Zobrazeno 1 - 10
of 24
pro vyhledávání: '"Chinmay Bhat"'
Autor:
Lien Moreels, Chinmay Bhat, Manuela Voráčová, Steve Peigneur, Hannah Goovaerts, Eero Mäki-Lohiluoma, Farrah Zahed, Luis A Pardo, Jari Yli-Kauhaluoma, Paula Kiuru, Jan Tytgat
Publikováno v:
PLoS ONE, Vol 12, Iss 12, p e0188811 (2017)
In the search for novel anticancer drugs, the potassium channel KV10.1 has emerged as an interesting cancer target. Here, we report a new group of KV10.1 inhibitors, namely the purpurealidin analogs. These alkaloids are produced by the Verongida spon
Externí odkaz:
https://doaj.org/article/e0035199f2d84432b06632e4aaa95559
Synthesis and Antiproliferative Activity of Marine Bromotyrosine Purpurealidin I and Its Derivatives
Autor:
Chinmay Bhat, Polina Ilina, Irene Tilli, Manuela Voráčová, Tanja Bruun, Victoria Barba, Nives Hribernik, Katja-Emilia Lillsunde, Eero Mäki-Lohiluoma, Tobias Rüffer, Heinrich Lang, Jari Yli-Kauhaluoma, Paula Kiuru, Päivi Tammela
Publikováno v:
Marine Drugs, Vol 16, Iss 12, p 481 (2018)
The first total synthesis of the marine bromotyrosine purpurealidin I (1) using trifluoroacetoxy protection group and its dimethylated analog (29) is reported along with 16 simplified bromotyrosine derivatives lacking the tyramine moiety. Their cytot
Externí odkaz:
https://doaj.org/article/5ec4018648f742feb9c4639468dbe4a4
Publikováno v:
Journal of Food Science and Technology. 55:2087-2094
Staphylococcus sciuri is an emerging human pathogen widely found in dairy industries. In this study, we have isolated methicillin resistant Staphylococcus sp. from biofilm formed on utensil used in the dairy society situated at Raia, Goa and was desi
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5ec28edd07d40c59eaa50731794d37b7
https://doi.org/10.1007/s13197-018-3123-0
https://doi.org/10.1007/s13197-018-3123-0
Publikováno v:
ChemistrySelect. 1:1723-1728
An unprecedented, green protocol for the combinatorial synthesis of 3-arylideneaminoquinazolin-4(1H)-ones is explored by a ‘solvent assisted grinding’ reaction of o-aminobenzhydrazide and aldehydes/ketones. The present methodology found special u
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::9d65e89e56c5eea6945d60a0719fd754
https://doi.org/10.1002/slct.201600362
https://doi.org/10.1002/slct.201600362
Synthesis and Antiproliferative Activity of Marine Bromotyrosine Purpurealidin I and Its Derivatives
Autor:
Manuela Voráčová, Katja-Emilia Lillsunde, Polina Ilina, Irene Tilli, Eero Mäki-Lohiluoma, Heinrich Lang, Tanja Bruun, Chinmay Bhat, Nives Hribernik, Jari Yli-Kauhaluoma, Victoria Barba, Paula Kiuru, Päivi Tammela, Tobias Rüffer
Publikováno v:
Marine Drugs
Volume 16
Issue 12
Marine Drugs, Vol 16, Iss 12, p 481 (2018)
Volume 16
Issue 12
Marine Drugs, Vol 16, Iss 12, p 481 (2018)
The first total synthesis of the marine bromotyrosine purpurealidin I (1) using trifluoroacetoxy protection group and its dimethylated analog (29) is reported along with 16 simplified bromotyrosine derivatives lacking the tyramine moiety. Their cytot
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::942966a64060bbbf6aa6b7faff788a02
Autor:
Chinmay Bhat
Publikováno v:
ChemistryOpen
Awarding Institute: Goa University (India) Date awarded: December, 2013 Supervisor: Prof. Santosh G. Tilve, HOD Chemistry, Goa University, Goa (India)
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::13d590210650ac3452313eb705a247b2
https://doi.org/10.1002/open.201402128
https://doi.org/10.1002/open.201402128
Autor:
Amit Kumar, Chinmay Bhat
Publikováno v:
Asian Journal of Organic Chemistry. 4:102-115
This Focus Review discusses the synthesis of an important member of the kainoid family; allokainic acid. The members of the kainoid family have attracted worldwide attention since their first isolation in 1953 due to their vast and potential medicina
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::43c8ee7ef5ad651daf702ba8d7c82d0a
https://doi.org/10.1002/ajoc.201402250
https://doi.org/10.1002/ajoc.201402250
Publikováno v:
Archives of microbiology. 199(10)
Listeria monocytogenes are Gram-positive well-known emerging food-borne pathogens causing listeriosis in humans. In the present study, we have isolated biofilm-forming Listeria sp. from utensils used by a local milk collection dairy society at Usgao
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::116f491cb2919d1cd6aad704f3fbb6e7
https://pubmed.ncbi.nlm.nih.gov/28762063
https://pubmed.ncbi.nlm.nih.gov/28762063
Publikováno v:
Synthesis. 46:2551-2573
Conhydrine is a naturally occurring 2-substituted piperidine alkaloid from the plant Conium maculatum L that exists in four different forms and is known for its high toxicity. This article focuses on the synthesis of conhydrine as its medicinal appli
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::828e82afa447158b2b1615f74ddd2a30
https://doi.org/10.1055/s-0034-1379023
https://doi.org/10.1055/s-0034-1379023
Autor:
Chinmay Bhat, Santosh G. Tilve
Publikováno v:
Tetrahedron. 69:10876-10883
A new diastereoselective pathway for the total synthesis of (+)-dexoxadrol, first asymmetric synthesis of (−)-epi-dexoxadrol and formal synthesis of conhydrine and (+)-lentiginosine is presented using commercially available (−)-pipecolinic acid.
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::a1428455e04832c794cbc7850af71fdd
https://doi.org/10.1016/j.tet.2013.10.082
https://doi.org/10.1016/j.tet.2013.10.082