Zobrazeno 1 - 10
of 28
pro vyhledávání: '"David B. Rusterholz"'
Publikováno v:
Molecules, Vol 2, Iss 5, Pp 80-86 (1997)
Two 1,3,8,10-undecatetraenes were synthesized to test the viability of the intramolecular radical cation induced Diels-Alder reaction in the diene - diene format. Cyclization was successful only for the substituted tetraene with the lower oxidation p
Externí odkaz:
https://doaj.org/article/d81afa2a92024dbca89e9e7e563ed12b
Autor:
Luciano De Petrocellis, David B. Rusterholz, Giorgio Ortar, Eric M. Serum, Aniello Schiano Moriello
Publikováno v:
Bioorganic & medicinal chemistry letters
25 (2015): 2285–2290. doi:10.1016/j.bmcl.2015.04.032
info:cnr-pdr/source/autori:De Petrocellis, Luciano; Ortar, Giorgio; Schiano Moriello, Aniello; Serum, Eric M.; Rusterholz, David B./titolo:Structure-activity relationships of the prototypical TRPM8 agonist icilin/doi:10.1016%2Fj.bmcl.2015.04.032/rivista:Bioorganic & medicinal chemistry letters (Print)/anno:2015/pagina_da:2285/pagina_a:2290/intervallo_pagine:2285–2290/volume:25
25 (2015): 2285–2290. doi:10.1016/j.bmcl.2015.04.032
info:cnr-pdr/source/autori:De Petrocellis, Luciano; Ortar, Giorgio; Schiano Moriello, Aniello; Serum, Eric M.; Rusterholz, David B./titolo:Structure-activity relationships of the prototypical TRPM8 agonist icilin/doi:10.1016%2Fj.bmcl.2015.04.032/rivista:Bioorganic & medicinal chemistry letters (Print)/anno:2015/pagina_da:2285/pagina_a:2290/intervallo_pagine:2285–2290/volume:25
A series of structural analogues of the TRPM8 agonist icilin was prepared. The compounds were examined for their ability to exert agonist or antagonist effects in HEK-293 cells expressing the TRPM8 receptor. Most structural modifications of the icili
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d1da59fbd129bc0f9637f37aff411ef1
https://pubmed.ncbi.nlm.nih.gov/25935641
https://pubmed.ncbi.nlm.nih.gov/25935641
Publikováno v:
The Chemical Educator. 2:1-8
Nuclear magnetic resonance spectroscopy holds a premier position as a tool for structure elucidation in organic chemistry. With the increased availability of high-field Fourier-transform spectrometers in undergraduate laboratories, there is an increa
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::3f62f1e7a867a387571cc8439708650e
https://doi.org/10.1007/s00897970105a
https://doi.org/10.1007/s00897970105a
Publikováno v:
The Chemical Educator. 2:1-5
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::1bfa444027205f3bf6a5af40b9810d20
https://doi.org/10.1007/s00897-997-0005-3
https://doi.org/10.1007/s00897-997-0005-3
Publikováno v:
ChemInform. 23
Higher imine esters 1a-h and 7a-b of amino acids and dipeptides are prepared in 68-91 % yield by saponification of the benzophenone Schiff base methyl esters 3a-d and 6 using phase-transfer techniques followed by O-alkylation with an alkyl halide. Th
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::83ca8b1ad53c2da5c00e32d4e81c613f
https://doi.org/10.1002/chin.199219289
https://doi.org/10.1002/chin.199219289
Publikováno v:
Synthesis. 1991:989-993
Higher imine esters 1a-h and 7a-b of amino acids and dipeptides are prepared in 68-91 % yield by saponification of the benzophenone Schiff base methyl esters 3a-d and 6 using phase-transfer techniques followed by O-alkylation with an alkyl halide. Th
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::352c4bc91e545324f8b29e308c161664
https://doi.org/10.1055/s-1991-26625
https://doi.org/10.1055/s-1991-26625
Publikováno v:
Molecules
Volume 2
Issue 5
Pages 80-86
Molecules, Vol 2, Iss 5, Pp 80-86 (1997)
Volume 2
Issue 5
Pages 80-86
Molecules, Vol 2, Iss 5, Pp 80-86 (1997)
Two 1,3,8,10-undecatetraenes were synthesized to test the viability of the intramolecular radical cation induced Diels-Alder reaction in the diene - diene format. Cyclization was successful only for the substituted tetraene with the lower oxidation p
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b24d1e021f31a9b8c71f542863588f95
Autor:
David B. Rusterholz
Publikováno v:
Journal of Chemical Education. 83:1809
Capsaicin, a fairly simple substituted amide of an aliphatic acid, has long been known as the active principle in hot chili peppers. In addition to causing a pronounced burning sensation, this substance has also been noted to produce a diminished sen
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::046f7c4c22c1b88e089dda2759c30b1a
https://doi.org/10.1021/ed083p1809
https://doi.org/10.1021/ed083p1809
Publikováno v:
Journal of Medicinal Chemistry. 19:99-102
In our attempts to elucidate the prolactin release inhibiting pharmacophore within the ergoline structure, we have prepared one indolealkylamine and several 2-aminotetralin derivatives. These congeners have been evaluated for inhibition of prolactin
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::43056677d940b7fa6c27d77486817d9a
https://doi.org/10.1021/jm00223a016
https://doi.org/10.1021/jm00223a016
Publikováno v:
Synthetic Communications. 19:1157-1165
α-Methylhistidine was prepared by two complementary routes using a catalytic phase-transfer alkylation procedure. Construction of the product was achieved either by alkylation of an alanine Schiff base ester with an imidazole-containing electrophile
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::1951177eac65d410a0a10602ef6e3863
https://doi.org/10.1080/00397918908054518
https://doi.org/10.1080/00397918908054518