Secosteroid thiosemicarbazides and secosteroid-1,2,4-triazoles as antiproliferative agents targeting breast cancer cells: Synthesis and biological evaluation.

Autor: Ilovaisky AI; N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, Leninsky prospect 47, Moscow 119991, Russia., Scherbakov AM; N.N. Blokhin National Medical Research Center of Oncology, Kashirskoye shosse 24, Moscow 115522, Russia., Chernoburova EI; N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, Leninsky prospect 47, Moscow 119991, Russia., Povarov AA; N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, Leninsky prospect 47, Moscow 119991, Russia., Shchetinina MA; N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, Leninsky prospect 47, Moscow 119991, Russia., Merkulova VM; N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, Leninsky prospect 47, Moscow 119991, Russia., Salnikova DI; N.N. Blokhin National Medical Research Center of Oncology, Kashirskoye shosse 24, Moscow 115522, Russia., Sorokin DV; N.N. Blokhin National Medical Research Center of Oncology, Kashirskoye shosse 24, Moscow 115522, Russia., Bozhenko EI; N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, Leninsky prospect 47, Moscow 119991, Russia., Zavarzin IV; N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, Leninsky prospect 47, Moscow 119991, Russia., Terent'ev AO; N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, Leninsky prospect 47, Moscow 119991, Russia. Electronic address: alterex@yandex.ru.

Publikováno v: The Journal of steroid biochemistry and molecular biology [J Steroid Biochem Mol Biol] 2023 Nov; Vol. 234, pp. 106386. Date of Electronic Publication: 2023 Sep 02.

Synthesis and evaluation of avermectin-imidazo[1,2-a]pyridine hybrids as potent GABA A receptor modulators.

Autor: Volkova YA; N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky prosp., 119991 Moscow, Russia. Electronic address: yavolkova@ioc.ac.ru., Rassokhina IV; N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky prosp., 119991 Moscow, Russia., Kondrakhin EA; V. V. Zakusov Institute of Pharmacology, Russian Academy of Sciences, 8 Baltiyskaya str., 125315 Moscow, Russia., Rossokhin AV; Research Center of Neurology, 5 by-str. Obukha, 105064 Moscow, Russia., Kolbaev SN; Research Center of Neurology, 5 by-str. Obukha, 105064 Moscow, Russia., Tihonova TB; N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky prosp., 119991 Moscow, Russia., Kh Dzhafarov M; Moscow State Academy of Veterinary Medicine and Biotechnology - MVA by K.I. Skryabin, 23 Academician Skryabin str., 109472 Moscow, Russia., Schetinina MA; N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky prosp., 119991 Moscow, Russia., Chernoburova EI; N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky prosp., 119991 Moscow, Russia., Vasileva EV; V. V. Zakusov Institute of Pharmacology, Russian Academy of Sciences, 8 Baltiyskaya str., 125315 Moscow, Russia., Dmitrenok AS; N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky prosp., 119991 Moscow, Russia., Kovalev GI; V. V. Zakusov Institute of Pharmacology, Russian Academy of Sciences, 8 Baltiyskaya str., 125315 Moscow, Russia., Sharonova IN; Research Center of Neurology, 5 by-str. Obukha, 105064 Moscow, Russia., Zavarzin IV; N. D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky prosp., 119991 Moscow, Russia.

Publikováno v: Bioorganic chemistry [Bioorg Chem] 2022 Oct; Vol. 127, pp. 105904. Date of Electronic Publication: 2022 Jun 03.

Novel steroidal 1,3,4-thiadiazines: Synthesis and biological evaluation in androgen receptor-positive prostate cancer 22Rv1 cells.

Autor: Komendantova AS; N.D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky Prosp., 119991 Moscow, Russia., Scherbakov AM; Department of Experimental Tumor Biology, N.N. Blokhin National Medical Research Center of Oncology, 24 Kashirskoe Shosse, 115522 Moscow, Russia. Electronic address: alex.scherbakov@gmail.com., Komkov AV; N.D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky Prosp., 119991 Moscow, Russia., Chertkova VV; N.D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky Prosp., 119991 Moscow, Russia., Gudovanniy AO; N.D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky Prosp., 119991 Moscow, Russia., Chernoburova EI; N.D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky Prosp., 119991 Moscow, Russia., Sorokin DV; Department of Experimental Tumor Biology, N.N. Blokhin National Medical Research Center of Oncology, 24 Kashirskoe Shosse, 115522 Moscow, Russia., Dzichenka YU; Institute of Bioorganic Chemistry of NAS of Belarus, Laboratory of Protein Engineering, Academician V.F. Kuprevich Str. 5/2, Minsk, Belarus., Shirinian VZ; N.D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky Prosp., 119991 Moscow, Russia., Volkova YA; N.D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky Prosp., 119991 Moscow, Russia. Electronic address: yavolkova@gmail.com., Zavarzin IV; N.D. Zelinsky Institute of Organic Chemistry, Russian Academy of Sciences, 47 Leninsky Prosp., 119991 Moscow, Russia.

Publikováno v: Bioorganic chemistry [Bioorg Chem] 2019 Oct; Vol. 91, pp. 103142. Date of Electronic Publication: 2019 Jul 23.

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