Zobrazeno 1 - 10
of 20
pro vyhledávání: '"David Dailler"'
Publikováno v:
Communications Chemistry, Vol 4, Iss 1, Pp 1-11 (2021)
Fidaxomicin is a narrow spectrum antibiotic, and broadening its activity through structural modification could provide new antibiotics. Here semi-synthetic derivatives are prepared through site-selective esterification and allylic substitution to eff
Externí odkaz:
https://doaj.org/article/c32e82beff5d448d939c9d14cc5a1314
Publikováno v:
Journal of the American Chemical Society. 144:11069-11074
Under Rh-catalyzed conditions, secondary amines and anilines function as directing groups to facilitate regioselective C-C bond activation of nonactivated cyclopropanes. The resulting amino-stabilized rhodacycles undergo carbonylative C-N bond format
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1812f00fd872aaa5e5e7c20808ce2299
https://doi.org/10.1021/jacs.2c02921
https://doi.org/10.1021/jacs.2c02921
Publikováno v:
Communications Chemistry, Vol 4, Iss 1, Pp 1-11 (2021)
Fidaxomicin (FDX) is a marketed antibiotic for the treatment Clostridium difficile infections (CDI). Although showing interesting antibacterial properties against many Gram-positive bacteria, the application of this antibiotic is currently limited to
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4d22dfb3abfecd6992f0a732259e2e06
https://doi.org/10.26434/chemrxiv.12593429
https://doi.org/10.26434/chemrxiv.12593429
Autor:
Florian Zellweger, Olivier Baudoin, Markus Neuburger, Christophe Salomé, David Dailler, Eric Clot, Ronan Rocaboy
Publikováno v:
Angewandte Chemie International Edition
Angewandte Chemie International Edition, Wiley-VCH Verlag, 2018, 57 (37), pp.12131-12135. ⟨10.1002/anie.201807097⟩
Angewandte Chemie International Edition, Wiley-VCH Verlag, 2018, 57 (37), pp.12131-12135. ⟨10.1002/anie.201807097⟩
The Pd0 -catalyzed C(sp3 )-H arylation of 2-bromo-N-methylanilides leads to unstable benzazetidine intermediates that rearrange to benzoxazines through 4π electrocyclic ring-opening and 6π electrocyclization. The introduction of a bulky, non-activa
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1402845f948fb5acac0eb8ec41a44e48
https://doi.org/10.1002/ange.201807097
https://doi.org/10.1002/ange.201807097
Autor:
Julien C. Vantourout, Olivier Baudoin, David Dailler, Philipp M. Holstein, Anthony Millet, Janah Shaya
Publikováno v:
Angewandte Chemie International Edition. 55:2805-2809
A variety of strained α-alkylidene-γ-lactams were synthesized by palladium(0)-catalyzed intramolecular C(sp(3) )-H alkenylation from easily accessible acyclic and monocyclic bromoalkene precursors. These lactams are valuable intermediates for acces
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::aaf0dc41703de8778b4a07794c9cbc0b
https://doi.org/10.1002/anie.201511457
https://doi.org/10.1002/anie.201511457
Autor:
Philipp M. Holstein, David Dailler, Julien Vantourout, Janah Shaya, Anthony Millet, Olivier Baudoin
Publikováno v:
Angewandte Chemie. 128:2855-2859
A variety of strained α-alkylidene-γ-lactams were synthesized by palladium(0)-catalyzed intramolecular C(sp3)−H alkenylation from easily accessible acyclic and monocyclic bromoalkene precursors. These lactams are valuable intermediates for access
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d9dc2b0ddfcc7f1d7b750936b6d398de
https://doi.org/10.1002/ange.201511457
https://doi.org/10.1002/ange.201511457
Autor:
Ronan, Rocaboy, David, Dailler, Florian, Zellweger, Markus, Neuburger, Christophe, Salomé, Eric, Clot, Olivier, Baudoin
Publikováno v:
Angewandte Chemie (International ed. in English). 57(37)
The Pd
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::926a8c645bbdc420d109d0749395f6f9
https://pubmed.ncbi.nlm.nih.gov/30020559
https://pubmed.ncbi.nlm.nih.gov/30020559
Publikováno v:
Organic letters. 20(3)
An expedient synthesis of lycorine alkaloids is reported using a palladium(0)-catalyzed double C-X/C-H arylation as the key step. The selectivity of this reaction was controlled through the judicious choice of the two halogen atoms, and its generalit
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::6ab256188625345b8c2cac64e2c3e159
https://pubmed.ncbi.nlm.nih.gov/29345138
https://pubmed.ncbi.nlm.nih.gov/29345138
An expedient synthesis of lycorine alkaloids is reported using a palladium(0)-catalyzed double C–X/C–H arylation as the key step. The selectivity of this reaction was controlled through the judicious choice of the two halogen atoms, and its gener
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2151b1de6340dc7f8710662026d84904
https://edoc.unibas.ch/62336/
https://edoc.unibas.ch/62336/
Publikováno v:
Angewandte Chemie. 127:5001-5004
An efficient and scalable access to the aeruginosin family of marine natural products, which exhibit potent inhibitory activity against serine proteases, is reported. This synthesis was enabled by the strategic use of two different, recently implemen
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::52c31363f5c0d9398858714197abf115
https://doi.org/10.1002/ange.201500066
https://doi.org/10.1002/ange.201500066