Zobrazeno 1 - 10
of 12
pro vyhledávání: '"Chantal Devin"'
Autor:
Annie Heitz, Michèle Cristau, Chantal Devin, Jean-Alain Fehrentz, Jean Martinez, Anne-Marie Artis-Noel, Nicole Bernad
Publikováno v:
Journal of Peptide Science. 5:176-184
Bombesin pseudo-peptide analogues containing a hydroxamide function on the C-terminal part of the molecule, e.g. H-D-Phe-Gln-Trp-Ala-Val-Gly-His-Leu-NHOBzl 1 and H-D-Phe-Gln-Trp-Ala-Val-Gly-His-Leu-NHOH 2 were synthesized. These compounds were tested
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::7d6a67be0827b51b7126052ce5f4a1eb
https://doi.org/10.1002/(sici)1099-1387(199904)5:4<176::aid-psc189>3.0.co
https://doi.org/10.1002/(sici)1099-1387(199904)5:4<176::aid-psc189>3.0.co
Autor:
M Llinares, Chantal Devin, Nicole Bernad, J Azay, José Luis Martínez, Jean-Alain Fehrentz, A. M. Noel-Artis, Olivier Chaloin
Publikováno v:
The Journal of Peptide Research. 53:275-283
Bombesin receptor antagonists are potential therapeutic agents due to their ability to act as inhibitors of cellular proliferation. On the basis of our hypothesis concerning the mechanism of action of gastrin associating an activating enzyme to the r
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::ae42c4c97feb821a7cbbd1d9d66e3563
https://doi.org/10.1034/j.1399-3011.1999.00028.x
https://doi.org/10.1034/j.1399-3011.1999.00028.x
Autor:
Patrick Garrouste, J.‐C. Califano, Albert Loffet, Chantal Devin, Jean Martinez, F. Winternitz, Francois Rieunier, Olivier Chaloin, M Llinares, Ana-Christina Lima-Leite, Jean-Alain Fehrentz, Jean Vizavonna, E. Bourdel
Publikováno v:
Tetrahedron Letters. 35:1557-1560
The synthesis of chiral N-protected tetramic acid derivatives which are important precursors of β-hydroxy γ-amino acid under mild conditions is described. Reaction of urethane-N-carboxyanhydrides (UNCAs) with Meldrum's acid in the presence of a ter
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::dde72966dd65f5551b18bebb9444a514
https://doi.org/10.1016/s0040-4039(00)76757-8
https://doi.org/10.1016/s0040-4039(00)76757-8
Autor:
Chantal Devin, Albert Loffet, M Llinares, Jean Martinez, F. Winternitz, Patrick Garrouste, Ana-Christina Lima-Leite, E. Bourdel, Olivier Chaloin, Jean-Alain Fehrentz, Jean Vizavonna, J.‐C. Califano, Francois Rieunier
Publikováno v:
ChemInform. 25
The synthesis of chiral N-protected tetramic acid derivatives which are important precursors of β-hydroxy γ-amino acid under mild conditions is described. Reaction of urethane-N-carboxyanhydrides (UNCAs) with Meldrum's acid in the presence of a ter
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::d424536bf472a5c606335f9ae129b236
https://doi.org/10.1002/chin.199430206
https://doi.org/10.1002/chin.199430206
Autor:
Chantal Devin, Julie Pannequin, Nicole Bernad, Michèle Cristau, Jean-Alain Fehrentz, Jean-Claude Galleyrand, Jean Martinez, Catherine Oiry
Publikováno v:
Peptides for the New Millennium ISBN: 0792364457
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::aa4d7bfba6b647d1939e56ba7279243d
https://doi.org/10.1007/0-306-46881-6_252
https://doi.org/10.1007/0-306-46881-6_252
Autor:
Francois Winternitz, José Luis Martínez, P. Chevallet, Chantal Devin, Marielle Paris, Jean-Alain Fehrentz, Catherine Pothion, A. Loffet
