Zobrazeno 1 - 5
of 5
pro vyhledávání: '"Claudia, Gioé"'
Autor:
Claudia Gioé-Gallo, Sandra Ortigueira, José Brea, Iu Raïch, Jhonny Azuaje, M. Rita Paleo, Maria Majellaro, María Isabel Loza, Cristian O. Salas, Xerardo García-Mera, Gemma Navarro, Eddy Sotelo
Publikováno v:
Biomedicine & Pharmacotherapy, Vol 164, Iss , Pp 114934- (2023)
Synthetic cannabinoid receptor agonists (SCRAs) constitute the largest and most defiant group of abuse designer drugs. These new psychoactive substances (NPS), developed as unregulated alternatives to cannabis, have potent cannabimimetic effects and
Externí odkaz:
https://doaj.org/article/3b0ddeb6be494b4382e24224b8f69591
Autor:
Silvia Novío, Christian Fernandez-Masaguer, Jhonny Azuaje, Hugo Gutiérrez-de-Terán, Olga Caamaño, Carlos Rodríguez-García, Manuel Freire-Garabal, Angela Stefanachi, Carlota Garcia-Santiago, Willem Jespers, Abel Crespo, María Isabel Loza, Javier F Sardina, José Brea, Johan Åqvist, Eddy Sotelo, Abdelaziz El Maatougui, Ana Mallo-Abreu, Rubén Prieto-Díaz, María Majellaro, Belma Alispahic, Xerardo García-Mera, María José Núñez, Claudia Gioé
Publikováno v:
Journal of Medicinal Chemistry. 64:458-480
We present and thoroughly characterize a large collection of 3,4-dihydropyrimidin-2(1H)-ones as A2BAR antagonists, an emerging strategy in cancer (immuno) therapy. Most compounds selectively bind A2BAR, with a number of potent and selective antagonis
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::183bc670446a761e38b64f15b490b0a5
https://doi.org/10.1021/acs.jmedchem.0c01431
https://doi.org/10.1021/acs.jmedchem.0c01431
Autor:
Darío Miranda-Pastoriza, Rodrigo Bernárdez, Jhonny Azuaje, Rubén Prieto-Díaz, Maria Majellaro, Ashish V. Tamhankar, Lucien Koenekoop, Alejandro González, Claudia Gioé-Gallo, Ana Mallo-Abreu, José Brea, M. Isabel Loza, Aitor García-Rey, Xerardo García-Mera, Hugo Gutiérrez-de-Terán, Eddy Sotelo
Publikováno v:
Minerva. Repositorio Institucional de la Universidad de Santiago de Compostela
instname
instname
A library of potent and highly A3AR selective pyrimidine-based compounds was designed to explore non-orthosteric interactions within this receptor. Starting from a prototypical orthosteric A3AR antagonist (ISVY130), the structure-based design explore
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7f450a7e587f0fca905ab1dda8c351a1
http://urn.kb.se/resolve?urn=urn:nbn:se:uu:diva-469742
http://urn.kb.se/resolve?urn=urn:nbn:se:uu:diva-469742
Autor:
Darío, Miranda-Pastoriza, Rodrigo, Bernárdez, Jhonny, Azuaje, Rubén, Prieto-Díaz, Maria, Majellaro, Ashish V, Tamhankar, Lucien, Koenekoop, Alejandro, González, Claudia, Gioé-Gallo, Ana, Mallo-Abreu, José, Brea, M Isabel, Loza, Aitor, García-Rey, Xerardo, García-Mera, Hugo, Gutiérrez-de-Terán, Eddy, Sotelo
Publikováno v:
ACS medicinal chemistry letters. 13(2)
A library of potent and highly A
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::8d0e5fc921da290ffb774c8b89fbb407
https://pubmed.ncbi.nlm.nih.gov/35178181
https://pubmed.ncbi.nlm.nih.gov/35178181
Autor:
María, Majellaro, Willem, Jespers, Abel, Crespo, María J, Núñez, Silvia, Novio, Jhonny, Azuaje, Rubén, Prieto-Díaz, Claudia, Gioé, Belma, Alispahic, José, Brea, María I, Loza, Manuel, Freire-Garabal, Carlota, Garcia-Santiago, Carlos, Rodríguez-García, Xerardo, García-Mera, Olga, Caamaño, Christian, Fernandez-Masaguer, Javier F, Sardina, Angela, Stefanachi, Abdelaziz, El Maatougui, Ana, Mallo-Abreu, Johan, Åqvist, Hugo, Gutiérrez-de-Terán, Eddy, Sotelo
Publikováno v:
Journal of medicinal chemistry. 64(1)
We present and thoroughly characterize a large collection of 3,4-dihydropyrimidin-2(1
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::056382dfcad27ebd05f6de8885e73c1f
https://pubmed.ncbi.nlm.nih.gov/33372800
https://pubmed.ncbi.nlm.nih.gov/33372800