Zobrazeno 1 - 6
of 6
pro vyhledávání: '"Christian Montopoli"'
Autor:
Barbara Cacciari, Stefano Moro, K. Varani, P. G. Baraldi, Bolcato C, G. Spalluto, P.A. Borea, Da Ros T, Giorgia Pastorin, Christian Montopoli
Publikováno v:
Journal of Medicinal Chemistry. 49:1720-1729
Some pyrazolotriazolopyrimidines bearing different heteroarylcarbamoylamino moieties at the N5-position are described. We previously reported the synthesis of a water soluble compound with high potency and selectivity versus the human A3 adenosine re
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::65f637e6c2d75c7973f1f54375a53f96
https://doi.org/10.1021/jm051147+
https://doi.org/10.1021/jm051147+
Autor:
Claudia Martini, Stefano Moro, Ombretta Lenzi, Guido Filacchioni, Christian Montopoli, Flavia Varano, Daniela Catarzi, Vittoria Colotta, Letizia Trincavelli
Publikováno v:
Università degli studi di Firenze-IRIS
A number of 4-oxo-substituted 1,2,4-triazolo[1,5-a]quinoxaline derivatives bearing at position-2 the claimed (hetero)aryl moiety (compounds 1-15) but also a carboxylate group (16-28, 32-36) or a hydrogen atom (29-31) were designed as human A3 (hA3) a
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::93d038db5d38428211b39fead602cd17
https://doi.org/10.1021/jm0504149
https://doi.org/10.1021/jm0504149
Autor:
Barbara Cacciari, Sonja Kachler, Karl-Norbert Klotz, Christian Montopoli, Stefano Moro, Giampiero Spalluto, Chiara Bolcato, Giorgia Pastorin
Publikováno v:
Il Farmaco. 60:643-651
A new series of potential adenosine receptor antagonists with a [1,2,4]-triazolo-[3,4-f]-purine structure bearing at the 1 and 3 position n-propyl groups have been synthesized, and their affinities at the four human adenosine receptor subtypes (A(1),
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d35d8a7d74ced39a61c6247d33c8dbe4
https://doi.org/10.1016/j.farmac.2005.04.012
https://doi.org/10.1016/j.farmac.2005.04.012
Autor:
Giorgia, Pastorin, Tatiana, Da Ros, Chiara, Bolcato, Christian, Montopoli, Stefano, Moro, Barbara, Cacciari, Pier Giovanni, Baraldi, Katia, Varani, Pier Andrea, Borea, Giampiero, Spalluto
Publikováno v:
Journal of medicinal chemistry. 49(5)
Some pyrazolotriazolopyrimidines bearing different heteroarylcarbamoylamino moieties at the N5-position are described. We previously reported the synthesis of a water soluble compound with high potency and selectivity versus the human A3 adenosine re
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=pmid________::acf8c1738cc878dceb5e257a9641688d
https://pubmed.ncbi.nlm.nih.gov/16509587
https://pubmed.ncbi.nlm.nih.gov/16509587
Autor:
Karl-Norbert Klotz, Giampiero Spalluto, Stefano Moro, Christian Montopoli, Chiara Bolcato, Sonja Kachler, Barbara Cacciari, Giorgia Pastorin
A new series of potential adenosine receptor antagonists with a [1,2,4]-triazolo-[3,4-f]-purine structure have been synthesized, and their affinities at the four adenosine receptor subtypes (A1, A2A, A2B and A3) have been evaluated. The design was ba
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4afa3c5d9f85e66e9f64c7e6a69d0b8c
http://hdl.handle.net/11392/1691701
http://hdl.handle.net/11392/1691701
Autor:
Guido Filacchioni, Vittoria Colotta, Andrea Tralli, Claudia Martini, Stefano Moro, Christian Montopoli, Ombretta Lenzi, Francesca Romana Calabri, Flavia Varano, Letizia Trincavelli, Daniela Catarzi
Publikováno v:
Università degli studi di Firenze-IRIS
Some 2-aryl-8-chloro-1,2,4-triazolo[1,5-a]quinoxaline derivatives 2-18, obtained by introducing different substituents on either the 4-amino moiety (acyl or carbamoyl groups) or the 2-phenyl ring (4-OCH3) of previously reported 8-chloro-2-phenyl-1,2,
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::adc1d940ef661aa2a6177916d85959c8
http://hdl.handle.net/11568/203272
http://hdl.handle.net/11568/203272