Zobrazeno 1 - 10
of 13
pro vyhledávání: '"Dechert-Schmitt AM"'
Autor:
Lees JA; Discovery Sciences, Medicine Design, Pfizer Inc., Groton, CT, USA., Dias JM; Discovery Sciences, Medicine Design, Pfizer Inc., Groton, CT, USA., Rajamohan F; Discovery Sciences, Medicine Design, Pfizer Inc., Groton, CT, USA., Fortin JP; Internal Medicine Research Unit, Pfizer Inc., Cambridge, MA, USA., O'Connor R; Discovery Sciences, Medicine Design, Pfizer Inc., Groton, CT, USA., Kong JX; Internal Medicine Research Unit, Pfizer Inc., Cambridge, MA, USA., Hughes EAG; Internal Medicine Research Unit, Pfizer Inc., Cambridge, MA, USA., Fisher EL; Internal Medicine, Medicine Design, Pfizer Inc., Groton, CT, USA., Tuttle JB; Internal Medicine, Medicine Design, Pfizer Inc., Cambridge, MA, USA., Lovett G; Internal Medicine, Medicine Design, Pfizer Inc., Cambridge, MA, USA., Kormos BL; Internal Medicine, Medicine Design, Pfizer Inc., Cambridge, MA, USA., Unwalla RJ; Internal Medicine, Medicine Design, Pfizer Inc., Cambridge, MA, USA., Zhang L; Internal Medicine, Medicine Design, Pfizer Inc., Cambridge, MA, USA., Dechert Schmitt AM; Internal Medicine, Medicine Design, Pfizer Inc., Groton, CT, USA., Zhou D; Internal Medicine, Medicine Design, Pfizer Inc., Groton, CT, USA., Moran M; Internal Medicine, Medicine Design, Pfizer Inc., Groton, CT, USA., Stevens KA; Internal Medicine Research Unit, Pfizer Inc., Cambridge, MA, USA., Fennell KF; Discovery Sciences, Medicine Design, Pfizer Inc., Groton, CT, USA., Varghese AE; Discovery Sciences, Medicine Design, Pfizer Inc., Groton, CT, USA., Maxwell A; Discovery Sciences, Medicine Design, Pfizer Inc., Groton, CT, USA., Cote EE; Discovery Sciences, Medicine Design, Pfizer Inc., Groton, CT, USA., Zhang Y; Internal Medicine, Medicine Design, Pfizer Inc., Cambridge, MA, USA., Han S; Discovery Sciences, Medicine Design, Pfizer Inc., Groton, CT, USA. seungil.han@pfizer.com.
Publikováno v:
Nature communications [Nat Commun] 2023 Sep 23; Vol. 14 (1), pp. 5938. Date of Electronic Publication: 2023 Sep 23.
Autor:
Aspnes GE; Pfizer Medicine Design, Pfizer Inc., Eastern Point Road, Groton, CT 06340, USA., Coffey SB; Pfizer Medicine Design, Pfizer Inc., Eastern Point Road, Groton, CT 06340, USA., Darout E; Pfizer Medicine Design, Pfizer Inc., Eastern Point Road, Groton, CT 06340, USA., Dechert-Schmitt AM; Pfizer Medicine Design, Pfizer Inc., Eastern Point Road, Groton, CT 06340, USA., Dullea RG; Pfizer Medicine Design, Pfizer Inc., Eastern Point Road, Groton, CT 06340, USA., Kamlet AS; Pfizer Medicine Design, Pfizer Inc., Eastern Point Road, Groton, CT 06340, USA., Limberakis C; Pfizer Medicine Design, Pfizer Inc., Eastern Point Road, Groton, CT 06340, USA., Londregan AT; Pfizer Medicine Design, Pfizer Inc., Eastern Point Road, Groton, CT 06340, USA., McClure KF; Pfizer Medicine Design, Pfizer Inc., Eastern Point Road, Groton, CT 06340, USA., Menhaji-Klotz E; Pfizer Medicine Design, Pfizer Inc., Eastern Point Road, Groton, CT 06340, USA., Piotrowski DW; Pfizer Medicine Design, Pfizer Inc., Eastern Point Road, Groton, CT 06340, USA. Electronic address: david.w.piotrowski@comcast.net., Polivkova J; Pfizer Medicine Design, Pfizer Inc., Eastern Point Road, Groton, CT 06340, USA., Raymer B; Pfizer Medicine Design, Pfizer Inc., Eastern Point Road, Groton, CT 06340, USA., Ruggeri RB; Pfizer Medicine Design, Pfizer Inc., Eastern Point Road, Groton, CT 06340, USA., Salatto CT; Pfizer Medicine Design, Pfizer Inc., Eastern Point Road, Groton, CT 06340, USA., Tu M; Pfizer Medicine Design, Pfizer Inc., Eastern Point Road, Groton, CT 06340, USA., Wei L; Pfizer Medicine Design, Pfizer Inc., Eastern Point Road, Groton, CT 06340, USA., Xiao J; Pfizer Medicine Design, Pfizer Inc., Eastern Point Road, Groton, CT 06340, USA.
