Zobrazeno 1 - 6
of 6
pro vyhledávání: '"Christophe Parsy"'
Publikováno v:
European Journal of Organic Chemistry. 2022
Autor:
Nerina Dodic, Nicolas Ancellin, Morgane Bordessoules, Anne Bouillot, Nathan Butin, Cedric Charrier, Marie-Helene Fouchet, Alain Laroze, Anne-Pascale Luzy, Alexandre Moquette, Julia Pilot, Guillaume Serin, Jean-François Mirjolet, Fabrice Viviani, Christophe Parsy
Publikováno v:
Cancer Research. 82:1398-1398
Small molecule macrocyclic kinase inhibitors have attracted significant attention in drug discovery over the past years with drugs approval such as lorlatinib demonstrating the clinical relevance of this approach. We developed our expertise to furthe
Autor:
François-René Alexandre, Eric Badaroux, John P. Bilello, Stéphanie Bot, Tony Bouisset, Guillaume Brandt, Sylvie Cappelle, Christopher Chapron, Dominique Chaves, Thierry Convard, Clément Counor, Daniel Da Costa, David Dukhan, Marion Gay, Gilles Gosselin, Jean-François Griffon, Kusum Gupta, Brenda Hernandez-Santiago, Massimiliano La Colla, Marie-Pierre Lioure, Julien Milhau, Jean-Laurent Paparin, Jérôme Peyronnet, Christophe Parsy, Claire Pierra Rouvière, Houcine Rahali, Rachid Rahali, Aurélien Salanson, Maria Seifer, Ilaria Serra, David Standring, Dominique Surleraux, Cyril B. Dousson
Publikováno v:
Bioorganicmedicinal chemistry letters. 27(18)
Herein we describe the discovery of IDX21437 35b, a novel RPd-aminoacid-based phosphoramidate prodrug of 2'-α-chloro-2'-β-C-methyluridine monophosphate. Its corresponding triphosphate 6 is a potent inhibitor of the HCV NS5B RNA-dependent RNA polyme
Autor:
Tina Schultheiss, Sophia G. Antimisiaris, Richard Storer, Roberta Loddo, Christophe Parsy, Nicole Stolte-Leeb, Ulrike Sauermann, Paolo La Colla, Christiane Stahl-Hennig, Monika Franz, Spyridon Mourtas
Publikováno v:
AIDS Research and Human Retroviruses. 27:933-943
The availability of an effective vaginal microbicide would be a major step toward containment of HIV transmission as well as allowing women self-protection against HIV infection. Here we evaluated the efficacy of vaginal application of the potent non
Autor:
Christine Bodemer, Laurence Jonard, Sylvie Freitag, M'hamed Grati, Delphine Feldmann, Rémy Couderc, Céleste Koval, Françoise Denoyelle, Martine Sinico, Sandrine Marlin, Smail Hadj-Rabia, Christophe Parsy
Publikováno v:
European Journal of Medical Genetics. 51:35-43
Keratitis-Ichthyosis-Deafness (KID) syndrome (OMIM 148210) is a congenital ectodermal defect. KID consists of an atypical ichthyosiform erythroderma associated with congenital sensorineural deafness. A rare form of the KID syndrome is a fatal course
Autor:
Nicole Stolte-Leeb, Roberta Loddo, Sophia Antimisiaris, Tina Schultheiss, Ulrike Sauermann, Monika Franz, Spyridon Mourtas, Christophe Parsy, Richard Storer, Paolo La Colla, Christiane Stahl-Hennig
Publikováno v:
AIDS Research & Human Retroviruses; Sep2011, Vol. 27 Issue 9, p933-943, 11p