Zobrazeno 1 - 10
of 13
pro vyhledávání: '"Davide Baraldi"'
Publikováno v:
Synthetic Communications. 29:3125-3135
This paper deals with a novel and versatile synthetic approach for the introduction of a functionalized ethynyl side chain at the C-3 position of the 2-carboxyindole nucleus. The key step of this process is represented by the coupling reaction betwee
Publikováno v:
ChemInform. 23
Adducts AlCl 3 .RCOC1 undergo highly regioselective self- and cross-condensation. 4-Hydroxy-2-pyrones and 2-acetyl-indan-1,3-diones are synthesized in good yields.
Publikováno v:
ChemInform. 24
Autor:
Xiaochun Tao, Franca Bigi, Giuseppe Casnati, Davide Baraldi, Giovanni Sartori, Raimondo Maggi
Publikováno v:
ChemInform. 25
The synthesis of a series of persubstituted 4-hydroxy-2-pyrones 6 by regioselective «one-pot» cyclotrimerization of aliphatic acyl chlorides promoted by aluminum chloride is reported
Publikováno v:
ChemInform. 29
Publikováno v:
ChemInform. 30
This paper deals with a novel and versatile synthetic approach for the introduction of a functionalized ethynyl side chain at the C-3 position of the 2-carboxyindole nucleus. The key step of this process is represented by the coupling reaction betwee
Autor:
Davide Baraldi, Paola Gastaldi, Alfredo Cugola, Daniele Donati, Simone Giacobbe, Gianluca Araldi, Giorgio Pentassuglia, Romano Di Fabio, Fabrizio Micheli
Publikováno v:
ChemInform. 33
Publikováno v:
J. Chem. Soc., Perkin Trans. 1. :2985-2988
Variously substituted indan-1,3-diones have been regioselectively prepared in a one-pot synthesis by sequential cross-condensation–cycloacylation of aromatic acyl chlorides and acetyl chloride or malonyl dichloride, electrophilic acylation of aroma
Publikováno v:
Tetrahedron Letters. 32:2153-2156
Adducts AlCl 3 .RCOC1 undergo highly regioselective self- and cross-condensation. 4-Hydroxy-2-pyrones and 2-acetyl-indan-1,3-diones are synthesized in good yields.
Autor:
Daniele Donati, Paola Gastaldi, Romano Di Fabio, Simone Giacobbe, Alfredo Cugola, Gianluca Araldi, Davide Baraldi, Giorgio Pentassuglia, Fabrizio Micheli
Publikováno v:
Farmaco (Societa chimica italiana : 1989). 56(10)
After the identification of GV150526, the indole-2-carboxylate template was further explored in order to identify novel potential anti-stroke agents. In particular, the SAR of the side chain present at the C-3 position of the indole nucleus was widel