Publikováno v:
Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2023 Aug 15; Vol. 92, pp. 129394. Date of Electronic Publication: 2023 Jun 26.
Autor:
Futatsugi K; Pfizer Inc. Medicine Design, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Cabral S; Pfizer Inc. Medicine Design, Eastern Point Road, Groton, Connecticut 06340, United States., Kung DW; Pfizer Inc. Medicine Design, Eastern Point Road, Groton, Connecticut 06340, United States., Huard K; Pfizer Inc. Medicine Design, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Lee E; Pfizer Inc. Medicine Design, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Boehm M; Pfizer Inc. Medicine Design, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Bauman J; Pfizer Inc. Medicine Design, Eastern Point Road, Groton, Connecticut 06340, United States., Clark RW; Pfizer Inc. Internal Medicine Research Unit, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Coffey SB; Pfizer Inc. Medicine Design, Eastern Point Road, Groton, Connecticut 06340, United States., Crowley C; Pfizer Inc. Internal Medicine Research Unit, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Dechert-Schmitt AM; Pfizer Inc. Medicine Design, Eastern Point Road, Groton, Connecticut 06340, United States., Dowling MS; Pfizer Inc. Medicine Design, Eastern Point Road, Groton, Connecticut 06340, United States., Dullea R; Pfizer Inc. Internal Medicine Research Unit, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Gosset JR; Pfizer Inc. Medicine Design, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Kalgutkar AS; Pfizer Inc. Medicine Design, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Kou K; Pfizer Inc. Internal Medicine Research Unit, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Li Q; Pfizer Inc. Medicine Design, Eastern Point Road, Groton, Connecticut 06340, United States., Lian Y; Pfizer Inc. Medicine Design, Eastern Point Road, Groton, Connecticut 06340, United States., Loria PM; Pfizer Inc. Medicine Design, Eastern Point Road, Groton, Connecticut 06340, United States., Londregan AT; Pfizer Inc. Medicine Design, Eastern Point Road, Groton, Connecticut 06340, United States., Niosi M; Pfizer Inc. Medicine Design, Eastern Point Road, Groton, Connecticut 06340, United States., Orozco C; Pfizer Inc. Medicine Design, Eastern Point Road, Groton, Connecticut 06340, United States., Pettersen JC; Pfizer Inc. Drug Safety R&D, Eastern Point Road, Groton, Connecticut 06340, United States., Pfefferkorn JA; Pfizer Inc. Internal Medicine Research Unit, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Polivkova J; Pfizer Inc. Medicine Design, Eastern Point Road, Groton, Connecticut 06340, United States., Ross TT; Pfizer Inc. Internal Medicine Research Unit, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Sharma R; Pfizer Inc. Medicine Design, Eastern Point Road, Groton, Connecticut 06340, United States., Stock IA; Pfizer Inc. Medicine Design, Eastern Point Road, Groton, Connecticut 06340, United States., Tesz G; Pfizer Inc. Internal Medicine Research Unit, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Wisniewska H; Pfizer Inc. Medicine Design, Eastern Point Road, Groton, Connecticut 06340, United States., Goodwin B; Pfizer Inc. Internal Medicine Research Unit, 1 Portland Street, Cambridge, Massachusetts 02139, United States., Price DA; Pfizer Inc. Medicine Design, 1 Portland Street, Cambridge, Massachusetts 02139, United States.
