Zobrazeno 1 - 5
of 5
pro vyhledávání: '"Chantal Fouchet"'
Autor:
Bruno Loillier, Pierre Bélichard, Chantal Fouchet, Jean Luc Paquet, Jean-Michel Luccarini, Pierre Dodey, Evelyne Defrêne, Claude Robert, Didier Pruneau, Rose-Marie Franck, Béatrice Cremers, Hervé Duclos
Publikováno v:
Immunopharmacology. 43:187-194
LF 16-0687 (1-[[2,4-dichloro-3-[[(2,4-dimethylquinolin-8-yl)oxy] methyl]phenyl]sulfonyl]-N-[3-[[4-(aminoimethyl) phenyl] carbonylamino]propyl]-2(S)-pyrrolidinecarboxamide) has been selected from a large-scale medicinal chemistry program for further d
Autor:
Pierre Bélichard, Didier Pruneau, Bruno Loillier, Evelyne Defrêne, Béatrice Cremers, Claude Robert, Chantal Fouchet, Jean-Luc Paquet, Jean-Michel Luccarini
Publikováno v:
British Journal of Pharmacology. 126:1083-1090
The present study addresses the differences in binding profiles and functional properties of the human and rat bradykinin (BK) B2 receptor using various kinin receptor peptide derivatives as well as the non-peptide receptor antagonists WIN 64338 (pho
Autor:
Chantal Fouchet, Evelyne Defrêne, Rose-Marie Franck, Jean-Michel Luccarini, Didier Pruneau, Pierre Bélichard, Béatrice Cremers, Claude Robert, Jean-Luc Paquet, Bruno Loillier, Hervé Duclos
Publikováno v:
Fundamental & Clinical Pharmacology. 13:75-83
Activation of the kinin-kallikrein system and stimulation of bradykinin (BK) B2 receptors are thought to play an important role in the pathophysiology of inflammation and pain. In the present study, we report the pharmacological properties of a novel
Autor:
Jean-Luc Paquet, Jean-Michel Luccarini, Evelyne Defrêne, Chantal Fouchet, Hervé Duclos, Béatrice Cremers, Claude Robert, Didier Pruneau, Pierre Bélichard, Bruno Loillier, Rose-Marie Franck
Publikováno v:
British Journal of Pharmacology. 125:365-372
1. In the present paper, we describe the in vitro pharmacological properties of LF 16.0335 (1-[[3-[(2,4-dimethylquinolin-8-yl)oxymethyl]-2,4-dichloro-p henyl]sulphonyl] -2(S) - [[4 -[4-(aminoiminomethyl)phenylcarbonyl]piperazin-1-yl]ca rbonyl]pyrroli
Autor:
P. Bélichard, Jean-Michel Luccarini, Evelyne Defrêne, P. Dodey, Muriel Amblard, D. Pruneau, I. Daffix, Rose-Marie Franck, Chantal Fouchet, J.-L. Paquet, Gilbert Bergé, José Luis Martínez
Publikováno v:
Scopus-Elsevier
The synthesis and pharmacological evaluation of dimer derivatives of the C-terminal fragments of the potent bradykinin antagonist HOE-140, linked through their N-termini, were performed. The influence of peptide moiety length was studied using the su