Publikováno v:
Chinese Peptide Symposia ISBN: 0792349636
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_________::195c1ab91d5c1913f623a0e1d29d62c9
https://doi.org/10.1007/0-306-46859-x_3
https://doi.org/10.1007/0-306-46859-x_3
Autor:
Julie Pannequin, Catherine Oiry, Anne-Marie Artis, Jean Martinez, Chantal Devin, Michèle Cristau, Jean-Claude Galleyrand, Nicole Bernad, Jean-Alain Fehrentz
Publikováno v:
European Journal of Pharmacology
European Journal of Pharmacology, Elsevier, 2000, 403, pp.17-25
HAL
European Journal of Pharmacology, Elsevier, 2000, 403, pp.17-25
HAL
alpha-amidation of a peptide (which takes place from a glycine-extended precursor) is required to produce biologically active amidated hormones, such as gastrin-releasing peptide (GRP)/Pyr-Gln-Arg-Leu-Gly-Asn-Gln-Trp-Ala-Val-Gly-His-Leu-Met-NH(2) (bo
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a30aa39fcf6841de2fe0f7e695871b56
https://pubmed.ncbi.nlm.nih.gov/10969139
https://pubmed.ncbi.nlm.nih.gov/10969139
Autor:
Olivier Chaloin, Michèle Cristau, Nicole Bernad, Jean Martinez, Annie Heitz, Muriel Amblard, Jean-Alain Fehrentz, Chantal Devin, Catherine Oiry
Publikováno v:
Journal of Medicinal Chemistry
Journal of Medicinal Chemistry, American Chemical Society, 2000, 43 (12), pp.2356-2361. ⟨10.1021/jm990942i⟩
Journal of Medicinal Chemistry, American Chemical Society, 2000, 43 (12), pp.2356-2361. ⟨10.1021/jm990942i⟩
Analogues of bombesin which incorporate dipeptide or turn mimetics have been synthesized. One of them (compound 11) containing a seven-membered lactam ring revealed a good affinity for GRP/BN receptors on rat pancreatic acini (K(i) value of 1.7 +/- 0
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::341ebf08f156a2107e1afa05372cdd9f
https://pubmed.ncbi.nlm.nih.gov/10882361
https://pubmed.ncbi.nlm.nih.gov/10882361
Autor:
M Llinares, C. Nagain, Chantal Devin, Jean-Alain Fehrentz, Claude Rozé, J Azay, José Luis Martínez, Nicole Bernad
Publikováno v:
Peptides / Peptides (Fayetteville)
Peptides / Peptides (Fayetteville), 1998, 19 (1), pp.57-63
Peptides / Peptides (Fayetteville), 1998, 19 (1), pp.57-63
Azay, J., C. Nagain, M. Llinares, C. Devin, J. A. Fehrentz, N. Bernad, C. Roze and J. Martinez. Comparative study of in vitro and vivo activities of bombesin pseudopeptide analogs modified on the C-terminal dipeptide fragment. Peptides 19(1) 57–63,
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d9a3a02ce7317eaa363e94cc0ee49a4c
https://hal.archives-ouvertes.fr/hal-00357478
https://hal.archives-ouvertes.fr/hal-00357478
Publikováno v:
European Journal of Medicinal Chemistry
European Journal of Medicinal Chemistry, Elsevier, 1997, 32, pp.767-780
European Journal of Medicinal Chemistry, Elsevier, 1997, 32, pp.767-780
Summary Bombesin receptor antagonists are possible therapeutic agents due to their ability to act as inhibitors of cellular proliferation. On the basis of our hypothesis on the mechanism of action of gastrin associating an activating enzyme system to
Externí odkaz:
https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8f08b10f4a660ea8c7f8a41d351bed1c
https://hal.archives-ouvertes.fr/hal-00357447
https://hal.archives-ouvertes.fr/hal-00357447