cortex was studied on a subsecond to minute time scale under different conditions by applying a rapid quenched incubation technique. In the absenc
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ff8c32af935e5c516919c32f454ccb11
https://pubmed.ncbi.nlm.nih.gov/7891893
https://pubmed.ncbi.nlm.nih.gov/7891893
Publikováno v:
Journal of biochemical and biophysical methods. 23(2)
Modifications to a quench-flow apparatus are described which allow a rapid, in-line filter assay with immediate washing, in conditions to give minimum background. A design for an effluent spout is presented, which decelerates the liquid by a large fa
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::99ac420439e2c88e174e07bebd606fda
https://pubmed.ncbi.nlm.nih.gov/1658108
https://pubmed.ncbi.nlm.nih.gov/1658108
Publikováno v:
Biochemical and Biophysical Research Communications. 92:896-904
The dependence of acetylcholine receptor-controlled transmembrane ion flux on carbamylcholine concentration was measured in the msec time region, using membrane vesicles and a quench flow technique. 4 Measurements were made: (1) transmembrane ion inf
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::005240071e0c8cfbe06e7ef318f1db14
https://doi.org/10.1016/0006-291x(80)90787-1
https://doi.org/10.1016/0006-291x(80)90787-1
Autor:
George P. Hess, Jayant B. Udgaonkar, Elena B. Pasquale, Derek J. Cash, Kunio Takeyasu, Matthew C. Severski
Publikováno v:
Biochemistry. 22:5967-5973
Suberyldicholine-induced ion translocation in the millisecond time region in acetylcholine receptor rich membrane vesicles prepared from the electric organ of Electrophorus electricus was investigated in eel Ringer's solution, pH 7.0, 1 degree C. A q
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8ea8358f84c6f2756f3a06c521105c18
https://doi.org/10.1021/bi00294a041
https://doi.org/10.1021/bi00294a041