Zobrazeno 1 - 10
of 192
pro vyhledávání: '"D. Nisato"'
Autor:
Rebecca M. Pruss, Claude Barberis, Jacques Simiand, Colette Lacour, D. Nisato, Gabrielle Brossard, Philippe Soubrie, Jean Wagnon, Guy Griebel, Claudine Serradeil-Le Gal, Gérard Le Fur, J P Maffrand, Marc Pascal, Bernard Scatton, Gilles Guillon
Publikováno v:
Journal of Pharmacology and Experimental Therapeutics. 300:1122-1130
(2S,4R)-1-[5-Chloro-1-[(2,4-dimethoxyphenyl)sulfonyl]-3-(2-methoxy-phenyl)-2-oxo-2,3-dihydro-1H-indol-3-yl]-4-hydroxy-N,N-dimethyl-2-pyrrolidine carboxamide (SSR149415), the first selective, nonpeptide vasopressin V1b receptor antagonist yet describe
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::58f67d43bd81433e1f53f82c12eebbf4
https://doi.org/10.1124/jpet.300.3.1122
https://doi.org/10.1124/jpet.300.3.1122
Autor:
C. Loichot, Jean-Louis Imbs, C. Cazaubon, D. Nisato, W. De Jong, Mariette Barthelmebs, Michèle Grima
Publikováno v:
Hypertension. 35:602-608
Abstract —Nitric oxide attenuates both vasopressin-induced vasoconstriction and vasopressin release. We tested whether hypertension and renal dysfunction elicited by chronic inhibition of nitric oxide (NO) synthesis using N G -nitro- l -arginine (L
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::12748623059e8f0d085bc69c32902713
https://doi.org/10.1161/01.hyp.35.2.602
https://doi.org/10.1161/01.hyp.35.2.602
Autor:
J.C. Brelière, C. Bernhart, Colette Lacour, A. Roccon, D. Nisato, Jean Gougat, Catherine Cazaubon, G. Le Fur, J.‐L. A. Assens, F.B. Hundricourt
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 4:157-162
A novel series of substituted 3H-dihydro-pyrimidinones, homologues of SR 47436, was identified as AT 1 receptor antagonists. The best compounds showed high affinity for the AT 1 receptor (rate liver membrane prepration) with IC 50 's in the nanomolar
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::4f53f8268321bc898186b33f98e7d686
https://doi.org/10.1016/s0960-894x(01)81139-2
https://doi.org/10.1016/s0960-894x(01)81139-2
Publikováno v:
Life Sciences. 54:PL95-PL100
In guinea pigs anaesthetized with sodium pentobarbital, SR 48692, a non peptide neurotensin receptor antagonist blunted the blood pressure increase induced by exogenous neurotensin in a dose dependent manner. Furthermore, in asolated spontaneously be
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a0b5352172f066ea334ac539ba027b4e
https://doi.org/10.1016/0024-3205(94)00411-0
https://doi.org/10.1016/0024-3205(94)00411-0
Autor:
Bernard Ferrari, Jacques Clement, A. Roccon, Yvette Muneaux, Claude Bernhart, Claude Muneaux, J.C. Brelière, J. Taillades, D. Nisato, P. Perreaut, G. Le Fur, Jean Gougat, F. Haudricourt, Colette Lacour, Catherine Cazaubon, J.‐L. A. Assens, P. Guiraudou, M.‐A. Vignal
Publikováno v:
ChemInform. 25
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::79832b20ce71215dd3cfb45d670eb24c
https://doi.org/10.1002/chin.199411140
https://doi.org/10.1002/chin.199411140
Publikováno v:
Biochemical and Biophysical Research Communications. 188:873-878
Starting from highly potent HIV-1 protease pepstatine analog inhibitors, we have tried to find the minimum consensus sequence which is necessary to conserve anti-protease potency and antiviral activity. We describe here some statine based tripeptides
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::31e8cd95cad44e17775b40c36532874a
https://doi.org/10.1016/0006-291x(92)91137-f
https://doi.org/10.1016/0006-291x(92)91137-f
The present study investigated the effects of dronedarone and amiodarone on plasma thyroid hormones and the possible consequences on the response of the heart to ischemia. Amiodarone (30 mg/kg/day per os) or dronedarone (30 mg/kg/day per os) were adm
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=od______2127::ac871f6f49e4aabfe883b3579bb8f3c4
https://pergamos.lib.uoa.gr/uoa/dl/object/uoadl:3022939
https://pergamos.lib.uoa.gr/uoa/dl/object/uoadl:3022939
Autor:
M J, Clair, M K, King, A T, Goldberg, J W, Hendrick, R, Nisato, D M, Gay, A E, Morrison, J H, McElmurray, R S, Krombach, B R, Bond, C, Cazaubon, D, Nisato, F G, Spinale
Publikováno v:
The Journal of pharmacology and experimental therapeutics. 293(3)
With developing congestive heart failure (CHF), activation of the vasopressin V(1a) and angiotensin II type 1 (AT(1)) receptors can occur. In the present study, we examined the direct effects of V(1a) receptor blockade (V(1a) block), selective AT(1)
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::04dedd7824355bdcf7cb001da57ac8fd
https://pubmed.ncbi.nlm.nih.gov/10869385
https://pubmed.ncbi.nlm.nih.gov/10869385
Publikováno v:
The Journal of pharmacology and experimental therapeutics. 292(1)
We studied the effects of dronedarone (SR 33589) on the action potentials, membrane ionic currents, and arrhythmic activity in control rats and in rats after myocardial infarction, a model known to develop anomalous electrical activity. Dronedarone i
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::1ed2f18517158603c52a29f6d3933789
https://pubmed.ncbi.nlm.nih.gov/10604978
https://pubmed.ncbi.nlm.nih.gov/10604978
Publikováno v:
Archives des maladies du coeur et des vaisseaux. 91(8)
Previously we reported that AVP is a potent vasoconstrictor in the TYRODE's perfused rat kidney. In vivo however AVP elicited only minor effects on renal blood flow. We hypothetized that differences in shear stress, particularly related to difference
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::5ae5efae30c4ece8e82e04fde5ed8a39
https://pubmed.ncbi.nlm.nih.gov/9749170
https://pubmed.ncbi.nlm.nih.gov/9749170