Publikováno v:
Journal of medicinal chemistry [J Med Chem] 2022 Nov 24; Vol. 65 (22), pp. 15000-15013. Date of Electronic Publication: 2022 Nov 02.
Autor:
Zhang M; Department of Chemistry, Boston College, 2609 Beacon Street, Chestnut Hill, MA 02467, USA., Xu P; Department of Chemistry, Boston College, 2609 Beacon Street, Chestnut Hill, MA 02467, USA., Vendola AJ; Department of Chemistry, Boston College, 2609 Beacon Street, Chestnut Hill, MA 02467, USA., Allais C; Pfizer Worldwide Research and Development, Eastern Point Road, Groton, CT 06430, USA., Dechert Schmitt AM; Pfizer Worldwide Research and Development, Eastern Point Road, Groton, CT 06430, USA., Singer RA; Pfizer Worldwide Research and Development, Eastern Point Road, Groton, CT 06430, USA., Morken JP; Department of Chemistry, Boston College, 2609 Beacon Street, Chestnut Hill, MA 02467, USA.
Publikováno v:
Angewandte Chemie (International ed. in English) [Angew Chem Int Ed Engl] 2022 Jul 25; Vol. 61 (30), pp. e202205454. Date of Electronic Publication: 2022 Jun 08.
Autor:
Chen TQ; Merck Center for Catalysis at Princeton University, Princeton, New Jersey 08544, United States., Pedersen PS; Merck Center for Catalysis at Princeton University, Princeton, New Jersey 08544, United States., Dow NW; Merck Center for Catalysis at Princeton University, Princeton, New Jersey 08544, United States., Fayad R; Department of Chemistry, North Carolina State University, Raleigh, North Carolina 27695, United States., Hauke CE; Department of Chemistry, North Carolina State University, Raleigh, North Carolina 27695, United States., Rosko MC; Department of Chemistry, North Carolina State University, Raleigh, North Carolina 27695, United States., Danilov EO; Department of Chemistry, North Carolina State University, Raleigh, North Carolina 27695, United States., Blakemore DC; Worldwide Research and Development, Pfizer, Inc., Eastern Point Road, Groton, Connecticut 06340, United States., Dechert-Schmitt AM; Worldwide Research and Development, Pfizer, Inc., Eastern Point Road, Groton, Connecticut 06340, United States., Knauber T; Worldwide Research and Development, Pfizer, Inc., Eastern Point Road, Groton, Connecticut 06340, United States., Castellano FN; Department of Chemistry, North Carolina State University, Raleigh, North Carolina 27695, United States., MacMillan DWC; Merck Center for Catalysis at Princeton University, Princeton, New Jersey 08544, United States.
Publikováno v:
Journal of the American Chemical Society [J Am Chem Soc] 2022 May 11; Vol. 144 (18), pp. 8296-8305. Date of Electronic Publication: 2022 Apr 29.
Autor:
Dow NW; Merck Center for Catalysis at Princeton University, Princeton, New Jersey 08544, United States., Pedersen PS; Merck Center for Catalysis at Princeton University, Princeton, New Jersey 08544, United States., Chen TQ; Merck Center for Catalysis at Princeton University, Princeton, New Jersey 08544, United States., Blakemore DC; Worldwide Research and Development, Pfizer, Inc., Eastern Point Road, Groton, Connecticut 06340, United States., Dechert-Schmitt AM; Worldwide Research and Development, Pfizer, Inc., Eastern Point Road, Groton, Connecticut 06340, United States., Knauber T; Worldwide Research and Development, Pfizer, Inc., Eastern Point Road, Groton, Connecticut 06340, United States., MacMillan DWC; Merck Center for Catalysis at Princeton University, Princeton, New Jersey 08544, United States.
