Zobrazeno 1 - 7
of 7
pro vyhledávání: '"Chris Riviello"'
Autor:
Chris Riviello, Neeraj Gupta
Publikováno v:
Visual Journal of Emergency Medicine. 29:101435
Publikováno v:
Visual Journal of Emergency Medicine. 22:100955
Autor:
Jack Pick, Mark Craighead, Heather A. Zanetakos, Jeffrey J. Letourneau, Rachel Milne, Hema Desai, Leigh Campbell-Wan, Jeremy Presland, Michael Ohlmeyer, James R. Baker, Nasrin Ansari, Ray Jui-Hsiang Chan, Cliona P MacSweeney, Douglas S. Auld, Maria L. Webb, Jiuqiao Zhao, Chris Riviello, J. Richard Morphy, Stuart A. Best, Irina Neagu, Susan Elizabeth Napier, Koc-Kan Ho
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 21:3813-3817
Synthesis and structure–activity relationships (SAR) of a novel series of vasopressin V1b antagonists are described. 2-(6-Aminomethylaryl-2-aryl-4-oxo-quinazolin-3(4H)-yl)acetamide have been identified with low nanomolar affinity for the V1b recept
Autor:
Maria L. Webb, Jeffrey J. Letourneau, Michael Ohlmeyer, Hong Li, Biji Jacob, Jinqi Liu, Kenneth C. Appell, Angela Wong, Shalini Bansal, Chris Riviello, Yajing Rong
Publikováno v:
Bioorganic & Medicinal Chemistry Letters. 19:352-355
The discovery, synthesis and preliminary SAR of a novel class of non-peptidic antagonists of the alpha(v)-integrins alpha(v)beta(3) and alpha(v)beta(5) is described. High-throughput screening of an extensive series of ECLiPStrade mark compound librar
Autor:
Jiuqiao Zhao, Gé S.F. Ruigt, J. Richard Morphy, Mark Craighead, Maria L. Webb, Susan Elizabeth Napier, Chris Riviello, Jeffrey J. Letourneau, Irina Neagu, Rachel Milne, Ard Peeters, Heather A. Zanetakos, Michael Ohlmeyer, Fiona Thomson, Koc-Kan Ho, Leigh Campbell-Wan, Cliona P MacSweeney, Katharine A. Goan, Douglas S. Auld, Jeremy Presland, Stuart A. Best, Jui-Hsiang Chan, Nasrin Ansari, James R. Baker, Ellen G.J. Hulskotte, Hema Desai
Publikováno v:
Bioorganicmedicinal chemistry letters. 21(6)
Synthesis and structure-activity relationships (SAR) of a novel series of vasopressin V(1b) (V(3)) antagonists are described. 2-(4-Oxo-2-aryl-quinazolin-3(4H)-yl)acetamides have been identified with low nanomolar affinity for the V(1b) receptor and g
Autor:
Jeffrey J, Letourneau, Jinqi, Liu, Michael H J, Ohlmeyer, Chris, Riviello, Yajing, Rong, Hong, Li, Kenneth C, Appell, Shalini, Bansal, Biji, Jacob, Angela, Wong, Maria L, Webb
Publikováno v:
Bioorganicmedicinal chemistry letters. 19(2)
The discovery, synthesis and preliminary SAR of a novel class of non-peptidic antagonists of the alpha(v)-integrins alpha(v)beta(3) and alpha(v)beta(5) is described. High-throughput screening of an extensive series of ECLiPStrade mark compound librar
Autor:
John Wityak, Kan Ho, James Wen, Rosemary Zhang, Jack Baldwin, John H. Dodd, Alaric J. Dyckman, Katerina Leftheris, John Hynes, Wei Li, Shuqun Lin, Arthur M. Doweyko, John S. Sack, David J. Shuster, Kevin J. Moriarty, Ran Chan, Zahid Hussain, Joel C. Barrish, Gulzar Ahmed, Gary L. Schieven, Derek Loo, Kim W. McIntyre, Hong Wu, Ding Ren Shen, Maria L. Webb, Chris Riviello, Stephen T. Wrobleski, David J. Diller, Axel Metzger, Steve Kanner, Yvonne Shimshock, Madhuri Desai, Junjun Wu, Jeffrey J. Letourneau, Ian Henderson, Kathleen M. Gillooly, Tsung H. Lin, Sidney Pitt
Publikováno v:
Journal of medicinal chemistry. 47(25)
A new structural class of triaminotriazine aniline amides possessing potent p38 enzyme activity has been discovered. The initial hit (compound 1a) was identified through screening the Pharmacopeia ECLiPS compound collection. SAR modification led to t