Synthesis and in vitro evaluation of new 5-substituted 6-nitroimidazooxazoles as antikinetoplastid agents

Autor: Mathias, Fanny, Cohen, Anita, Kabri, Youssef, Negrão, Núria Waddington, Crozet, Maxime D., Docampo, Roberto, Azas, Nadine, Vanelle, Patrice

Publikováno v: In European Journal of Medicinal Chemistry 1 April 2020 191

8-Aryl-6-chloro-3-nitro-2-(phenylsulfonylmethyl)imidazo[1,2-a]pyridines as potent antitrypanosomatid molecules bioactivated by type 1 nitroreductases

Autor: Fersing, Cyril, Boudot, Clotilde, Pedron, Julien, Hutter, Sébastien, Primas, Nicolas, Castera-Ducros, Caroline, Bourgeade-Delmas, Sandra, Sournia-Saquet, Alix, Moreau, Alain, Cohen, Anita, Stigliani, Jean-Luc, Pratviel, Geneviève, Crozet, Maxime D., Wyllie, Susan, Fairlamb, Alan, Valentin, Alexis, Rathelot, Pascal, Azas, Nadine, Courtioux, Bertrand, Verhaeghe, Pierre, Vanelle, Patrice

Publikováno v: In European Journal of Medicinal Chemistry 5 September 2018 157:115-126

Synthesis and Antimalarial Evaluation of New 1,3,5- tris [(4-(Substituted-aminomethyl)phenyl)methyl]benzene Derivatives: A Novel Alternative Antiparasitic Scaffold.

Autor: Albenque-Rubio, Sandra, Guillon, Jean, Cohen, Anita, Agnamey, Patrice, Savrimoutou, Solène, Moreau, Stéphane, Mergny, Jean-Louis, Ronga, Luisa, Kanavos, Ioannis, Moukha, Serge, Dozolme, Pascale, Sonnet, Pascal

Publikováno v: Drugs & Drug Candidates; Sep2023, Vol. 2 Issue 3, p653-672, 20p

Discovery of new thienopyrimidinone derivatives displaying antimalarial properties toward both erythrocytic and hepatic stages of Plasmodium

Autor: Cohen, Anita, Suzanne, Peggy, Lancelot, Jean-Charles, Verhaeghe, Pierre, Lesnard, Aurélien, Basmaciyan, Louise, Hutter, Sébastien, Laget, Michèle, Dumètre, Aurélien, Paloque, Lucie, Deharo, Eric, Crozet, Maxime D., Rathelot, Pascal, Dallemagne, Patrick, Lorthiois, Audrey, Sibley, Carol Hopkins, Vanelle, Patrice, Valentin, Alexis, Mazier, Dominique, Rault, Sylvain, Azas, Nadine

Publikováno v: In European Journal of Medicinal Chemistry 5 May 2015 95:16-28

Design, synthesis, and antiprotozoal evaluation of new 2,4-bis[(substituted-aminomethyl)phenyl]quinoline, 1,3-bis[(substituted-aminomethyl)phenyl]isoquinoline and 2,4-bis[(substituted-aminomethyl)phenyl]quinazoline derivatives.

Autor: Guillon, Jean¹ (AUTHOR), Cohen, Anita² (AUTHOR), Boudot, Clotilde³ (AUTHOR), Valle, Alessandra¹ (AUTHOR), Milano, Vittoria¹ (AUTHOR), Das, Rabindra Nath¹ (AUTHOR), Guédin, Aurore¹ (AUTHOR), Moreau, Stéphane¹ (AUTHOR), Ronga, Luisa⁴ (AUTHOR), Savrimoutou, Solène¹ (AUTHOR), Demourgues, Maxime¹ (AUTHOR), Reviriego, Elodie¹ (AUTHOR), Rubio, Sandra¹ (AUTHOR), Ferriez, Sandie¹ (AUTHOR), Agnamey, Patrice⁵ (AUTHOR), Pauc, Cécile⁵ (AUTHOR), Moukha, Serge⁶ (AUTHOR), Dozolme, Pascale⁶ (AUTHOR), Nascimento, Sophie Da⁵ (AUTHOR), Laumaillé, Pierre⁵ (AUTHOR)

Publikováno v: Journal of Enzyme Inhibition & Medicinal Chemistry. Dec2020, Vol. 35 Issue 1, p432-459. 28p.