Cyclization of acyl thiosemicarbazides led to new Helicobacter pylori α‐carbonic anhydrase inhibitors.

Autor: Gumus, Arzu, D'Agostino, Ilaria, Puca, Valentina, Crocetta, Valentina, Carradori, Simone, Cutarella, Luigi, Mori, Mattia, Carta, Fabrizio, Angeli, Andrea, Capasso, Clemente, Supuran, Claudiu T.

Publikováno v: Archiv der Pharmazie; Nov2024, Vol. 357 Issue 11, p1-16, 16p

Lasamide Containing Sulfonylpiperazines as Effective Agents for the Management of Glaucoma Associated Symptoms.

Autor: Kilbile JT; Department of Chemistry, School of Basic and Applied Sciences, MGM University, Chhatrapati Sambhajinagar, 431003, MS, India., Sapkal SB; Department of Chemistry, School of Basic and Applied Sciences, MGM University, Chhatrapati Sambhajinagar, 431003, MS, India., Renzi G; NEUROFARBA Department, Sezione di Scienze Farmaceutiche e Nutraceutiche, University of Florence, 50019, Sesto Fiorentino, Florence, Italy., D'Agostino I; NEUROFARBA Department, Sezione di Scienze Farmaceutiche e Nutraceutiche, University of Florence, 50019, Sesto Fiorentino, Florence, Italy.; Department of Pharmacy, University of Pisa, 56126, Pisa, Italy.; Department of Pharmacy, University 'G. d'Annunzio' Chieti-Pescara, 66100, Chieti, Italy., Boudjelal M; King Abdullah International Medical Research Center (KAIMRC), King Saud Bin Abdulaziz University for Health Sciences, Ministry of National Guard-Health Affairs, Riyadh, 14811, Saudi Arabia., Tamboli Y; King Abdullah International Medical Research Center (KAIMRC), King Saud Bin Abdulaziz University for Health Sciences, Ministry of National Guard-Health Affairs, Riyadh, 14811, Saudi Arabia., Cutarella L; Department of Biotechnology, Chemistry and Pharmacy, University of Siena, via Aldo Moro 2, 53100, Siena, Italy., Mori M; Department of Biotechnology, Chemistry and Pharmacy, University of Siena, via Aldo Moro 2, 53100, Siena, Italy., Sgambellone S; NEUROFARBA Department, Section of Pharmacology and Toxicology, University of Florence, 50139, Florence, Italy., Villano S; NEUROFARBA Department, Section of Pharmacology and Toxicology, University of Florence, 50139, Florence, Italy., Marri S; NEUROFARBA Department, Section of Pharmacology and Toxicology, University of Florence, 50139, Florence, Italy., Lucarini L; NEUROFARBA Department, Section of Pharmacology and Toxicology, University of Florence, 50139, Florence, Italy., Carradori S; Department of Pharmacy, University 'G. d'Annunzio' Chieti-Pescara, 66100, Chieti, Italy., Carta F; NEUROFARBA Department, Sezione di Scienze Farmaceutiche e Nutraceutiche, University of Florence, 50019, Sesto Fiorentino, Florence, Italy., Supuran CT; NEUROFARBA Department, Sezione di Scienze Farmaceutiche e Nutraceutiche, University of Florence, 50019, Sesto Fiorentino, Florence, Italy.

Publikováno v: ChemMedChem [ChemMedChem] 2024 Sep 25, pp. e202400601. Date of Electronic Publication: 2024 Sep 25.