Zobrazeno 1 - 10
of 14
pro vyhledávání: '"Daniele Zonari"'
Autor:
Silvia Arpicco, Michał Bartkowski, Alessandro Barge, Daniele Zonari, Loredana Serpe, Paola Milla, Franco Dosio, Barbara Stella, Silvia Giordani
Publikováno v:
Frontiers in Chemistry, Vol 8 (2020)
Hyaluronic acid (HA) is a ubiquitous biopolymer involved in many pathophysiological roles. One HA receptor, the cluster of differentiation CD44 protein, is often overexpressed in tumor cells. As such, HA has attracted considerable interest in the dev
Externí odkaz:
https://doaj.org/article/a15df633a4bb425fab92b7f66174bc71
Autor:
Alessio Malfanti, Ivana Miletto, Emanuela Bottinelli, Daniele Zonari, Giulia Blandino, Gloria Berlier, Silvia Arpicco
Publikováno v:
Molecules, Vol 21, Iss 4, p 522 (2016)
In this paper, mesoporous silica nanoparticles (MSNs) were studied as vehicles for the delivery of the antitumoral drug gemcitabine (GEM) and of its 4-(N)-acyl derivatives, (4-(N)-valeroyl-(C5GEM), 4-(N)-lauroyl-(C12GEM) and 4-(N)-stearoyl-gemcitabin
Externí odkaz:
https://doaj.org/article/1d86f2cce2bf43638fb6ec02d2b8691d
Autor:
Agnese Chiara Pippione, Zühal Kilic-Kurt, Sandra Kovachka, Stefano Sainas, Barbara Rolando, Enrica Denasio, Klaus Pors, Salvatore Adinolfi, Daniele Zonari, Renzo Bagnati, Marco Lucio Lolli, Francesca Spyrakis, Simonetta Oliaro-Bosso, Donatella Boschi
Publikováno v:
European Journal of Medicinal Chemistry. 237:114366
The aldo-keto reductase 1C3 (AKR1C3) enzyme is considered an attractive target in Castration Resistant Prostate Cancer (CRPC) because of its role in the biosynthesis of androgens. Flufenamic acid, a non-selective AKR1C3 inhibitor, has previously been
Autor:
Elisabetta Marini, Daniele Zonari, Irene Maria Carnovale, Rosmarie Friemann, Agnese Chiara Pippione, Parveen Goyal, Valentina Boscaro, Barbara Rolando, Simonetta Oliaro-Bosso, Salvatore Adinolfi, Marco Lucio Lolli, Weixiao Yuan Wahlgren, Renzo Bagnati, Margherita Gallicchio, Davide Bonanni, Donatella Boschi
Publikováno v:
ACS Medicinal Chemistry Letters. 10:437-443
[Image: see text] Aldo-keto reductase 1C3 (AKR1C3) is an attractive target in drug design for its role in resistance to anticancer therapy. Several nonsteroidal anti-inflammatory drugs such as indomethacin are known to inhibit AKR1C3 in a nonselectiv
Autor:
Barbara Stella, Alessandro Barge, Loredana Serpe, Michał Bartkowski, Franco Dosio, Silvia Giordani, Silvia Arpicco, Paola Milla, Daniele Zonari
Publikováno v:
Frontiers in Chemistry
Frontiers in Chemistry, Vol 8 (2020)
Frontiers in Chemistry, Vol 8 (2020)
Hyaluronic acid (HA) is a ubiquitous biopolymer involved in many pathophysiological roles. One HA receptor, the cluster of differentiation CD44 protein, is often overexpressed in tumor cells. As such, HA has attracted considerable interest in the dev
Autor:
Ingrid Corazzari, Roberto Canaparo, Alessandro Barge, Franco Dosio, Daniele Zonari, Silvia Arpicco, Federica Bosca, Linda Pastero, Gianni Durando, Giancarlo Cravotto, Federica Foglietta, Loredana Serpe, Francesco Turci, Silvia Tagliapietra
Publikováno v:
RSC advances. 10(37)
Sonodynamic therapy (SDT) is an innovative anticancer approach, based on the excitation of a given molecule (usually a porphyrin) by inertial acoustic cavitation that leads to cell death via the production of reactive oxygen species (ROS). This study
Autor:
Flavia Carton, Daniele Zonari, Stefania Cannito, Alessandro Marengo, Valentina Ricci, Manuela Malatesta, Silvia Arpicco, Maria Teresa Scupoli, Gloria Berlier, Federico Boschi
Publikováno v:
Journal of Colloid and Interface Science. 516:484-497
We have prepared and evaluated the physico-chemical and biological properties of four different hyaluronated mesoporous silica nanoparticles (MSNs) samples (MSN/HA). Hyaluronic acid (HA) with two different molecular weights (200 and 6.4 kDa) was used
Autor:
Davide Bonanni, Marco Lucio Lolli, Weixiao Yuan Wahlgren, Rosmarie Friemann, Renzo Bagnati, Daniele Zonari, Agnese Chiara Pippione, Simonetta Oliaro-Bosso, Donatella Boschi, Parveen Goyal, Salvatore Adinolfi, Claudio Festuccia, Klaus Pors, Elisabetta Marini, Irene Maria Carnovale, Marcella Sini
Publikováno v:
European Journal of Medicinal Chemistry. 150:930-945
The aldo-keto reductase 1C3 (AKR1C3) isoform plays a vital role in the biosynthesis of androgens and is considered an attractive target in prostate cancer (PCa). No AKR1C3-targeted agent has to date been approved for clinical use. Flufenamic acid and
Publikováno v:
International Journal of Pharmaceutics. 530:239-248
The systemic administration of methotrexate (MTX), a commonly used, antineoplastic drug which is also used in cutaneous disorders, is primarily associated with prolonged retention in the body and consequently with side effects. Innovative drug delive
Publikováno v:
International Journal of Pharmaceutics. 454:653-659
Paclitaxel has been found to be very effective against several human cancers; one of the major problems with its use is its poor solubility, which makes necessary its solubilization with excipients that can determine allergic reactions often severe.