Publikováno v:
Journal of the American Chemical Society [J Am Chem Soc] 2022 Apr 13; Vol. 144 (14), pp. 6163-6172. Date of Electronic Publication: 2022 Apr 04.
Liver-Targeted Small-Molecule Inhibitors of Proprotein Convertase Subtilisin/Kexin Type 9 Synthesis.
Autor:
McClure KF; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Piotrowski DW; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Petersen D; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Wei L; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Xiao J; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Londregan AT; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Kamlet AS; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Dechert-Schmitt AM; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Raymer B; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Ruggeri RB; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Canterbury D; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Limberakis C; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Liras S; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., DaSilva-Jardine P, Dullea RG; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Loria PM; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Reidich B; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Salatto CT; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Eng H; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Kimoto E; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Atkinson K; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., King-Ahmad A; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Scott D; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Beaumont K; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Chabot JR; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Bolt MW; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Maresca K; Department of Medicinal Chemistry, Pfizer Inc, 1 Portland Street, Cambridge, MA, 02139, USA., Dahl K; Department of Clinical Neuroscience, Center for Psychiatry Research, Karolinska Institutet, Stockholm, Sweden., Arakawa R; Department of Clinical Neuroscience, Center for Psychiatry Research, Karolinska Institutet, Stockholm, Sweden., Takano A; Department of Clinical Neuroscience, Center for Psychiatry Research, Karolinska Institutet, Stockholm, Sweden., Halldin C; Department of Clinical Neuroscience, Center for Psychiatry Research, Karolinska Institutet, Stockholm, Sweden.
Publikováno v:
Angewandte Chemie (International ed. in English) [Angew Chem Int Ed Engl] 2017 Dec 18; Vol. 56 (51), pp. 16218-16222. Date of Electronic Publication: 2017 Nov 24.
Autor:
Piotrowski DW; Worldwide Medicinal Chemistry, Pfizer, Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Kamlet AS; Worldwide Medicinal Chemistry, Pfizer, Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Dechert-Schmitt AM; Worldwide Medicinal Chemistry, Pfizer, Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Yan J; Worldwide Medicinal Chemistry, Pfizer, Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Brandt TA; Chemical Research and Development, Pfizer, Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Xiao J; Worldwide Medicinal Chemistry, Pfizer, Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Wei L; Worldwide Medicinal Chemistry, Pfizer, Inc. , Eastern Point Road, Groton, Connecticut 06340, United States., Barrila MT; Chemical Research and Development, Pfizer, Inc. , Eastern Point Road, Groton, Connecticut 06340, United States.
Publikováno v:
Journal of the American Chemical Society [J Am Chem Soc] 2016 Apr 13; Vol. 138 (14), pp. 4818-23. Date of Electronic Publication: 2016 Mar 30.
Autor:
Tsai AS; Pfizer Worldwide Medicinal Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States., Curto JM; Pfizer Worldwide Medicinal Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States., Rocke BN; Pfizer Worldwide Medicinal Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States., Dechert-Schmitt AM; Pfizer Worldwide Medicinal Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States., Ingle GK; Pfizer Worldwide Medicinal Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States., Mascitti V; Pfizer Worldwide Medicinal Chemistry, Eastern Point Road, Groton, Connecticut 06340, United States.
Publikováno v:
Organic letters [Org Lett] 2016 Feb 05; Vol. 18 (3), pp. 508-11. Date of Electronic Publication: 2016 Jan 15.
Autor:
Dechert-Schmitt AM; University of Texas at Austin, Department of Chemistry and Biochemistry, 105 E 24th St., Welch Hall A5300, Austin, TX 78712-1165, USA. mkrische@mail.utexas.edu., Schmitt DC, Gao X, Itoh T, Krische MJ
Publikováno v:
Natural product reports [Nat Prod Rep] 2014 Apr; Vol. 31 (4), pp. 504-13. Date of Electronic Publication: 2014 Feb 11.