Synthesis, Analytical Characterization, and Human CB 1 Receptor Binding Studies of the Chloroindole Analogues of the Synthetic Cannabinoid MDMB-CHMICA.

Autor: Münster-Müller, Sascha^1,2 (AUTHOR) smuenster@eu.sterigenics.com, Hansen, Steven³ (AUTHOR) steven.hansen@sgs.com, Lucas, Tobias³ (AUTHOR) tobiaslucas.chem@gmail.com, Giorgetti, Arianna^4,5 (AUTHOR) arianna.giorgetti@unibo.it, Mogler, Lukas^5,6 (AUTHOR) volker.auwaerter@uniklinik-freiburg.de, Fischmann, Svenja⁷ (AUTHOR) svenja.fischmann@projekt-adebar.eu, Westphal, Folker⁷ (AUTHOR) folker.dr.westphal@polizei.landsh.de, Auwärter, Volker^5,6 (AUTHOR), Pütz, Michael¹ (AUTHOR) michael.puetz@bka.bund.de, Opatz, Till³ (AUTHOR) opatz@uni-mainz.de

Publikováno v: Biomolecules (2218-273X). Nov2024, Vol. 14 Issue 11, p1414. 15p.

A novel monoacylglycerol lipase inhibitor with analgesic and anti-inflammatory activity

Autor: Magrioti, V. Naxakis, G. Hadjipavlou-Litina, D. Makriyannis, A. Kokotos, G.

A variety of long chain 1,2-diamines and related compounds were synthesized and tested for their activity on fatty acid amide hydrolase (FAAH) and monoacyglycerol lipase (MGL). (2S,9Z)-Octadec-9-ene-1,2-diamine selectively inhibits MGL (Ki 21.8μ M)

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=od______2127::c4ed6f727ef8e626ec62c87489a24c45
https://pergamos.lib.uoa.gr/uoa/dl/object/uoadl:3062290

Clinical, laboratory and immunologic effects of the treatment of endemic goiter with T4, T3 and KI

Autor: D A, Koutras, G D, Piperingos, D, Pallas, K, Katsouyanni, K S, Karaiskos, P, Marafelia, D, Makriyannis, J, Kitsopanides, J, Sfontouris, J, Mantzos

Publikováno v: Thyroidology. 2(2)

We treated 204 patients with endemic nontoxic goiter with T4, T3 and KI, singly or in combination. Definitely nodular goiters were excluded, since the possibility of autonomy would be increased. Goiter size was evaluated before and 6 months after tre

Externí odkaz: https://explore.openaire.eu/search/publication?articleId=pmid________::8869b0043bfdecc2dea6631672d2c9de
https://pubmed.ncbi.nlm.nih.gov/1724914

Systematic Modification of the Substitution Pattern of the 7-Hydroxy-5-oxopyrazolo[4,3- b ]pyridine-6-carboxamide Scaffold Enabled the Discovery of New Ligands with High Affinity and Selectivity for the Cannabinoid Type 2 Receptor.

Autor: Mugnaini, Claudia¹ (AUTHOR) marta.casini94@gmail.com, Kostrzewa, Magdalena² (AUTHOR) m.kostrzewka@gmail.com, Casini, Marta¹ (AUTHOR) valeriacatallo@gmail.com, Kumar, Poulami² (AUTHOR) p.kumar@icb.cnr.it, Catallo, Valeria¹ (AUTHOR) guastaferro.laura@gmail.com, Allarà, Marco² (AUTHOR) mallara@icb.cnr.it, Guastaferro, Laura¹ (AUTHOR) antonella.brizzi@unisi.it, Brizzi, Antonella¹ (AUTHOR) paolino3@unisi.it, Paolino, Marco¹ (AUTHOR) andrea.tafi@unisi.it, Tafi, Andrea¹ (AUTHOR) kapatais@student.unisi.it, Kapatais, Christelos¹ (AUTHOR) gianluca.giorgi@unisi.it, Giorgi, Gianluca¹ (AUTHOR) federico.corelli@unisi.it, Vacondio, Federica³ (AUTHOR) federica.vacondio@unipr.it, Mor, Marco³ (AUTHOR) marco.mor@unipr.it, Corelli, Federico¹ (AUTHOR), Ligresti, Alessia² (AUTHOR) claudia.mugnaini@unisi.it

Publikováno v: Molecules. Jul2023, Vol. 28 Issue 13, p4958. 29p.

Impact of dietary changes on retinal neuronal plasticity in rodent models of physical and psychological trauma.

Autor: Patel, Mital Y., Yang, Ruoting, Chakraborty, Nabarun, Miller, Stacy-Ann, DeMar, James C., Batuure, Andrew, Wilder, Donna, Long, Joseph, Hammamieh, Rasha, Gautam, Aarti

Publikováno v: Frontiers in Genetics; 9/27/2024, p1-13, 13p