Zobrazeno 1 - 10
of 757
pro vyhledávání: '"Constantin G. Daniliuc"'
Publikováno v:
Nature Communications, Vol 14, Iss 1, Pp 1-8 (2023)
Abstract Partially saturated, fluorine-containing rings are ubiquitous across the drug discovery spectrum. This capitalises upon the biological significance of the native structure and the physicochemical advantages conferred by fluorination. Motivat
Externí odkaz:
https://doaj.org/article/93424e46ee464c13ba513d50bcefc52e
Publikováno v:
Molecules, Vol 28, Iss 5, p 2011 (2023)
A complex [Zn(bpy)(acr)2]·H2O (1) was converted in a DMF medium (DMF = N,N′-dimethylformamide) into a coordination polymer [Zn(bpy)(acr)(HCOO)]n (1a) (bpy = 2,2′-bipyridine, and Hacr = acrylic acid), and the species was fully characterized throu
Externí odkaz:
https://doaj.org/article/5968176edef0455fa0ddee6afa7f517e
Publikováno v:
Beilstein Journal of Organic Chemistry, Vol 16, Iss 1, Pp 1627-1635 (2020)
Substrate specificity is ubiquitous in biological catalysis, but less pervasive in the realm of small-molecule catalysis. Herein, we disclose an intriguing example of substrate specificity that was observed whilst exploring catalysis-based routes to
Externí odkaz:
https://doaj.org/article/490fc3c76f254a5f82146c6a78a25ced
Autor:
Calvin Dunker, Lukas Imberg, Alena I. Siutkina, Catharina Erbacher, Constantin G. Daniliuc, Uwe Karst, Dmitrii V. Kalinin
Publikováno v:
Pharmaceuticals, Vol 15, Iss 11, p 1340 (2022)
New antithrombotic drugs are needed to combat thrombosis, a dangerous pathology that causes myocardial infarction and ischemic stroke. In this respect, thrombin (FIIa) represents an important drug target. We herein report the synthesis and biological
Externí odkaz:
https://doaj.org/article/ebd9022cc2cd4fea8131c332891daf74
Autor:
Rodica Olar, Constantin G. Daniliuc, Gina Vasile Scăețeanu, Romana Cerc Korosec, Nataša Čelan Korošin, Mariana Carmen Chifiriuc, Mihaela Badea
Publikováno v:
Crystals, Vol 12, Iss 8, p 1078 (2022)
A new co-crystal with the formula [Ni(bpy)(acr)2(H2O)]·MA (bpy = 2,2′-bipyridine, acr = acrylate and MA = melamine) has been synthesized and characterized using IR, UV-Vis, thermogravimetric analysis and single crystal X-ray diffraction. The compl
Externí odkaz:
https://doaj.org/article/303e7a11019b4fd09c2a15ef40de44b2
Autor:
Jan Phillip Lemmerhirt, Andreas Isaak, Rongfang Liu, Max Kock, Constantin G. Daniliuc, Kenneth A. Jacobson, Laura H. Heitman, Anna Junker
Publikováno v:
Molecules, Vol 27, Iss 7, p 2283 (2022)
The adenosine A3 receptor is a promising target for treating and diagnosing inflammation and cancer. In this paper, a series of bicyclo[3.1.0]hexane-based nucleosides was synthesized and evaluated for their P1 receptor affinities in radioligand bindi
Externí odkaz:
https://doaj.org/article/ff4540a03cd6405b9529e70cd9c00188
Autor:
Babita Aneja, Mudsser Azam, Shadab Alam, Ahmad Perwez, Ronan Maguire, Umesh Yadava, Kevin Kavanagh, Constantin G. Daniliuc, M. Moshahid A. Rizvi, Qazi Mohd. Rizwanul Haq, Mohammad Abid
Publikováno v:
ACS Omega, Vol 3, Iss 6, Pp 6912-6930 (2018)
Externí odkaz:
https://doaj.org/article/152477dc83b24dd69873c55453ef48e7
Autor:
Felix Scheidt, Christian Thiehoff, Gülay Yilmaz, Stephanie Meyer, Constantin G. Daniliuc, Gerald Kehr, Ryan Gilmour
Publikováno v:
Beilstein Journal of Organic Chemistry, Vol 14, Iss 1, Pp 1021-1027 (2018)
Herein, we describe a catalytic fluorooxygenation of readily accessible N-allylcarboxamides via an I(I)/I(III) manifold to generate 2-oxazolines containing a fluoromethyl group. Catalysis is conditional on the oxidation competence of Selectfluor®, w
Externí odkaz:
https://doaj.org/article/8f44c7183a2d4562a88dc1f4f05c2339
Autor:
Anna Galkina, Nico Krause, Mairin Lenz, Constantin G. Daniliuc, Marcel Kaiser, Thomas J. Schmidt
Publikováno v:
Molecules, Vol 24, Iss 6, p 1068 (2019)
As part of our efforts to exploit the antitrypanosomal potential of sesquiterpene lactones (STL) from Helianthus tuberosus L. (Asteraceae), besides the known 4,15-iso-atriplicolide tiglate, -methacrylate and -isobutyrate, a hitherto unknown STL was i
Externí odkaz:
https://doaj.org/article/bfbefcf267a8495bb2c4a569fafc59d6
Autor:
Ioana Dorina Vlaicu, Gheorghe Borodi, Gina Vasile Scăețeanu, Mariana Carmen Chifiriuc, Luminița Măruțescu, Marcela Popa, Mariana Stefan, Ionel Florinel Mercioniu, Martin Maurer, Constantin G. Daniliuc, Rodica Olar, Mihaela Badea
Publikováno v:
Molecules, Vol 23, Iss 12, p 3253 (2018)
Five new copper(II) acrylate complexes (acr is the acrylate anion: C3H3O2) with imidazole derivatives (2-methylimidazole/2-MeIm, 5-methylimidazole/5-MeIm, 2-ethylimidazole/2-EtIm) of type: cis-[Cu(2-RIm)2(acr)2]·xH2O ((1): R = ⁻CH3, x = 2; (4): R
Externí odkaz:
https://doaj.org/article/6420c4ee100648e6850e4b04e9c7debe