Zobrazeno 1 - 5
of 5
pro vyhledávání: '"Chunning, Shao"'
Autor:
Narayanan Hariharan, Kasim A. Mookhtiar, Liqun Gu, Jimmy Ren, Chen Sean, Ramakrishna Seethala, Michael Cap, Lori Kunselman, Min Zhou, Peter T. W. Cheng, William Fenderson, Chunning Shao, Cuixia Chu, Scott A. Biller, Hao Zhang, Fucheng Qu, Pratik Devasthale, Dennis Farrelly, Jeon Yoon T, Randolph P. Ponticiello, John R. Wetterau, Wei Wang, Wen-Pin Yang, Thomas Harrity, Aaron Tieman, Denis E. Ryono, Richard E. Gregg
Publikováno v:
Diabetes. 55:240-248
Muraglitazar, a novel dual (alpha/gamma) peroxisome proliferator-activated receptor (PPAR) activator, was investigated for its antidiabetic properties and its effects on metabolic abnormalities in genetically obese diabetic db/db mice. In db/db mice
Autor:
Denis E. Ryono, Chen Sean, Pratik Devasthale, Shu Y Chang, John R. Wetterau, W. Griffith Humphreys, Gary J. Grover, Dennis Farrelly, Jeon Yoon T, Fucheng Qu, Ramakrishna Seethala, Narayanan Hariharan, Wei Wang, Zhengping Ma, Scott A. Biller, Rajasree Golla, Lisa Moore, Arthur M. Doweyko, Michael Cap, Fred Selan, Jimmy Ren, Paul G. Sleph, Hao Zhang, Aaron Tieman, Vito G. Sasseville, Thomas Harrity, Gamini Chandrasena, Chunning Shao, Peter T. W. Cheng, Lin Cheng, Wei Sun
Publikováno v:
Journal of Medicinal Chemistry. 48:2248-2250
Muraglitazar/BMS-298585 (2) has been identified as a non-thiazolidinedione PPAR alpha/gamma dual agonist that shows potent activity in vitro at human PPARalpha (EC(50) = 320 nM) and PPARgamma(EC(50) = 110 nM). Compound 2 shows excellent efficacy for
Autor:
Thomas, Harrity, Dennis, Farrelly, Aaron, Tieman, Cuixia, Chu, Lori, Kunselman, Liqun, Gu, Randolph, Ponticiello, Michael, Cap, Fucheng, Qu, Chunning, Shao, Wei, Wang, Hao, Zhang, William, Fenderson, Sean, Chen, Pratik, Devasthale, Yoon, Jeon, Ramakrishna, Seethala, Wen-Pin, Yang, Jimmy, Ren, Min, Zhou, Denis, Ryono, Scott, Biller, Kasim A, Mookhtiar, John, Wetterau, Richard, Gregg, Peter T, Cheng, Narayanan, Hariharan
Publikováno v:
Diabetes. 55(1)
Muraglitazar, a novel dual (alpha/gamma) peroxisome proliferator-activated receptor (PPAR) activator, was investigated for its antidiabetic properties and its effects on metabolic abnormalities in genetically obese diabetic db/db mice. In db/db mice
Autor:
Schoen William R, Margit L. MacDougall, Gaetan H. Ladouceur, Roger A. Smith, Romulo Romero, Donald L. Hertzog, James N. Livingston, Chunning Shao, J.Howard Jones, James H. Cook, Kathleen M. Phelan, Martin H. Osterhout, Timothy G. Lease, Mary Korpusik, Thomas Hundertmark
Publikováno v:
Bioorganicmedicinal chemistry letters. 12(23)
Optimized substituent patterns in 4-aryl-pyridine glucagon receptor antagonists were merged to produce highly potent derivatives containing both a 3-[(1R)-hydroxyethyl] and a 2'-hydroxy group. Due to restricted rotation of the phenyl-pyridine bond, t
Autor:
Harrity, Thomas, Farrelly, Dennis, Tieman, Aaron, Cuixia Chu, Kunselman, Lori, Liqun Gu, Ponticiello, Randolph, Cap, Michael, Seethala, Ramakrishna, Ren, Jimmy, Min Zhou, Mookhtiar, Kasim A., Wetterau, John, Gregg, Richard, Hariharan, Narayanan, Fucheng Qu, Chunning Shao, Wei Wang, Hao Zhang, Chen, Scan
Publikováno v:
Diabetes; Jan2006, Vol. 55 Issue 1, p240-248, 9p, 1 Diagram, 3 Charts, 5 Graphs