Zobrazeno 1 - 2
of 2
pro vyhledávání: '"Dajiang Jing"'
Autor:
Andrew Dalgleish, Keith R. Mulholland, Andrew D. Campbell, David Dave, Hannah Askey, Zhaoshan Cui, Gareth AstraZeneca R D Charnwood Ensor, Shenghua Wang, Peter R. Hamilton, Simone Tomasi, Mark A. Graham, Claire Heffernan, Lai Chan, Pengpeng Liu, Emma Randles, Martin F. Jones, Michael Popadynec, Dajiang Jing, Cooper Katie Grace, Mohammed Pervez, Maria Rita Galan Espinosa, Jackson Lucinda Victoria
Publikováno v:
Organic Process Research & Development. 25:43-56
Ceralasertib is currently being evaluated in multiple phase I/II clinical trials for the treatment of cancer. Its structure, comprising a pyrimidine core decorated with a chiral morpholine, a cyclo...
Autor:
Hao Sun, Michael O. Frederick, Roger Ryan Rothhaar, Amy C. DeBaillie, Brian Morgan Watson, Carlos Mateos, Leonard L. Winneroski, Carlos Jaramillo, Talbi Kaoudi, Matthew Johnson, Pablo Garcia-Losada, Srinivas Gangula, Peter J. Lindsay-Scott, Steven James Green, Dustin J. Mergott, Dajiang Jing, Marvin M. Hansen, José Eugenio de Diego, Juan A. Rincón, Kevin D. Seibert, Lei Zhang, Jiuyuan Li
Publikováno v:
Organic Process Research & Development. 24:306-314
Herein we report a summary of the synthetic development of LY3202626 from the initial discovery route to a final route that was scaled to make 150 kg. Key developments include the use of a [3 + 2] ...